IL77661A - Process for the preparation of 4,4-azetidinones,and novel intermediates thereof - Google Patents

Process for the preparation of 4,4-azetidinones,and novel intermediates thereof

Info

Publication number
IL77661A
IL77661A IL77661A IL7766186A IL77661A IL 77661 A IL77661 A IL 77661A IL 77661 A IL77661 A IL 77661A IL 7766186 A IL7766186 A IL 7766186A IL 77661 A IL77661 A IL 77661A
Authority
IL
Israel
Prior art keywords
azetidinones
preparation
novel intermediates
intermediates
novel
Prior art date
Application number
IL77661A
Other languages
English (en)
Original Assignee
Squibb & Sons Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Squibb & Sons Inc filed Critical Squibb & Sons Inc
Publication of IL77661A publication Critical patent/IL77661A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D205/00—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom
    • C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
    • C07D205/06—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member
    • C07D205/08—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams
    • C07D205/085—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having one double bond between ring members or between a ring member and a non-ring member with one oxygen atom directly attached in position 2, e.g. beta-lactams with a nitrogen atom directly attached in position 3
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D213/00—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members
    • C07D213/02—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members
    • C07D213/04—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D213/06—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom
    • C07D213/16—Heterocyclic compounds containing six-membered rings, not condensed with other rings, with one nitrogen atom as the only ring hetero atom and three or more double bonds between ring members or between ring members and non-ring members having three double bonds between ring members or between ring members and non-ring members having no bond between the ring nitrogen atom and a non-ring member or having only hydrogen or carbon atoms directly attached to the ring nitrogen atom containing only hydrogen and carbon atoms in addition to the ring nitrogen atom containing only one pyridine ring
    • C07D213/18—Salts thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Cephalosporin Compounds (AREA)
  • Pyridine Compounds (AREA)
  • Pyrane Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
IL77661A 1985-01-28 1986-01-21 Process for the preparation of 4,4-azetidinones,and novel intermediates thereof IL77661A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US06/695,775 US4638061A (en) 1985-01-28 1985-01-28 [3S(Z)]-2-[[[1-(2-amino-4-thiazolyl)-2-[[2,2-dimethyl-4-oxo-1-(sulfooxy)-3-azetidinyl]amino]-2-oxoethylidene]-amino]oxy] acetic acid and intermediate

Publications (1)

Publication Number Publication Date
IL77661A true IL77661A (en) 1989-06-30

Family

ID=24794413

Family Applications (1)

Application Number Title Priority Date Filing Date
IL77661A IL77661A (en) 1985-01-28 1986-01-21 Process for the preparation of 4,4-azetidinones,and novel intermediates thereof

Country Status (35)

Country Link
US (1) US4638061A (ja)
JP (2) JPH0780840B2 (ja)
KR (1) KR900000675B1 (ja)
CN (1) CN1014894B (ja)
AR (1) AR242024A1 (ja)
AT (1) AT389511B (ja)
AU (1) AU588017B2 (ja)
BE (1) BE904121A (ja)
CA (2) CA1283924C (ja)
CH (3) CH667872A5 (ja)
CS (1) CS253740B2 (ja)
DD (3) DD248592A5 (ja)
DE (1) DE3602347A1 (ja)
DK (1) DK39486A (ja)
EG (1) EG17682A (ja)
ES (3) ES8706112A1 (ja)
FI (1) FI85022C (ja)
FR (1) FR2576596B1 (ja)
GB (2) GB2170201B (ja)
GR (1) GR860239B (ja)
HU (1) HU196367B (ja)
IE (2) IE59629B1 (ja)
IL (1) IL77661A (ja)
IT (1) IT1190604B (ja)
LU (1) LU86262A1 (ja)
NL (1) NL8600136A (ja)
NO (1) NO170014C (ja)
NZ (1) NZ214836A (ja)
PH (3) PH22425A (ja)
PL (3) PL149156B1 (ja)
PT (1) PT81914B (ja)
RO (1) RO93483B (ja)
SE (3) SE467824B (ja)
YU (2) YU45760B (ja)
ZA (1) ZA86302B (ja)

Families Citing this family (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4751220A (en) * 1986-12-19 1988-06-14 E. R. Squibb & Sons, Inc. Crystalline salts of [3S(Z)]-2[[[1-(2-amino-4-thiazolyl)-2-[[2,2-dimethyl-4-oxo-1-(sulfooxy)-3-azetidinyl]amino]-2-oxoethylidene]-amino]oxy]acetic acid
US5143913A (en) * 1988-04-04 1992-09-01 E. R. Squibb & Sons, Inc. [3S(Z)]-3-[[(2-amino-4-thiazolyl)[[2-(hydroxyamino)-2-oxoethoxy]imino]acetyl]amino]-2,2-dimethyl-4-oxo-1-azetidinyl sulfate
JPH01290674A (ja) * 1988-04-04 1989-11-22 E R Squibb & Sons Inc アゼチジニル誘導体
US4973747A (en) * 1989-08-15 1990-11-27 E. R. Squibb & Sons, Inc. Process for preparing 3-hydroxy 2-keto acids
CA2783572C (en) * 2005-12-07 2016-08-09 Basilea Pharmaceutica Ag Useful combinations of monobactam antibiotics with beta-lactamase inhibitors
WO2017180794A1 (en) 2016-04-13 2017-10-19 Skyline Antiinfectives, Inc. Deuterated o-sulfated beta-lactam hydroxamic acids and deuterated n-sulfated beta-lactams

Family Cites Families (5)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4337197A (en) * 1980-10-31 1982-06-29 E. R. Squibb & Sons, Inc. O-sulfated β-lactam hydroxamic acids and intermediates
JPS58113174A (ja) * 1981-12-26 1983-07-05 Toyama Chem Co Ltd 新規なアゼチジン誘導体またはその塩類を含有する抗菌剤
JPS58194856A (ja) * 1982-05-10 1983-11-12 Yamanouchi Pharmaceut Co Ltd 新規２−アゼチジノン誘導体
JPS58206589A (ja) * 1982-05-26 1983-12-01 Yamanouchi Pharmaceut Co Ltd ２−アゼチジノン誘導体
US4565654A (en) * 1983-03-28 1986-01-21 University Of Notre Dame Du Lac N-Acyloxy monocyclic β-lactams

Also Published As

Publication number Publication date
GB8800425D0 (en) 1988-02-10
IE860205L (en) 1986-07-28
FR2576596A1 (fr) 1986-08-01
FI860247A (fi) 1986-07-29
YU167087A (en) 1988-04-30
ATA20386A (de) 1989-05-15
SE467824B (sv) 1992-09-21
ES8800897A1 (es) 1987-12-01
PL262317A1 (en) 1987-09-07
RO93483B (ro) 1988-01-01
SE8600355L (sv) 1986-07-29
RO93483A (ro) 1987-12-31
FI85022C (fi) 1992-02-25
PL262318A1 (en) 1987-09-07
NO170014C (no) 1992-09-02
SE8600355D0 (sv) 1986-01-27
HUT40407A (en) 1986-12-28
NO170014B (no) 1992-05-25
AR242024A1 (es) 1993-02-26
SE9002338L (sv) 1990-07-03
CN1014894B (zh) 1991-11-27
CA1279322C (en) 1991-01-22
EG17682A (en) 1990-10-30
DE3602347A1 (de) 1986-07-31
GB2170201B (en) 1989-01-11
PH23084A (en) 1989-04-10
SE9002337D0 (sv) 1990-07-03
DD241600A5 (de) 1986-12-17
PL257668A1 (en) 1987-03-09
CA1283924C (en) 1991-05-07
NZ214836A (en) 1988-10-28
CH667872A5 (fr) 1988-11-15
PL149156B1 (en) 1990-01-31
PH22425A (en) 1988-09-12
CN86100736A (zh) 1986-10-22
GB2198133B (en) 1989-01-11
CH670825A5 (ja) 1989-07-14
SE9002337L (sv) 1990-07-03
KR860005812A (ko) 1986-08-13
ES8706112A1 (es) 1987-06-01
PH23093A (en) 1989-04-10
JPH0780840B2 (ja) 1995-08-30
NL8600136A (nl) 1986-08-18
PT81914A (en) 1986-02-01
CH670824A5 (ja) 1989-07-14
AU588017B2 (en) 1989-09-07
SE9002338D0 (sv) 1990-07-03
ZA86302B (en) 1986-08-27
GB2198133A (en) 1988-06-08
ES8801917A1 (es) 1988-03-01
CS253740B2 (en) 1987-12-17
SE502442C2 (sv) 1995-10-16
DD248584A5 (de) 1987-08-12
YU45760B (sh) 1992-07-20
KR900000675B1 (ko) 1990-02-02
NO860273L (no) 1986-07-29
ES557056A0 (es) 1987-12-01
LU86262A1 (fr) 1986-08-04
FR2576596B1 (fr) 1989-12-15
IT8619206A0 (it) 1986-01-28
GR860239B (en) 1986-05-28
DK39486A (da) 1986-07-29
IT1190604B (it) 1988-02-16
HU196367B (en) 1988-11-28
ES551252A0 (es) 1987-06-01
PT81914B (pt) 1987-11-30
AU5246086A (en) 1986-07-31
AT389511B (de) 1989-12-27
IE930750L (en) 1986-07-28
SE468896B (sv) 1993-04-05
JPS61176563A (ja) 1986-08-08
FI860247A0 (fi) 1986-01-20
JPH0853404A (ja) 1996-02-27
BE904121A (fr) 1986-05-15
FI85022B (fi) 1991-11-15
US4638061A (en) 1987-01-20
GB2170201A (en) 1986-07-30
DK39486D0 (da) 1986-01-27
IE59629B1 (en) 1994-03-09
YU5886A (en) 1988-02-29
DD248592A5 (de) 1987-08-12
ES557057A0 (es) 1988-03-01

Similar Documents

Publication Publication Date Title
PT82226A (en) Process for the preparation of 3-aryluraciles and pesticeides therewith
IL71274A (en) Process and intermediates for the preparation of 1alpha,25-dihydroxyergocalciffrol
HU900192D0 (en) Process for preparation of 1,1,1-trifluor-2-aryl-prop-2-ene-oxides
DE3662256D1 (en) Process for the preparation of (2,2)-paracyclophane
IL92681A0 (en) Process and intermediates for the preparation of 4-phenylpiperidines
DE3569375D1 (en) Process for the preparation of 1,2-benzisothiazolones
ZA862747B (en) Intermediates for the production of epipodophyilotoxin and related compounds and processes for the preparation and use thereof
EP0194144A3 (en) Process for the preparation of 2-alkyl-cyclopent-2-enones
IL80305A (en) Process for the preparation of ypsilon-butyrolactams and some novel intermediates
IL77661A (en) Process for the preparation of 4,4-azetidinones,and novel intermediates thereof
EP0206147A3 (en) Process for the preparation of 4,4'-dinitrodibenzyls
GB2180237B (en) Process for the preparation of n-sulfamyl-3-(2-guanidino-thiazol-4-yl-methylthio)-propionamidine
PT83799A (en) Process for the preparation of novel 2,2:-bi-1h-imidazoles
DE3660590D1 (en) Process for the preparation of 2-alkyl-cyclopentanones
DE3660623D1 (en) Process for the preparation of 2-methyl-2-alkenals
GB2176479B (en) Process for the preparation of 2-bromo-a-ergocryptine
PT85023A (en) Process for the preparation of substituted 2-phenylacetil-1,3,5-cyclohexanetriones and of intermediates
PH22955A (en) Process for the preparation of aromatic 1,4-oxazepinones and intermediates thereof
EP0190994A3 (en) Process for the preparation of 1-amino-2-bromo-4-hydroxyanthraquinone
EP0198795A3 (en) Process for the preparation of 1,4-diaminoanthraquinones
EP0190101A3 (en) Process for the preparation of n-alkyl-anilines
ZA861025B (en) Process for the preparation of thiocyanatomethylthiobenzothiazoles
PT83637A (en) Process for the preparation of antidepressant 5-heterocyclic-2,4-dialkyl-3h-1,2,4-triazole-3-thiones
EP0206293A3 (en) Process for the preparation of 3,5-dichloro-2-pyridone
DE3662784D1 (en) Process for the preparation of 1,3,6,8-tetrabromopyrene

Legal Events

Date Code Title Description
KB Patent renewed
RH Patent void