IL114142A - Amidino sulphone derivatives their preparation pharmaceutical compositions containing them and their use - Google Patents

Amidino sulphone derivatives their preparation pharmaceutical compositions containing them and their use

Info

Publication number
IL114142A
IL114142A IL11414295A IL11414295A IL114142A IL 114142 A IL114142 A IL 114142A IL 11414295 A IL11414295 A IL 11414295A IL 11414295 A IL11414295 A IL 11414295A IL 114142 A IL114142 A IL 114142A
Authority
IL
Israel
Prior art keywords
amidino
pharmaceutical compositions
compositions containing
preparation pharmaceutical
sulphone derivatives
Prior art date
Application number
IL11414295A
Other languages
English (en)
Other versions
IL114142A0 (en
Original Assignee
Wellcome Found
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GBGB9509774.7A external-priority patent/GB9509774D0/en
Application filed by Wellcome Found filed Critical Wellcome Found
Publication of IL114142A0 publication Critical patent/IL114142A0/xx
Priority to IL12871799A priority Critical patent/IL128717A0/xx
Publication of IL114142A publication Critical patent/IL114142A/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C323/00—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups
    • C07C323/50—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton
    • C07C323/51—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton
    • C07C323/60—Thiols, sulfides, hydropolysulfides or polysulfides substituted by halogen, oxygen or nitrogen atoms, or by sulfur atoms not being part of thio groups containing thio groups and carboxyl groups bound to the same carbon skeleton having the sulfur atoms of the thio groups bound to acyclic carbon atoms of the carbon skeleton with the carbon atom of at least one of the carboxyl groups bound to nitrogen atoms
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07C—ACYCLIC OR CARBOCYCLIC COMPOUNDS
    • C07C317/00—Sulfones; Sulfoxides
    • C07C317/44—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton
    • C07C317/48—Sulfones; Sulfoxides having sulfone or sulfoxide groups and carboxyl groups bound to the same carbon skeleton the carbon skeleton being further substituted by singly-bound nitrogen atoms, not being part of nitro or nitroso groups
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Engineering & Computer Science (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Saccharide Compounds (AREA)
  • Immobilizing And Processing Of Enzymes And Microorganisms (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Hydrogenated Pyridines (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
  • Steroid Compounds (AREA)
IL11414295A 1994-06-15 1995-06-14 Amidino sulphone derivatives their preparation pharmaceutical compositions containing them and their use IL114142A (en)

Priority Applications (1)

Application Number Priority Date Filing Date Title
IL12871799A IL128717A0 (en) 1994-06-15 1999-02-25 Amino sulphone derivatives

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP94304314 1994-06-15
GBGB9509774.7A GB9509774D0 (en) 1995-05-15 1995-05-15 Enzyme inhibitors

Publications (2)

Publication Number Publication Date
IL114142A0 IL114142A0 (en) 1995-10-31
IL114142A true IL114142A (en) 2000-02-17

Family

ID=26137155

Family Applications (2)

Application Number Title Priority Date Filing Date
IL11414295A IL114142A (en) 1994-06-15 1995-06-14 Amidino sulphone derivatives their preparation pharmaceutical compositions containing them and their use
IL12871799A IL128717A0 (en) 1994-06-15 1999-02-25 Amino sulphone derivatives

Family Applications After (1)

Application Number Title Priority Date Filing Date
IL12871799A IL128717A0 (en) 1994-06-15 1999-02-25 Amino sulphone derivatives

Country Status (29)

Country Link
US (2) USRE39576E1 (xx)
EP (2) EP0957087B1 (xx)
JP (2) JP2989010B2 (xx)
KR (1) KR100430207B1 (xx)
CN (1) CN1070849C (xx)
AT (2) ATE191470T1 (xx)
AU (1) AU692892B2 (xx)
BR (1) BR9507995A (xx)
CA (1) CA2192668A1 (xx)
CY (2) CY2238B1 (xx)
DE (2) DE69529101T2 (xx)
DK (2) DK0765308T3 (xx)
ES (2) ES2189322T3 (xx)
FI (1) FI965019A (xx)
GR (1) GR3033746T3 (xx)
HK (1) HK1003935A1 (xx)
HU (1) HUT77407A (xx)
IL (2) IL114142A (xx)
IS (1) IS4384A (xx)
MX (1) MX9606136A (xx)
MY (1) MY115437A (xx)
NO (1) NO308655B1 (xx)
NZ (1) NZ289157A (xx)
PT (2) PT957087E (xx)
RU (1) RU2162841C2 (xx)
SI (2) SI0957087T1 (xx)
TW (1) TW442453B (xx)
WO (1) WO1995034534A1 (xx)
ZA (1) ZA954940B (xx)

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FR2740339B1 (fr) * 1995-10-26 1997-12-05 Oreal Utilisation d'au moins un inhibiteur de no-synthase dans le traitement des peaux sensibles
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US6620848B2 (en) 1997-01-13 2003-09-16 Smithkline Beecham Corporation Nitric oxide synthase inhibitors
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AU8647198A (en) * 1997-08-12 1999-03-01 Chugai Seiyaku Kabushiki Kaisha Remedies for diseases associated with bone resorption
DE69920670T2 (de) * 1998-03-11 2006-02-16 G.D. Searle & Co., Chicago Halogenierte aminosäure derivate als hemmstoffe der stickstoffmonoxid-synthase
US6534503B1 (en) 1998-04-28 2003-03-18 Lion Bioscience Ag Melanocortin receptor-3 ligands to treat sexual dysfunction
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US6284735B1 (en) * 1998-04-28 2001-09-04 Lion Bioscience Ag HP-3228 and related peptides to treat sexual dysfunction
GB9811599D0 (en) 1998-05-30 1998-07-29 Glaxo Group Ltd Nitric oxide synthase inhibitors
AU6605800A (en) * 1999-07-16 2001-02-05 Trega Biosciences, Inc. Melanocortin receptor-3 ligands to treat sexual dysfunction
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DE10111049A1 (de) * 2001-03-06 2002-09-12 Beiersdorf Ag Verwendung von Substanzen, die verhindern, daß die NO-Synthese des warmblütigen Organismus ihre Wirkung entfaltet, zur Herstellung von kosmetischen oder dermatologischen Zubereitungen, zur Prophylaxe und Behandlung von entzündlichen Hautzuständen und/oder zum Hautschutz bei empfindlich determinierter trockener Haut
DE10111050A1 (de) * 2001-03-06 2002-09-12 Beiersdorf Ag Verwendung von Substanzen, die verhindern, daß die NO-Synthase des warmblütigenOrganismus ihre Wirkung entfaltet, zur Herstellung von kosmetischewn oder dermatologischen Zubereitungen zur Behandlung und/oder Prophylaxe unerwünschter Hautpigmentierung
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DE4310202A1 (de) * 1992-03-30 1993-10-07 Ciba Geigy µ-Ketoimidoester als Stabilisatoren für chlorhaltige Polymerisate
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Also Published As

Publication number Publication date
NZ289157A (en) 1998-03-25
JP2000026402A (ja) 2000-01-25
MY115437A (en) 2003-06-30
JP3614711B2 (ja) 2005-01-26
CY2455B1 (en) 2005-06-03
SI0957087T1 (en) 2003-04-30
DE69529101T2 (de) 2003-11-13
TW442453B (en) 2001-06-23
AU2891795A (en) 1996-01-05
IL114142A0 (en) 1995-10-31
EP0765308B1 (en) 2000-04-05
CN1070849C (zh) 2001-09-12
USRE39576E1 (en) 2007-04-17
RU2162841C2 (ru) 2001-02-10
AU692892B2 (en) 1998-06-18
KR100430207B1 (ko) 2004-07-19
DK0765308T3 (da) 2000-09-11
SI0765308T1 (en) 2000-08-31
CA2192668A1 (en) 1995-12-21
HUT77407A (hu) 1998-04-28
MX9606136A (es) 1998-06-30
NO965379L (no) 1996-12-13
EP0957087B1 (en) 2002-12-04
ZA954940B (en) 1996-12-17
DK0957087T3 (da) 2003-03-24
CN1155276A (zh) 1997-07-23
US5889056A (en) 1999-03-30
DE69516141D1 (de) 2000-05-11
HK1003935A1 (en) 1998-11-13
ATE229001T1 (de) 2002-12-15
FI965019A0 (fi) 1996-12-13
FI965019A (fi) 1996-12-13
NO308655B1 (no) 2000-10-09
HU9603454D0 (en) 1997-02-28
PT957087E (pt) 2003-04-30
WO1995034534A1 (en) 1995-12-21
JPH10506371A (ja) 1998-06-23
IS4384A (is) 1996-11-13
DE69529101D1 (de) 2003-01-16
IL128717A0 (en) 2000-01-31
ATE191470T1 (de) 2000-04-15
BR9507995A (pt) 1997-08-05
GR3033746T3 (en) 2000-10-31
EP0957087A2 (en) 1999-11-17
EP0957087A3 (en) 2000-12-20
EP0765308A1 (en) 1997-04-02
ES2189322T3 (es) 2003-07-01
NO965379D0 (no) 1996-12-13
DE69516141T2 (de) 2000-10-19
ES2145282T3 (es) 2000-07-01
JP2989010B2 (ja) 1999-12-13
PT765308E (pt) 2000-09-29
CY2238B1 (en) 2003-07-04

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