IL32836A - Benzothiazine 1,1-dioxides and their preparation - Google Patents

Benzothiazine 1,1-dioxides and their preparation

Info

Publication number
IL32836A
IL32836A IL32836A IL3283669A IL32836A IL 32836 A IL32836 A IL 32836A IL 32836 A IL32836 A IL 32836A IL 3283669 A IL3283669 A IL 3283669A IL 32836 A IL32836 A IL 32836A
Authority
IL
Israel
Prior art keywords
dioxide
oxo
dihydro
benzothiazine
methyl
Prior art date
Application number
IL32836A
Other languages
English (en)
Other versions
IL32836A0 (en
Original Assignee
Pfizer
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Pfizer filed Critical Pfizer
Publication of IL32836A0 publication Critical patent/IL32836A0/xx
Publication of IL32836A publication Critical patent/IL32836A/en

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
    • A61K31/5415—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame ortho- or peri-condensed with carbocyclic ring systems, e.g. phenothiazine, chlorpromazine, piroxicam
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines
IL32836A 1968-08-27 1969-08-15 Benzothiazine 1,1-dioxides and their preparation IL32836A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
US76759468A 1968-08-27 1968-08-27

Publications (2)

Publication Number Publication Date
IL32836A0 IL32836A0 (en) 1969-11-12
IL32836A true IL32836A (en) 1972-08-30

Family

ID=25079964

Family Applications (1)

Application Number Title Priority Date Filing Date
IL32836A IL32836A (en) 1968-08-27 1969-08-15 Benzothiazine 1,1-dioxides and their preparation

Country Status (18)

Country Link
US (1) US3591584A (ja)
JP (2) JPS50677B1 (ja)
AT (2) AT298503B (ja)
BE (1) BE737962A (ja)
BR (1) BR6911817D0 (ja)
CH (1) CH520705A (ja)
DE (2) DE1943265C3 (ja)
DK (1) DK145297C (ja)
ES (1) ES370861A1 (ja)
FI (1) FI51189C (ja)
FR (1) FR2016455B1 (ja)
GB (1) GB1257180A (ja)
IL (1) IL32836A (ja)
MY (1) MY7300310A (ja)
NL (1) NL157013B (ja)
NO (1) NO129746B (ja)
PH (1) PH10029A (ja)
SE (2) SE373854B (ja)

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JPS59179683U (ja) * 1983-05-19 1984-11-30 寺田毛織株式会社 貼り合わせふとん
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DE3437232A1 (de) * 1984-10-10 1986-04-17 Mack Chem Pharm Stabilisierte injektionsloesungen von piroxicam
US4582831A (en) * 1984-11-16 1986-04-15 Pfizer Inc. Anti-inflammatory polymorphic monoethanolamine salt of N-(2-pyridyl)-2-methyl-4-hydroxy-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxide compound, composition, and method of use therefor
CH663899A5 (fr) * 1985-03-20 1988-01-29 Nestle Sa Procede pour la preparation d'une composition a base d'un principe actif de faible hydrosolubilite finement divise.
US4623486A (en) * 1985-05-29 1986-11-18 Pfizer Inc. [4-substituted benzoyloxy]-N-substituted-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides having anti-arthritic activity
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US4829062A (en) * 1986-05-16 1989-05-09 Pfizer Inc. Benzothiazine dioxide derivatives
ATE66477T1 (de) * 1986-08-29 1991-09-15 Pfizer 2-guanidino-4-aryl-thiazole fuer die behandlung von peptischen geschwueren.
US5196410A (en) * 1986-10-31 1993-03-23 Pfizer Inc. Transdermal flux enhancing compositions
WO1988009793A1 (en) * 1987-06-10 1988-12-15 Pfizer Inc. 3,4-DIHYDRO-2-ALKYL-3-OXO-N-ARYL-2H-[1]BENZOTHIENO[3,2-e]-1,2-THIAZINE-4-CARBOXAMIDE-1,1-DIOXIDES
US5081118A (en) * 1987-10-26 1992-01-14 Pfizer Inc. Benzothiazine dioxide derivatives
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JPH0717589B2 (ja) * 1990-01-22 1995-03-01 ファイザー製薬株式会社 新規１，３―ジカルボニル化合物およびその組成物
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JP2964195B2 (ja) * 1992-04-28 1999-10-18 エスエス製薬株式会社 ピロキシカム錠及びその製造法
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IT1318673B1 (it) * 2000-08-08 2003-08-27 Nicox Sa Farmaci per le disfunzioni sessuali.
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Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE1302858B (ja) * 1962-09-21 1972-05-04

Also Published As

Publication number Publication date
SE402459B (sv) 1978-07-03
FI51189B (ja) 1976-08-02
SE373854B (ja) 1975-02-17
IL32836A0 (en) 1969-11-12
BE737962A (ja) 1970-02-26
DK145297C (da) 1983-03-14
FR2016455A1 (ja) 1970-05-08
DE1943265C3 (de) 1982-02-04
DK145297B (da) 1982-10-25
MY7300310A (en) 1973-12-31
JPS50677B1 (ja) 1975-01-10
DE1967325C2 (de) 1982-03-18
BR6911817D0 (pt) 1973-02-13
AT298503B (de) 1972-05-10
US3591584A (en) 1971-07-06
DE1967325B2 (de) 1981-08-13
AT294113B (de) 1971-11-10
FR2016455B1 (ja) 1974-02-01
DE1943265B2 (de) 1981-05-14
NL6912981A (ja) 1970-03-03
NL157013B (nl) 1978-06-15
NO129746B (ja) 1974-05-20
JPS5142114B1 (ja) 1976-11-13
PH10029A (en) 1976-07-13
CH520705A (fr) 1972-03-31
ES370861A1 (es) 1971-07-01
FI51189C (fi) 1976-11-10
GB1257180A (ja) 1971-12-15
DE1943265A1 (de) 1970-08-13

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