SMT201500223B - Polimorfi e sali di n-[5-[4-(5-{[(2R,6S)-2,6-dimetil-4-morfolinil]metil}-1,3-ossazol-2-il)-1H-indazol-6-IL]-2-(metilossi)-3-piridinilÜmetansolfonammide - Google Patents
Polimorfi e sali di n-[5-[4-(5-{[(2R,6S)-2,6-dimetil-4-morfolinil]metil}-1,3-ossazol-2-il)-1H-indazol-6-IL]-2-(metilossi)-3-piridinilÜmetansolfonammideInfo
- Publication number
- SMT201500223B SMT201500223B SM201500223T SM201500223T SMT201500223B SM T201500223 B SMT201500223 B SM T201500223B SM 201500223 T SM201500223 T SM 201500223T SM 201500223 T SM201500223 T SM 201500223T SM T201500223 B SMT201500223 B SM T201500223B
- Authority
- SM
- San Marino
- Prior art keywords
- piridinilümetansolfonammide
- methyloxy
- indazol
- oxazol
- polymorphs
- Prior art date
Links
Classifications
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
- A61K31/00—Medicinal preparations containing organic active ingredients
- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/04—Centrally acting analgesics, e.g. opioids
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/14—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing three or more hetero rings
Applications Claiming Priority (2)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US38074810P | 2010-09-08 | 2010-09-08 | |
| PCT/EP2011/065419 WO2012032067A1 (en) | 2010-09-08 | 2011-09-06 | Polymorphs and salts of n- [5- [4- (5- { [(2r,6s) -2, 6 - dimethyl - 4 -morpholinyl] methyl} - 1, 3 - oxazol - 2 - yl) - 1h- inda zol-6-yl] -2- (methyloxy) - 3 - pyridinyl] methanesulfonamide |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| SMT201500223B true SMT201500223B (it) | 2015-10-30 |
Family
ID=44645691
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| SM201500223T SMT201500223B (it) | 2010-09-08 | 2015-09-22 | Polimorfi e sali di n-[5-[4-(5-{[(2R,6S)-2,6-dimetil-4-morfolinil]metil}-1,3-ossazol-2-il)-1H-indazol-6-IL]-2-(metilossi)-3-piridinilÜmetansolfonammide |
Country Status (13)
| Country | Link |
|---|---|
| US (1) | US8735390B2 (xx) |
| EP (1) | EP2614058B1 (xx) |
| JP (1) | JP5965402B2 (xx) |
| DK (1) | DK2614058T3 (xx) |
| ES (1) | ES2548036T3 (xx) |
| HR (1) | HRP20151017T1 (xx) |
| HU (1) | HUE026059T2 (xx) |
| PL (1) | PL2614058T3 (xx) |
| PT (1) | PT2614058E (xx) |
| RS (1) | RS54286B1 (xx) |
| SI (1) | SI2614058T1 (xx) |
| SM (1) | SMT201500223B (xx) |
| WO (1) | WO2012032067A1 (xx) |
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| WO2006000398A1 (en) | 2004-06-28 | 2006-01-05 | Glaxo Group Limited | 2,3-benzoxazin derivatives as non-steroidal glucocorticoid receptor modulators |
| WO2006000401A1 (en) | 2004-06-28 | 2006-01-05 | Glaxo Group Limited | Substituted oxazines as glucocorticoid receptor modulators |
| GB0418045D0 (en) | 2004-08-12 | 2004-09-15 | Glaxo Group Ltd | Compounds |
| MX2007004465A (es) | 2004-10-19 | 2007-05-07 | Hoffmann La Roche | Derivados de quinolina. |
| ATE517908T1 (de) | 2005-01-10 | 2011-08-15 | Glaxo Group Ltd | Androstan-17-alpha-carbonat-derivate zur verwendung bei der behandlung allergischer und entzündlicher zustände |
| US20090124588A1 (en) | 2005-01-10 | 2009-05-14 | Glaxo Group Limited | Androstane 17-Alpha-Carbonate for Use in the Treatment of Inflammatory and Allergic Conditions |
| ES2566339T3 (es) * | 2008-06-05 | 2016-04-12 | Glaxo Group Limited | Derivados de 4-carboxamida indazol útiles como inhibidores de PI3-quinasas |
| JP5656880B2 (ja) * | 2009-03-09 | 2015-01-21 | グラクソ グループ リミテッドＧｌａｘｏ Ｇｒｏｕｐ Ｌｉｍｉｔｅｄ | Ｐｉ３キナーゼの阻害剤としての４−オキサジアゾール−２−イル−インダゾール |
| DK2899191T3 (da) | 2009-04-30 | 2017-11-13 | Glaxo Group Ltd | Oxazol-substituerede indazoler som pi3-kinaseinhibitorer |
| JP5876051B2 (ja) * | 2010-09-08 | 2016-03-02 | グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッドＧｌａｘｏｓｍｉｔｈｋｌｉｎｅ Ｉｎｔｅｌｌｅｃｔｕａｌ Ｐｒｏｐｅｒｔｙ Ｄｅｖｅｌｏｐｍｅｎｔ Ｌｉｍｉｔｅｄ | インフルエンザウィルス感染の治療に使用するためのインダゾール誘導体 |
-
2011
- 2011-09-06 RS RS20150611A patent/RS54286B1/en unknown
- 2011-09-06 JP JP2013527583A patent/JP5965402B2/ja active Active
- 2011-09-06 HU HUE11755311A patent/HUE026059T2/en unknown
- 2011-09-06 ES ES11755311.5T patent/ES2548036T3/es active Active
- 2011-09-06 SI SI201130595T patent/SI2614058T1/sl unknown
- 2011-09-06 WO PCT/EP2011/065419 patent/WO2012032067A1/en active Application Filing
- 2011-09-06 US US13/821,585 patent/US8735390B2/en active Active
- 2011-09-06 DK DK11755311.5T patent/DK2614058T3/en active
- 2011-09-06 EP EP11755311.5A patent/EP2614058B1/en active Active
- 2011-09-06 PL PL11755311T patent/PL2614058T3/pl unknown
- 2011-09-06 PT PT117553115T patent/PT2614058E/pt unknown
-
2015
- 2015-09-22 SM SM201500223T patent/SMT201500223B/xx unknown
- 2015-09-28 HR HRP20151017TT patent/HRP20151017T1/hr unknown
Also Published As
| Publication number | Publication date |
|---|---|
| JP5965402B2 (ja) | 2016-08-03 |
| US8735390B2 (en) | 2014-05-27 |
| DK2614058T3 (en) | 2015-09-28 |
| PT2614058E (pt) | 2015-10-27 |
| ES2548036T3 (es) | 2015-10-13 |
| HUE026059T2 (en) | 2016-05-30 |
| US20130165441A1 (en) | 2013-06-27 |
| HRP20151017T1 (hr) | 2015-10-23 |
| EP2614058B1 (en) | 2015-07-08 |
| JP2013537175A (ja) | 2013-09-30 |
| SI2614058T1 (sl) | 2015-10-30 |
| RS54286B1 (en) | 2016-02-29 |
| WO2012032067A1 (en) | 2012-03-15 |
| EP2614058A1 (en) | 2013-07-17 |
| PL2614058T3 (pl) | 2015-12-31 |
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