IL237749A - A process for the preparation of phenyl and pyridyl pyrolidines is conserved - Google Patents

A process for the preparation of phenyl and pyridyl pyrolidines is conserved

Info

Publication number
IL237749A
IL237749A IL237749A IL23774915A IL237749A IL 237749 A IL237749 A IL 237749A IL 237749 A IL237749 A IL 237749A IL 23774915 A IL23774915 A IL 23774915A IL 237749 A IL237749 A IL 237749A
Authority
IL
Israel
Prior art keywords
formula
compounds
iii
alkyl
above mentioned
Prior art date
Application number
IL237749A
Other languages
English (en)
Hebrew (he)
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of IL237749A publication Critical patent/IL237749A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/02—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to acyclic carbon atoms
    • C07C317/10—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/14—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/16—Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C317/18—Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton with sulfone or sulfoxide groups bound to acyclic carbon atoms of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/01—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton
    • C07C323/02—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton having sulfur atoms of thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/07—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton having sulfur atoms of thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/10—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C323/11—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/16—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pyrrole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
IL237749A 2012-09-27 2015-03-16 A process for the preparation of phenyl and pyridyl pyrolidines is conserved IL237749A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12186243 2012-09-27
PCT/EP2013/069919 WO2014048958A1 (en) 2012-09-27 2013-09-25 Process for the preparation of optionally substituted phenyl and pyridyl pyrrolidines

Publications (1)

Publication Number Publication Date
IL237749A true IL237749A (en) 2017-09-28

Family

ID=47044827

Family Applications (1)

Application Number Title Priority Date Filing Date
IL237749A IL237749A (en) 2012-09-27 2015-03-16 A process for the preparation of phenyl and pyridyl pyrolidines is conserved

Country Status (13)

Country Link
US (1) US9447036B2 (Direct)
EP (1) EP2900634B1 (Direct)
JP (1) JP6251749B2 (Direct)
KR (1) KR20150059778A (Direct)
CN (1) CN104619683B (Direct)
BR (1) BR112015006825A2 (Direct)
DK (1) DK2900634T3 (Direct)
ES (1) ES2625547T3 (Direct)
IL (1) IL237749A (Direct)
IN (1) IN2015DN02542A (Direct)
MX (1) MX350575B (Direct)
TW (1) TWI601713B (Direct)
WO (1) WO2014048958A1 (Direct)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JP7058719B2 (ja) * 2017-08-09 2022-04-22 アークサーダ・アー・ゲー ４－（ヘプタフルオロ－２－プロピル）アニリン類の調製方法

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US4092349A (en) 1976-11-10 1978-05-30 Pfizer Inc. 11-Desoxy-15-thiaprostaglandins
US4173463A (en) 1978-10-31 1979-11-06 Shell Oil Company Phosphonium salts as herbicides
EP0393424B1 (de) 1989-04-17 1995-09-27 Bayer Ag Verfahren zur Herstellung von 2,7-Diazabicyclo(3.3.0)octanen
IT1274021B (it) 1994-02-28 1997-07-14 Italfarmaco Spa Diesteri dell'acido carbonico ad attivita' antivirale ed antinfiammatoria
ES2180811T3 (es) 1995-11-23 2003-02-16 Rhodia Chimie Sa Procedimiento para la perfluoro-alquilacion y reaccionante para poner en practica dicho procedimiento.
AU4064597A (en) * 1996-08-16 1998-03-06 Du Pont Pharmaceuticals Company Amidinophenyl-pyrrolidines, -pyrrolines, and -isoxazolidines and derivatives thereof
PL372246A1 (en) 2002-05-28 2005-07-11 3-Dimensional Pharmaceuticals, Inc. Novel thiophene amidines, compositions thereof, and methods of treating complement-mediated diseases and conditions
US7230119B2 (en) 2004-08-25 2007-06-12 Biocryst Pharmaceuticals, Inc. Process for the preparation of substituted pyrrolidine derivatives and intermediates
US7521427B2 (en) 2004-11-09 2009-04-21 Georgia Tech Research Corporation Peptidyl allyl sulfones
AR057032A1 (es) 2005-05-27 2007-11-14 Wyeth Corp Tigeciclina y metodos de preparacion
US20080234280A1 (en) 2005-08-01 2008-09-25 Mcmurray Gordon Use of Mc4 Receptor Agonist Compounds
US7750167B2 (en) 2006-07-05 2010-07-06 N.V. Organon Process for the preparation of asenapine and intermediate products used in said process
JP5164510B2 (ja) * 2006-10-06 2013-03-21 日本曹達株式会社 含窒素複素環化合物および有害生物防除剤
GB0623209D0 (en) 2006-11-21 2007-01-03 F2G Ltd Antifungal agents
WO2008129811A1 (ja) 2007-03-23 2008-10-30 Panasonic Corporation 無線送信装置及び無線受信装置
JP2010116389A (ja) 2008-10-17 2010-05-27 Bayer Cropscience Ag 殺虫性アリールピロリジン類
JP2008266230A (ja) 2007-04-23 2008-11-06 Bayer Cropscience Ag 殺虫性アリールピロリジン類
MX2010007404A (es) 2008-01-04 2010-10-05 Organon Nv Procedimiento para la preparacion de asenapina y productos intermediarios utilizados en dicho procedimiento.
CZ305085B6 (cs) 2008-03-14 2015-04-29 Zentiva, K.S. Způsob přípravy dabigatranu
TW201038580A (en) 2009-02-02 2010-11-01 Pfizer 4-amino-5-oxo-7,8-dihydropyrimido[5,4-f][1,4]oxazepin-6(5H)-yl)phenyl derivatives
JP5746981B2 (ja) 2009-02-27 2015-07-08 アムビト ビオスシエンセス コルポラチオン Ｊａｋキナーゼ調節キナゾリン誘導体、及びその使用方法
CN102414175A (zh) 2009-04-30 2012-04-11 拜耳作物科学公司 杀虫的芳基吡咯烷
RU2542103C2 (ru) * 2009-05-22 2015-02-20 Эббви Инк. Модуляторы рецепторов 5-нт и способы их применения
RU2012105122A (ru) 2009-07-16 2013-08-27 Байер Кропсайенс Аг Способ получения хиральных производных 3-триазолилсульфоксида
JP2011136928A (ja) 2009-12-28 2011-07-14 Bayer Cropscience Ag 殺虫性アリールピロリジン類
JP2012082186A (ja) 2010-09-15 2012-04-26 Bayer Cropscience Ag 殺虫性アリールピロリジン類
EP2892902A1 (en) * 2012-09-07 2015-07-15 Zoetis LLC Spirocyclic derivatives as antiparasitic agents

Also Published As

Publication number Publication date
US20150246880A1 (en) 2015-09-03
TWI601713B (zh) 2017-10-11
US9447036B2 (en) 2016-09-20
EP2900634B1 (en) 2017-02-22
EP2900634A1 (en) 2015-08-05
DK2900634T3 (en) 2017-05-22
JP6251749B2 (ja) 2017-12-20
TW201418215A (zh) 2014-05-16
KR20150059778A (ko) 2015-06-02
CN104619683A (zh) 2015-05-13
BR112015006825A2 (pt) 2017-08-08
WO2014048958A1 (en) 2014-04-03
MX350575B (es) 2017-09-11
ES2625547T3 (es) 2017-07-19
MX2015003902A (es) 2015-07-17
CN104619683B (zh) 2017-05-10
JP2015535835A (ja) 2015-12-17
IN2015DN02542A (Direct) 2015-09-11

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