IL129018A0 - 1H-pyrido (3,4-b) indole-4-carboxamide derivatives their preparation and application thereof in therapeutics - Google Patents

1H-pyrido (3,4-b) indole-4-carboxamide derivatives their preparation and application thereof in therapeutics

Info

Publication number
IL129018A0
IL129018A0 IL12901897A IL12901897A IL129018A0 IL 129018 A0 IL129018 A0 IL 129018A0 IL 12901897 A IL12901897 A IL 12901897A IL 12901897 A IL12901897 A IL 12901897A IL 129018 A0 IL129018 A0 IL 129018A0
Authority
IL
Israel
Prior art keywords
pyrido
therapeutics
indole
preparation
application
Prior art date
Application number
IL12901897A
Other languages
English (en)
Original Assignee
Synthelabo
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Synthelabo filed Critical Synthelabo
Publication of IL129018A0 publication Critical patent/IL129018A0/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/04—Ortho-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/08—Antiepileptics; Anticonvulsants
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/14—Drugs for disorders of the nervous system for treating abnormal movements, e.g. chorea, dyskinesia
    • A61P25/16—Anti-Parkinson drugs
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/20—Hypnotics; Sedatives
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/30—Drugs for disorders of the nervous system for treating abuse or dependence

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Neurosurgery (AREA)
  • Engineering & Computer Science (AREA)
  • Biomedical Technology (AREA)
  • Public Health (AREA)
  • Neurology (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Psychology (AREA)
  • Addiction (AREA)
  • Psychiatry (AREA)
  • Anesthesiology (AREA)
  • Pain & Pain Management (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Indole Compounds (AREA)
IL12901897A 1996-10-08 1997-10-03 1H-pyrido (3,4-b) indole-4-carboxamide derivatives their preparation and application thereof in therapeutics IL129018A0 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
FR9612229A FR2754262B1 (fr) 1996-10-08 1996-10-08 Derives de 1h-pyrido[3,4-b]indole-4-carboxamide, leur preparation et leur application en therapeutique
PCT/FR1997/001750 WO1998015552A1 (fr) 1996-10-08 1997-10-03 DERIVES DE 1H-PYRIDO[3,4-b]INDOLE-4-CARBOXAMIDE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE

Publications (1)

Publication Number Publication Date
IL129018A0 true IL129018A0 (en) 2000-02-17

Family

ID=9496449

Family Applications (1)

Application Number Title Priority Date Filing Date
IL12901897A IL129018A0 (en) 1996-10-08 1997-10-03 1H-pyrido (3,4-b) indole-4-carboxamide derivatives their preparation and application thereof in therapeutics

Country Status (33)

Country Link
US (1) US6075021A (ja)
EP (1) EP0934319B1 (ja)
JP (1) JP4227197B2 (ja)
KR (1) KR100488095B1 (ja)
CN (1) CN1089765C (ja)
AR (1) AR009112A1 (ja)
AT (1) ATE218567T1 (ja)
AU (1) AU721102B2 (ja)
BG (1) BG63751B1 (ja)
BR (1) BR9711879A (ja)
CA (1) CA2266376A1 (ja)
CO (1) CO4910141A1 (ja)
CY (1) CY2291B1 (ja)
CZ (1) CZ298906B6 (ja)
DE (1) DE69713124T2 (ja)
DK (1) DK0934319T3 (ja)
EE (1) EE03830B1 (ja)
ES (1) ES2178008T3 (ja)
FR (1) FR2754262B1 (ja)
HK (1) HK1023338A1 (ja)
HU (1) HUP9904623A3 (ja)
IL (1) IL129018A0 (ja)
NO (1) NO311938B1 (ja)
NZ (1) NZ334708A (ja)
PL (1) PL188244B1 (ja)
PT (1) PT934319E (ja)
RU (1) RU2180904C2 (ja)
SK (1) SK282970B6 (ja)
TR (1) TR199900712T2 (ja)
TW (1) TW461889B (ja)
UA (1) UA57037C2 (ja)
WO (1) WO1998015552A1 (ja)
ZA (1) ZA978970B (ja)

Families Citing this family (17)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2766823B1 (fr) 1997-07-30 1999-10-08 Synthelabo Derives de 4-oxo-3,5-dihydro-4h-pyridazino[4,5-b] indole-1-acetamide, leur preparation et leur application en therapeutique
FR2788776B1 (fr) * 1999-01-26 2001-02-23 Synthelabo Derives de 4-oxo-3, 5-dihydro-4h-pyridazino [4,5-b] indole-1 -carboxamide, leur preparation et leur application en therapeutique
FR2788696B1 (fr) * 1999-01-26 2004-03-05 Synthelabo Utilisation de derives de pyridazino [4,5-b] indole-1-acetamide pour la preparation de medicaments destines aux maladies du systeme nerveux central
FR2811897A1 (fr) * 2000-07-24 2002-01-25 Sanofi Synthelabo UTILISATION DE DERIVES DE PYRIDAZINO[4,5-b]INDOLE-1- ACETAMIDE POUR LA PREPARATION DE MEDICAMENTS DESTINES AU TRAITEMENT DES DYSFONCTIONNEMENTS DES RECEPTEURS DE TYPE PERIPHERIQUE AUX BENZODIAZEPINES
FR2811990A1 (fr) * 2000-07-24 2002-01-25 Sanofi Synthelabo DERIVES DE 1-(4-OXO-3,5-DIHYDRO-4H-PYRIDAZINO[4,5-b]INDOLE-1 -CARBONYL)PIPERAZINE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
FR2833953B1 (fr) * 2001-12-21 2004-12-03 Sanofi Synthelabo DERIVES DE 3-HETEROARYL-3,5-DIHYDRO-4-OXO-4H-PYRIDAZINO [4,5-b]INDOLE-1-CARBOXAMIDE, LEUR PREPARATION ET LEUR APPLICATION EN THERAPEUTIQUE
FR2838124B1 (fr) * 2002-04-03 2004-05-28 Sanofi Synthelabo Derives de 3-heteroaryl-3,5-dihydro-4-oxo-4h-pyridazino [4,5-b]indole-1-acetamide, leur preparation et leur application en therapeutique
PA8586801A1 (es) * 2002-10-31 2005-02-04 Pfizer Inhibidores de hiv-integrasa, composiciones farmaceuticas y metodos para su uso
BRPI0407052A (pt) * 2003-01-27 2006-01-17 Pfizer Inibidores da hiv-integrase, composições farmacêuticas, e métodos para sua utilização
WO2005103003A2 (en) * 2004-04-26 2005-11-03 Pfizer Inc. Pyrrolopyridine derivatives and their use as hiv-integrase inhibitors
CA2563761C (en) * 2004-04-26 2009-12-29 Pfizer Inc. Inhibitors of the hiv integrase enzyme
NZ562559A (en) * 2005-05-05 2011-03-31 Sanofi Aventis Us Llc Stable nanoparticle formulations smaller than 1000 nm without the use of any surface modifier or stabilizzer absorbed onto the surface of the particles
RS20080141A (en) * 2005-10-07 2009-07-15 Pfizer Products Inc., Inhibitors of the hiv integrase enzyme
UA95788C2 (en) 2005-12-15 2011-09-12 Ф. Хоффманн-Ля Рош Аг Fused pyrrole derivatives
KR101124070B1 (ko) * 2006-06-05 2012-04-12 제논 파마슈티칼스 인크. 유기 화합물
CN1946120B (zh) * 2006-10-20 2010-05-12 华为技术有限公司 实现话单关联的方法及系统
KR100688448B1 (ko) * 2006-12-06 2007-03-02 (주)경진건축사사무소 건축물 내부 조적구조

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2724384B1 (fr) * 1994-09-14 1999-04-16 Cemaf Nouveaux derives de la 3,4-dihydro beta-carboline agonistes de la melatonine, leur procede de preparation et leur utilisation a titre de medicament

Also Published As

Publication number Publication date
DE69713124D1 (de) 2002-07-11
PL188244B1 (pl) 2005-01-31
SK45199A3 (en) 2000-02-14
AU4559497A (en) 1998-05-05
HUP9904623A2 (hu) 2000-06-28
CN1089765C (zh) 2002-08-28
EE9900155A (et) 1999-12-15
NO311938B1 (no) 2002-02-18
SK282970B6 (sk) 2003-01-09
ES2178008T3 (es) 2002-12-16
EE03830B1 (et) 2002-08-15
BG103301A (en) 2000-05-31
ZA978970B (en) 1998-04-20
DK0934319T3 (da) 2002-09-30
AU721102B2 (en) 2000-06-22
FR2754262A1 (fr) 1998-04-10
JP2001508403A (ja) 2001-06-26
FR2754262B1 (fr) 1998-10-30
KR20000048992A (ko) 2000-07-25
CN1233248A (zh) 1999-10-27
CA2266376A1 (en) 1998-04-16
NO991624D0 (no) 1999-04-06
CZ119399A3 (cs) 1999-07-14
TW461889B (en) 2001-11-01
CY2291B1 (en) 2003-07-04
PT934319E (pt) 2002-10-31
CO4910141A1 (es) 2000-04-24
UA57037C2 (uk) 2003-06-16
TR199900712T2 (xx) 1999-06-21
CZ298906B6 (cs) 2008-03-12
WO1998015552A1 (fr) 1998-04-16
US6075021A (en) 2000-06-13
DE69713124T2 (de) 2003-01-30
HK1023338A1 (en) 2000-09-08
AR009112A1 (es) 2000-03-08
HUP9904623A3 (en) 2001-03-28
BG63751B1 (bg) 2002-11-29
EP0934319A1 (fr) 1999-08-11
NO991624L (no) 1999-06-07
EP0934319B1 (fr) 2002-06-05
ATE218567T1 (de) 2002-06-15
RU2180904C2 (ru) 2002-03-27
BR9711879A (pt) 1999-08-24
PL332643A1 (en) 1999-09-27
KR100488095B1 (ko) 2005-05-09
JP4227197B2 (ja) 2009-02-18
NZ334708A (en) 2000-10-27

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Legal Events

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KB Patent renewed
MM9K Patent not in force due to non-payment of renewal fees