PL2614058T3 - Polimorfy i sole n-[5-[4-(5-{[(2r,6s)-2,6-dimetylo-4-morfolinylo]-metylo}-1,3-oksazol-2-ilo)-1h-indazol-6-ilo]-2-(metyloksy)-3-pirydynylo]metanosulfonamidu - Google Patents
Polimorfy i sole n-[5-[4-(5-{[(2r,6s)-2,6-dimetylo-4-morfolinylo]-metylo}-1,3-oksazol-2-ilo)-1h-indazol-6-ilo]-2-(metyloksy)-3-pirydynylo]metanosulfonamiduInfo
- Publication number
- PL2614058T3 PL2614058T3 PL11755311T PL11755311T PL2614058T3 PL 2614058 T3 PL2614058 T3 PL 2614058T3 PL 11755311 T PL11755311 T PL 11755311T PL 11755311 T PL11755311 T PL 11755311T PL 2614058 T3 PL2614058 T3 PL 2614058T3
- Authority
- PL
- Poland
- Prior art keywords
- methyloxy
- indazol
- methanesulfonamide
- oxazol
- polymorphs
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US38074810P | 2010-09-08 | 2010-09-08 | |
EP11755311.5A EP2614058B1 (en) | 2010-09-08 | 2011-09-06 | POLYMORPHS AND SALTS OF N-[5-[4-(5-{[(2R,6S)-2,6-DIMETHYL-4-MORPHOLINYL]METHYL}-& xA;1,3-OXAZOL-2-YL)-1H-INDAZOL-6-YL]-2-(METHYLOXY)-3-PYRIDINYL]METHANESULFONAMIDE |
PCT/EP2011/065419 WO2012032067A1 (en) | 2010-09-08 | 2011-09-06 | Polymorphs and salts of n- [5- [4- (5- { [(2r,6s) -2, 6 - dimethyl - 4 -morpholinyl] methyl} - 1, 3 - oxazol - 2 - yl) - 1h- inda zol-6-yl] -2- (methyloxy) - 3 - pyridinyl] methanesulfonamide |
Publications (1)
Publication Number | Publication Date |
---|---|
PL2614058T3 true PL2614058T3 (pl) | 2015-12-31 |
Family
ID=44645691
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
PL11755311T PL2614058T3 (pl) | 2010-09-08 | 2011-09-06 | Polimorfy i sole n-[5-[4-(5-{[(2r,6s)-2,6-dimetylo-4-morfolinylo]-metylo}-1,3-oksazol-2-ilo)-1h-indazol-6-ilo]-2-(metyloksy)-3-pirydynylo]metanosulfonamidu |
Country Status (13)
Country | Link |
---|---|
US (1) | US8735390B2 (pl) |
EP (1) | EP2614058B1 (pl) |
JP (1) | JP5965402B2 (pl) |
DK (1) | DK2614058T3 (pl) |
ES (1) | ES2548036T3 (pl) |
HR (1) | HRP20151017T1 (pl) |
HU (1) | HUE026059T2 (pl) |
PL (1) | PL2614058T3 (pl) |
PT (1) | PT2614058E (pl) |
RS (1) | RS54286B1 (pl) |
SI (1) | SI2614058T1 (pl) |
SM (1) | SMT201500223B (pl) |
WO (1) | WO2012032067A1 (pl) |
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US20080275078A1 (en) | 2004-03-16 | 2008-11-06 | Glaxo Group Limited | Pyrazolo[3,4-B] Pyridine Compounds and Their Use as Pde4 Inhibitors |
AR050902A1 (es) | 2004-04-27 | 2006-12-06 | Glaxo Group Ltd | Compuesto de quinuclidina, composicion farmaceutica que lo comprende y su usopara preparar dicha composicion |
WO2006000401A1 (en) | 2004-06-28 | 2006-01-05 | Glaxo Group Limited | Substituted oxazines as glucocorticoid receptor modulators |
WO2006000398A1 (en) | 2004-06-28 | 2006-01-05 | Glaxo Group Limited | 2,3-benzoxazin derivatives as non-steroidal glucocorticoid receptor modulators |
GB0418045D0 (en) | 2004-08-12 | 2004-09-15 | Glaxo Group Ltd | Compounds |
BRPI0518222A (pt) | 2004-10-19 | 2008-11-04 | Hoffmann La Roche | composto, processo para a sua manufatura, composições farmacêuticas que os compreendem, método para o tratamento e/ou prevenção de enfermidades que estão associadas com a modulação de receptores de h3 e utilização dos mesmos |
US20090124588A1 (en) | 2005-01-10 | 2009-05-14 | Glaxo Group Limited | Androstane 17-Alpha-Carbonate for Use in the Treatment of Inflammatory and Allergic Conditions |
EP1841780B1 (en) | 2005-01-10 | 2011-07-27 | Glaxo Group Limited | Androstane 17-alpha-carbonate derivatives for use in the treatment of allergic and inflammatory conditions |
ES2566339T3 (es) * | 2008-06-05 | 2016-04-12 | Glaxo Group Limited | Derivados de 4-carboxamida indazol útiles como inhibidores de PI3-quinasas |
WO2010102958A1 (en) * | 2009-03-09 | 2010-09-16 | Glaxo Group Limited | 4-oxadiazol-2 -yl- indazoles as inhibitors of p13 kinases |
BRPI1016219B8 (pt) * | 2009-04-30 | 2021-05-25 | Glaxo Group Ltd | composto indazol substituído com oxazol, e, composição farmacêutica |
ES2602972T3 (es) * | 2010-09-08 | 2017-02-23 | Glaxosmithkline Intellectual Property Development Limited | Derivados de indazol para su uso en el tratamiento de infección por virus de la gripe |
-
2011
- 2011-09-06 PL PL11755311T patent/PL2614058T3/pl unknown
- 2011-09-06 US US13/821,585 patent/US8735390B2/en active Active
- 2011-09-06 SI SI201130595T patent/SI2614058T1/sl unknown
- 2011-09-06 PT PT117553115T patent/PT2614058E/pt unknown
- 2011-09-06 WO PCT/EP2011/065419 patent/WO2012032067A1/en active Application Filing
- 2011-09-06 DK DK11755311.5T patent/DK2614058T3/en active
- 2011-09-06 EP EP11755311.5A patent/EP2614058B1/en active Active
- 2011-09-06 RS RS20150611A patent/RS54286B1/en unknown
- 2011-09-06 ES ES11755311.5T patent/ES2548036T3/es active Active
- 2011-09-06 JP JP2013527583A patent/JP5965402B2/ja active Active
- 2011-09-06 HU HUE11755311A patent/HUE026059T2/en unknown
-
2015
- 2015-09-22 SM SM201500223T patent/SMT201500223B/xx unknown
- 2015-09-28 HR HRP20151017TT patent/HRP20151017T1/hr unknown
Also Published As
Publication number | Publication date |
---|---|
JP5965402B2 (ja) | 2016-08-03 |
SI2614058T1 (sl) | 2015-10-30 |
HRP20151017T1 (hr) | 2015-10-23 |
US8735390B2 (en) | 2014-05-27 |
SMT201500223B (it) | 2015-10-30 |
PT2614058E (pt) | 2015-10-27 |
ES2548036T3 (es) | 2015-10-13 |
EP2614058A1 (en) | 2013-07-17 |
HUE026059T2 (en) | 2016-05-30 |
DK2614058T3 (en) | 2015-09-28 |
WO2012032067A1 (en) | 2012-03-15 |
RS54286B1 (en) | 2016-02-29 |
EP2614058B1 (en) | 2015-07-08 |
US20130165441A1 (en) | 2013-06-27 |
JP2013537175A (ja) | 2013-09-30 |
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