NO20021213L - Amfifile prodroger - Google Patents

Amfifile prodroger

Info

Publication number
NO20021213L
NO20021213L NO20021213A NO20021213A NO20021213L NO 20021213 L NO20021213 L NO 20021213L NO 20021213 A NO20021213 A NO 20021213A NO 20021213 A NO20021213 A NO 20021213A NO 20021213 L NO20021213 L NO 20021213L
Authority
NO
Norway
Prior art keywords
amphiphilic prodrugs
amphiphilic
prodrugs
Prior art date
Application number
NO20021213A
Other languages
English (en)
Other versions
NO20021213D0 (no
Inventor
Nnochiri N Ekwuribe
Tatyana A Dyakonov
Christopher H Price
Original Assignee
Nobex Corp
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Nobex Corp filed Critical Nobex Corp
Publication of NO20021213D0 publication Critical patent/NO20021213D0/no
Publication of NO20021213L publication Critical patent/NO20021213L/no

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K47/00—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient
    • A61K47/50—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates
    • A61K47/51—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent
    • A61K47/56—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule
    • A61K47/59—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes
    • A61K47/60—Medicinal preparations characterised by the non-active ingredients used, e.g. carriers or inert additives; Targeting or modifying agents chemically bound to the active ingredient the non-active ingredient being chemically bound to the active ingredient, e.g. polymer-drug conjugates the non-active ingredient being a modifying agent the modifying agent being an organic macromolecular compound, e.g. an oligomeric, polymeric or dendrimeric molecule obtained otherwise than by reactions only involving carbon-to-carbon unsaturated bonds, e.g. polyureas or polyurethanes the organic macromolecular compound being a polyoxyalkylene oligomer, polymer or dendrimer, e.g. PEG, PPG, PEO or polyglycerol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/04—Antineoplastic agents specific for metastasis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00

Landscapes

  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Epidemiology (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Coloring Foods And Improving Nutritive Qualities (AREA)
NO20021213A 1999-09-13 2002-03-12 Amfifile prodroger NO20021213L (no)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US15364999P 1999-09-13 1999-09-13
US09/474,915 US6713454B1 (en) 1999-09-13 1999-12-31 Prodrugs of etoposide and etoposide analogs
PCT/US2000/024520 WO2001019406A2 (en) 1999-09-13 2000-09-07 Amphiphilic prodrugs

Publications (2)

Publication Number Publication Date
NO20021213D0 NO20021213D0 (no) 2002-03-12
NO20021213L true NO20021213L (no) 2002-05-13

Family

ID=26850733

Family Applications (1)

Application Number Title Priority Date Filing Date
NO20021213A NO20021213L (no) 1999-09-13 2002-03-12 Amfifile prodroger

Country Status (17)

Country Link
US (3) US6713454B1 (no)
EP (1) EP1212099A2 (no)
JP (1) JP2003509385A (no)
KR (1) KR20020059398A (no)
CN (1) CN1390143A (no)
AU (1) AU7575600A (no)
BR (1) BR0013948A (no)
CA (1) CA2384645A1 (no)
CZ (1) CZ2002928A3 (no)
HU (1) HUP0204110A3 (no)
IL (1) IL148558A0 (no)
MX (1) MXPA02002712A (no)
NO (1) NO20021213L (no)
NZ (1) NZ517681A (no)
PL (1) PL354261A1 (no)
RU (1) RU2002109595A (no)
WO (1) WO2001019406A2 (no)

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US6541508B2 (en) * 1999-09-13 2003-04-01 Nobex Corporation Taxane prodrugs
US6713454B1 (en) * 1999-09-13 2004-03-30 Nobex Corporation Prodrugs of etoposide and etoposide analogs
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Also Published As

Publication number Publication date
WO2001019406A2 (en) 2001-03-22
CA2384645A1 (en) 2001-03-22
EP1212099A2 (en) 2002-06-12
US20040180840A1 (en) 2004-09-16
BR0013948A (pt) 2002-05-14
IL148558A0 (en) 2002-09-12
US20040253206A1 (en) 2004-12-16
PL354261A1 (en) 2003-12-29
MXPA02002712A (es) 2003-10-14
HUP0204110A3 (en) 2003-08-28
AU7575600A (en) 2001-04-17
US7119074B2 (en) 2006-10-10
HUP0204110A2 (hu) 2003-04-28
WO2001019406A3 (en) 2002-01-17
NZ517681A (en) 2004-01-30
CZ2002928A3 (cs) 2002-09-11
NO20021213D0 (no) 2002-03-12
RU2002109595A (ru) 2003-11-27
KR20020059398A (ko) 2002-07-12
CN1390143A (zh) 2003-01-08
US6713454B1 (en) 2004-03-30
JP2003509385A (ja) 2003-03-11

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