IN2015DN02542A - - Google Patents

Info

Publication number
IN2015DN02542A
IN2015DN02542A IN2542DEN2015A IN2015DN02542A IN 2015DN02542 A IN2015DN02542 A IN 2015DN02542A IN 2542DEN2015 A IN2542DEN2015 A IN 2542DEN2015A IN 2015DN02542 A IN2015DN02542 A IN 2015DN02542A
Authority
IN
India
Prior art keywords
preparation
pyrrolidines
pyridyl
optionally substituted
substituted aryl
Prior art date
Application number
Inventor
Friedrich August Mühlthau
Mark James Ford
Original Assignee
Bayer Cropscience Ag
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Bayer Cropscience Ag filed Critical Bayer Cropscience Ag
Publication of IN2015DN02542A publication Critical patent/IN2015DN02542A/en

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
    • C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/02—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to acyclic carbon atoms
    • C07C317/10—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to acyclic carbon atoms of an unsaturated carbon skeleton containing rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/14—Sulfones; Sulfoxides having sulfone or sulfoxide groups bound to carbon atoms of six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/16—Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C317/18—Sulfones; Sulfoxides having sulfone or sulfoxide groups and singly-bound oxygen atoms bound to the same carbon skeleton with sulfone or sulfoxide groups bound to acyclic carbon atoms of the carbon skeleton
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/01—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton
    • C07C323/02—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton having sulfur atoms of thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/07—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and halogen atoms, or nitro or nitroso groups bound to the same carbon skeleton having sulfur atoms of thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/10—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton
    • C07C323/11—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/16—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and singly-bound oxygen atoms bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton the carbon skeleton containing six-membered aromatic rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F7/00—Compounds containing elements of Groups 4 or 14 of the Periodic Table
    • C07F7/02—Silicon compounds
    • C07F7/08—Compounds having one or more C—Si linkages
    • C07F7/0803—Compounds with Si-C or Si-Si linkages
    • C07F7/081—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te
    • C07F7/0812—Compounds with Si-C or Si-Si linkages comprising at least one atom selected from the elements N, O, halogen, S, Se or Te comprising a heterocyclic ring

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Pyrrole Compounds (AREA)

Abstract

The present invention relates to a method for the preparation of optionally substituted aryl and pyridyl pyrrolidines which are useful intermediates for the preparation of certain biologically active compounds.
IN2542DEN2015 2012-09-27 2013-09-25 IN2015DN02542A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP12186243 2012-09-27
PCT/EP2013/069919 WO2014048958A1 (en) 2012-09-27 2013-09-25 Process for the preparation of optionally substituted phenyl and pyridyl pyrrolidines

Publications (1)

Publication Number Publication Date
IN2015DN02542A true IN2015DN02542A (en) 2015-09-11

Family

ID=47044827

Family Applications (1)

Application Number Title Priority Date Filing Date
IN2542DEN2015 IN2015DN02542A (en) 2012-09-27 2013-09-25

Country Status (13)

Country Link
US (1) US9447036B2 (en)
EP (1) EP2900634B1 (en)
JP (1) JP6251749B2 (en)
KR (1) KR20150059778A (en)
CN (1) CN104619683B (en)
BR (1) BR112015006825A2 (en)
DK (1) DK2900634T3 (en)
ES (1) ES2625547T3 (en)
IL (1) IL237749A (en)
IN (1) IN2015DN02542A (en)
MX (1) MX350575B (en)
TW (1) TWI601713B (en)
WO (1) WO2014048958A1 (en)

Families Citing this family (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US10882816B2 (en) * 2017-08-09 2021-01-05 Lonza Ltd Method for the preparation of 4-(heptafluoro-2-propyl) anilines

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US4092349A (en) 1976-11-10 1978-05-30 Pfizer Inc. 11-Desoxy-15-thiaprostaglandins
US4173463A (en) 1978-10-31 1979-11-06 Shell Oil Company Phosphonium salts as herbicides
EP0393424B1 (en) 1989-04-17 1995-09-27 Bayer Ag Process for the preparation of 2,7-Diazabicyclo(3.3.O)octanes
IT1274021B (en) 1994-02-28 1997-07-14 Italfarmaco Spa DIFFERENCES OF CARBONIC ACID WITH ANTI-VIRAL AND ANTI-INFLAMMATORY ACTIVITY
AU7699196A (en) 1995-11-23 1997-06-11 Rhodia Chimie Perfluoroalkylation method and reagent therefor
JP2000516234A (en) * 1996-08-16 2000-12-05 デュポン ファーマシューティカルズ カンパニー Amidinophenyl-pyrrolidines, amidinophenyl-pyrrolines, and amidinophenyl-isoxazolidines and derivatives thereof
JP2005538953A (en) 2002-05-28 2005-12-22 ３−ディメンショナル ファーマシューティカルズ， インコーポレイテッド Novel thiophenamidines, compositions thereof, and methods of treating complement-mediated diseases and conditions
US7230119B2 (en) 2004-08-25 2007-06-12 Biocryst Pharmaceuticals, Inc. Process for the preparation of substituted pyrrolidine derivatives and intermediates
US7521427B2 (en) 2004-11-09 2009-04-21 Georgia Tech Research Corporation Peptidyl allyl sulfones
AR057032A1 (en) 2005-05-27 2007-11-14 Wyeth Corp TIGECICLINE AND PREPARATION METHODS
EP1928460A2 (en) 2005-08-01 2008-06-11 Pfizer Limited Mc4r-agonists for the treatment of urinary tract dysfunction
US7750167B2 (en) 2006-07-05 2010-07-06 N.V. Organon Process for the preparation of asenapine and intermediate products used in said process
JP5164510B2 (en) * 2006-10-06 2013-03-21 日本曹達株式会社 Nitrogen-containing heterocyclic compounds and pest control agents
GB0623209D0 (en) 2006-11-21 2007-01-03 F2G Ltd Antifungal agents
WO2008129811A1 (en) 2007-03-23 2008-10-30 Panasonic Corporation Radio transmission device and radio reception device
JP2008266230A (en) 2007-04-23 2008-11-06 Bayer Cropscience Ag Insecticidal arylpyrrolidines
JP2010116389A (en) 2008-10-17 2010-05-27 Bayer Cropscience Ag Insecticidal arylpyrrolidines
CA2710800A1 (en) 2008-01-04 2009-07-16 N.V. Organon Process for the preparation of asenapine and intermediate products used in said process
CZ305085B6 (en) 2008-03-14 2015-04-29 Zentiva, K.S. Process for preparing dabigatran
WO2010086820A1 (en) 2009-02-02 2010-08-05 Pfizer Inc. 4-amino-5-oxo-7, 8-dihydropyrimido [5,4-f] [1,4] oxazepin-6 (5h) -yl) phenyl derivatives, pharmaceutical compositions and uses thereof
SI2401267T1 (en) 2009-02-27 2014-05-30 Ambit Biosciences Corporation Jak kinase modulating quinazoline derivatives and their use in methods
WO2010124845A1 (en) 2009-04-30 2010-11-04 Bayer Cropscience Ag Pesticidal arylpyrrolidines
RU2014147175A (en) * 2009-05-22 2015-06-27 Эббви Инк. 5-NT RECEPTOR MODULATORS AND WAYS OF THEIR APPLICATION
EP2454242B1 (en) 2009-07-16 2014-10-15 Bayer CropScience AG Method for producing chiral 3-triazolyl-sulfoxide derivatives
JP2011136928A (en) 2009-12-28 2011-07-14 Bayer Cropscience Ag Insecticidal arylpyrrolidines
JP2012082186A (en) 2010-09-15 2012-04-26 Bayer Cropscience Ag Insecticidal arylpyrrolidines
CN104603139B (en) * 2012-09-07 2016-12-07 硕腾服务有限责任公司 Spirocyclic derivatives as antiparasitic

Also Published As

Publication number Publication date
WO2014048958A1 (en) 2014-04-03
ES2625547T3 (en) 2017-07-19
DK2900634T3 (en) 2017-05-22
CN104619683B (en) 2017-05-10
US20150246880A1 (en) 2015-09-03
JP2015535835A (en) 2015-12-17
EP2900634A1 (en) 2015-08-05
US9447036B2 (en) 2016-09-20
EP2900634B1 (en) 2017-02-22
MX350575B (en) 2017-09-11
MX2015003902A (en) 2015-07-17
CN104619683A (en) 2015-05-13
BR112015006825A2 (en) 2017-08-08
TW201418215A (en) 2014-05-16
JP6251749B2 (en) 2017-12-20
TWI601713B (en) 2017-10-11
IL237749A (en) 2017-09-28
KR20150059778A (en) 2015-06-02

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