IL148558A0 - Amphiphilic prodrugs - Google Patents

Amphiphilic prodrugs

Info

Publication number
IL148558A0
IL148558A0 IL14855800A IL14855800A IL148558A0 IL 148558 A0 IL148558 A0 IL 148558A0 IL 14855800 A IL14855800 A IL 14855800A IL 14855800 A IL14855800 A IL 14855800A IL 148558 A0 IL148558 A0 IL 148558A0
Authority
IL
Israel
Prior art keywords
amphiphilic prodrugs
amphiphilic
prodrugs
Prior art date
Application number
IL14855800A
Other languages
English (en)
Original Assignee
Nobex Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nobex Corp filed Critical Nobex Corp
Publication of IL148558A0 publication Critical patent/IL148558A0/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/59—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
    • A61K47/60—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes the organic macromolecular compound being a polyoxyalkylene oligomer, polymer or dendrimer, e.g. PEG, PPG, PEO or polyglycerol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
IL14855800A 1999-09-13 2000-09-07 Amphiphilic prodrugs IL148558A0 (en)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US15364999P 1999-09-13 1999-09-13
US09/474,915 US6713454B1 (en) 1999-09-13 1999-12-31 Prodrugs of etoposide and etoposide analogs
PCT/US2000/024520 WO2001019406A2 (en) 1999-09-13 2000-09-07 Amphiphilic prodrugs

Publications (1)

Publication Number Publication Date
IL148558A0 true IL148558A0 (en) 2002-09-12

Family

ID=26850733

Family Applications (1)

Application Number Title Priority Date Filing Date
IL14855800A IL148558A0 (en) 1999-09-13 2000-09-07 Amphiphilic prodrugs

Country Status (17)

Country Link
US (3) US6713454B1 (US06713454-20040330-C00009.png)
EP (1) EP1212099A2 (US06713454-20040330-C00009.png)
JP (1) JP2003509385A (US06713454-20040330-C00009.png)
KR (1) KR20020059398A (US06713454-20040330-C00009.png)
CN (1) CN1390143A (US06713454-20040330-C00009.png)
AU (1) AU7575600A (US06713454-20040330-C00009.png)
BR (1) BR0013948A (US06713454-20040330-C00009.png)
CA (1) CA2384645A1 (US06713454-20040330-C00009.png)
CZ (1) CZ2002928A3 (US06713454-20040330-C00009.png)
HU (1) HUP0204110A3 (US06713454-20040330-C00009.png)
IL (1) IL148558A0 (US06713454-20040330-C00009.png)
MX (1) MXPA02002712A (US06713454-20040330-C00009.png)
NO (1) NO20021213L (US06713454-20040330-C00009.png)
NZ (1) NZ517681A (US06713454-20040330-C00009.png)
PL (1) PL354261A1 (US06713454-20040330-C00009.png)
RU (1) RU2002109595A (US06713454-20040330-C00009.png)
WO (1) WO2001019406A2 (US06713454-20040330-C00009.png)

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Also Published As

Publication number Publication date
AU7575600A (en) 2001-04-17
EP1212099A2 (en) 2002-06-12
HUP0204110A3 (en) 2003-08-28
US20040180840A1 (en) 2004-09-16
CN1390143A (zh) 2003-01-08
MXPA02002712A (es) 2003-10-14
NZ517681A (en) 2004-01-30
CA2384645A1 (en) 2001-03-22
RU2002109595A (ru) 2003-11-27
JP2003509385A (ja) 2003-03-11
US20040253206A1 (en) 2004-12-16
HUP0204110A2 (hu) 2003-04-28
BR0013948A (pt) 2002-05-14
KR20020059398A (ko) 2002-07-12
NO20021213D0 (no) 2002-03-12
WO2001019406A2 (en) 2001-03-22
US7119074B2 (en) 2006-10-10
US6713454B1 (en) 2004-03-30
NO20021213L (no) 2002-05-13
WO2001019406A3 (en) 2002-01-17
PL354261A1 (en) 2003-12-29
CZ2002928A3 (cs) 2002-09-11

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