ID28695A - TURUNAN-TURUNAN BENZO (b) TIEPIN 1,1-DIOKSIDA, PROSES PENYIAPAN, SEDIAAN FARMASI YANG MENGANDUNG SENYAWA-SENYAWA INI, DAN PENGGUNAANNYA - Google Patents

TURUNAN-TURUNAN BENZO (b) TIEPIN 1,1-DIOKSIDA, PROSES PENYIAPAN, SEDIAAN FARMASI YANG MENGANDUNG SENYAWA-SENYAWA INI, DAN PENGGUNAANNYA

Info

Publication number
ID28695A
ID28695A IDW20002562A ID20002562A ID28695A ID 28695 A ID28695 A ID 28695A ID W20002562 A IDW20002562 A ID W20002562A ID 20002562 A ID20002562 A ID 20002562A ID 28695 A ID28695 A ID 28695A
Authority
ID
Indonesia
Prior art keywords
tiepin
benzo
designs
dioxide
compounds
Prior art date
Application number
IDW20002562A
Other languages
English (en)
Indonesian (id)
Inventor
Wendelin Dr Frick
Alfons Dr Enhsen
Heiner Dr Glombik
Hubert Dr Heuer
Original Assignee
Aventis Pharma Deutschland
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Aventis Pharma Deutschland filed Critical Aventis Pharma Deutschland
Publication of ID28695A publication Critical patent/ID28695A/id

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D337/00Heterocyclic compounds containing rings of more than six members having one sulfur atom as the only ring hetero atom
    • C07D337/02Seven-membered rings
    • C07D337/06Seven-membered rings condensed with carbocyclic rings or ring systems
    • C07D337/08Seven-membered rings condensed with carbocyclic rings or ring systems condensed with one six-membered ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/335Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A61K31/35Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom
    • A61K31/351Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin having six-membered rings with one oxygen as the only ring hetero atom not condensed with another ring
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/38Heterocyclic compounds having sulfur as a ring hetero atom
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P1/00Drugs for disorders of the alimentary tract or the digestive system
    • A61P1/16Drugs for disorders of the alimentary tract or the digestive system for liver or gallbladder disorders, e.g. hepatoprotective agents, cholagogues, litholytics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P13/00Drugs for disorders of the urinary system
    • A61P13/04Drugs for disorders of the urinary system for urolithiasis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00Drugs for disorders of the metabolism
    • A61P3/06Antihyperlipidemics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00Drugs for disorders of the cardiovascular system
    • A61P9/10Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07KPEPTIDES
    • C07K5/00Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
    • C07K5/04Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
    • C07K5/06Dipeptides
    • C07K5/06086Dipeptides with the first amino acid being basic
    • CCHEMISTRY; METALLURGY
    • C08ORGANIC MACROMOLECULAR COMPOUNDS; THEIR PREPARATION OR CHEMICAL WORKING-UP; COMPOSITIONS BASED THEREON
    • C08GMACROMOLECULAR COMPOUNDS OBTAINED OTHERWISE THAN BY REACTIONS ONLY INVOLVING UNSATURATED CARBON-TO-CARBON BONDS
    • C08G65/00Macromolecular compounds obtained by reactions forming an ether link in the main chain of the macromolecule
    • C08G65/02Macromolecular compounds obtained by reactions forming an ether link in the main chain of the macromolecule from cyclic ethers by opening of the heterocyclic ring
    • C08G65/32Polymers modified by chemical after-treatment
    • C08G65/329Polymers modified by chemical after-treatment with organic compounds
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K38/00Medicinal preparations containing peptides
    • YGENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02PCLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00Technologies relating to chemical industry
    • Y02P20/50Improvements relating to the production of bulk chemicals
    • Y02P20/55Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • Medicinal Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Obesity (AREA)
  • Biochemistry (AREA)
  • Epidemiology (AREA)
  • Proteomics, Peptides & Aminoacids (AREA)
  • Diabetes (AREA)
  • Hematology (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Polymers & Plastics (AREA)
  • Urology & Nephrology (AREA)
  • Biophysics (AREA)
  • Gastroenterology & Hepatology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
IDW20002562A 1998-06-10 1999-05-28 TURUNAN-TURUNAN BENZO (b) TIEPIN 1,1-DIOKSIDA, PROSES PENYIAPAN, SEDIAAN FARMASI YANG MENGANDUNG SENYAWA-SENYAWA INI, DAN PENGGUNAANNYA ID28695A (id)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19825804A DE19825804C2 (de) 1998-06-10 1998-06-10 1,4-Benzothiepin-1,1-dioxidderivate, Verfahren zu deren Herstellung und diese Verbindungen enthaltende Arzneimittel

Publications (1)

Publication Number Publication Date
ID28695A true ID28695A (id) 2001-06-28

Family

ID=7870440

Family Applications (2)

Application Number Title Priority Date Filing Date
IDW20002562A ID28695A (id) 1998-06-10 1999-05-28 TURUNAN-TURUNAN BENZO (b) TIEPIN 1,1-DIOKSIDA, PROSES PENYIAPAN, SEDIAAN FARMASI YANG MENGANDUNG SENYAWA-SENYAWA INI, DAN PENGGUNAANNYA
IDW20002564A ID26876A (id) 1998-06-10 1999-05-29 Derivat-derivat benzotiepin 1,1-dioksida, proses pembuatannya, bahan-bahan farmasi yang terdiri dari senyawa-senyawa ini dan penggunaannya

Family Applications After (1)

Application Number Title Priority Date Filing Date
IDW20002564A ID26876A (id) 1998-06-10 1999-05-29 Derivat-derivat benzotiepin 1,1-dioksida, proses pembuatannya, bahan-bahan farmasi yang terdiri dari senyawa-senyawa ini dan penggunaannya

Country Status (26)

Country Link
US (1) US6387944B1 (es)
EP (2) EP1086092B1 (es)
JP (2) JP4374426B2 (es)
KR (2) KR100681721B1 (es)
CN (2) CN1127497C (es)
AR (2) AR018634A1 (es)
AT (2) ATE227715T1 (es)
AU (2) AU753275B2 (es)
BR (2) BR9912188B1 (es)
CA (2) CA2334775C (es)
CZ (2) CZ297989B6 (es)
DE (3) DE19825804C2 (es)
DK (2) DK1086092T3 (es)
ES (2) ES2182535T3 (es)
HK (2) HK1039490A1 (es)
HU (2) HU229761B1 (es)
ID (2) ID28695A (es)
IL (1) IL140078A (es)
NO (1) NO327075B1 (es)
NZ (1) NZ508681A (es)
PL (2) PL196074B1 (es)
PT (2) PT1086092E (es)
RU (2) RU2215001C2 (es)
TR (2) TR200003634T2 (es)
WO (2) WO1999064410A1 (es)
ZA (2) ZA200007060B (es)

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EG26979A (en) 2000-12-21 2015-03-01 Astrazeneca Ab Chemical compounds
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GB0121337D0 (en) 2001-09-04 2001-10-24 Astrazeneca Ab Chemical compounds
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GB0209467D0 (en) 2002-04-25 2002-06-05 Astrazeneca Ab Chemical compounds
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SE0201937D0 (sv) 2002-06-20 2002-06-20 Astrazeneca Ab Therapeutic agents
US20040138145A1 (en) * 2002-12-12 2004-07-15 Aventis Pharma S.A. Application of intestinal biliary acid reuptake inhibitors for the prevention and treatment of alzheimer's disease
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Also Published As

Publication number Publication date
AU4503199A (en) 1999-12-30
NO20006251L (no) 2001-02-07
IL140078A0 (en) 2002-02-10
AR018633A1 (es) 2001-11-28
BR9911123B1 (pt) 2010-12-14
HK1039490A1 (en) 2002-04-26
ATE259372T1 (de) 2004-02-15
NO20006251D0 (no) 2000-12-08
KR20010052682A (ko) 2001-06-25
CA2334775A1 (en) 1999-12-16
AU4501999A (en) 1999-12-30
DE19825804A1 (de) 1999-12-16
PL196074B1 (pl) 2007-12-31
AU753275B2 (en) 2002-10-10
HUP0102256A3 (en) 2002-04-29
KR20010052701A (ko) 2001-06-25
JP2002517491A (ja) 2002-06-18
CZ297925B6 (cs) 2007-05-02
TR200003634T2 (tr) 2001-06-21
JP2002517490A (ja) 2002-06-18
BR9912188A (pt) 2001-04-10
ZA200007060B (en) 2001-07-18
KR100562184B1 (ko) 2006-03-20
PL345901A1 (en) 2002-01-14
US6387944B1 (en) 2002-05-14
CN1152039C (zh) 2004-06-02
NO327075B1 (no) 2009-04-20
DE59903411D1 (de) 2002-12-19
DK1086113T3 (da) 2004-05-24
ES2182535T3 (es) 2003-03-01
BR9912188B1 (pt) 2010-12-14
IL140078A (en) 2004-08-31
HU229761B1 (hu) 2014-06-30
PL196057B1 (pl) 2007-11-30
WO1999064409A2 (de) 1999-12-16
NZ508681A (en) 2002-06-28
DE19825804C2 (de) 2000-08-24
HUP0102256A1 (hu) 2001-12-28
CN1305469A (zh) 2001-07-25
CA2334773C (en) 2009-05-26
AR018634A1 (es) 2001-11-28
EP1086113A2 (de) 2001-03-28
DE59908522D1 (de) 2004-03-18
RU2215001C2 (ru) 2003-10-27
ZA200007061B (en) 2001-07-18
AU752633B2 (en) 2002-09-26
EP1086092A1 (de) 2001-03-28
EP1086092B1 (de) 2002-11-13
CN1127497C (zh) 2003-11-12
PT1086092E (pt) 2003-03-31
ES2215387T3 (es) 2004-10-01
EP1086113B1 (de) 2004-02-11
RU2220141C2 (ru) 2003-12-27
CZ297989B6 (cs) 2007-05-16
WO1999064409A3 (de) 2000-03-02
HUP0102554A1 (hu) 2001-10-28
KR100681721B1 (ko) 2007-02-15
PL344827A1 (en) 2001-11-19
TR200003632T2 (tr) 2001-04-20
HUP0102554A3 (en) 2002-12-28
CN1305487A (zh) 2001-07-25
JP3374129B2 (ja) 2003-02-04
HK1036799A1 (en) 2002-01-18
CA2334773A1 (en) 1999-12-16
ID26876A (id) 2001-02-15
BR9911123A (pt) 2006-01-03
CZ20004592A3 (cs) 2001-04-11
HU228570B1 (en) 2013-04-29
DK1086092T3 (da) 2003-03-10
CZ20004591A3 (cs) 2001-04-11
ATE227715T1 (de) 2002-11-15
JP4374426B2 (ja) 2009-12-02
WO1999064410A1 (de) 1999-12-16
PT1086113E (pt) 2004-06-30
CA2334775C (en) 2009-10-13

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