HU225051B1 - Sublingual or buccal pharmaceutical compositions containing trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1h-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole - Google Patents

Sublingual or buccal pharmaceutical compositions containing trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1h-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole Download PDF

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Publication number
HU225051B1
HU225051B1 HU9602383A HU9602383A HU225051B1 HU 225051 B1 HU225051 B1 HU 225051B1 HU 9602383 A HU9602383 A HU 9602383A HU 9602383 A HU9602383 A HU 9602383A HU 225051 B1 HU225051 B1 HU 225051B1
Authority
HU
Hungary
Prior art keywords
oxepino
dibenz
tetrahydro
chloro
methyl
Prior art date
Application number
HU9602383A
Other languages
English (en)
Hungarian (hu)
Other versions
HUT76319A (en
HU9602383D0 (en
Inventor
Leonardus Petrus C Delbressine
Johannes Hubertus Wieringa
Original Assignee
Organon Ireland Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8216678&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=HU225051(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by Organon Ireland Ltd filed Critical Organon Ireland Ltd
Publication of HU9602383D0 publication Critical patent/HU9602383D0/hu
Publication of HUT76319A publication Critical patent/HUT76319A/hu
Publication of HU225051B1 publication Critical patent/HU225051B1/hu

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
HU9602383A 1994-03-02 1995-03-01 Sublingual or buccal pharmaceutical compositions containing trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1h-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole HU225051B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
EP94200521 1994-03-02
PCT/EP1995/000765 WO1995023600A1 (en) 1994-03-02 1995-03-01 Sublingual or buccal pharmaceutical composition

Publications (3)

Publication Number Publication Date
HU9602383D0 HU9602383D0 (en) 1996-10-28
HUT76319A HUT76319A (en) 1997-08-28
HU225051B1 true HU225051B1 (en) 2006-05-29

Family

ID=8216678

Family Applications (1)

Application Number Title Priority Date Filing Date
HU9602383A HU225051B1 (en) 1994-03-02 1995-03-01 Sublingual or buccal pharmaceutical compositions containing trans-5-chloro-2-methyl-2,3,3a,12b-tetrahydro-1h-dibenz[2,3:6,7]oxepino[4,5-c]pyrrole

Country Status (23)

Country Link
US (1) US5763476A (https=)
EP (1) EP0746317B1 (https=)
JP (2) JP4099224B2 (https=)
KR (1) KR100330942B1 (https=)
CN (1) CN1079670C (https=)
AT (1) ATE167057T1 (https=)
AU (1) AU692530B2 (https=)
BR (2) BR9506924A (https=)
CA (1) CA2182981C (https=)
CZ (1) CZ284633B6 (https=)
DE (2) DE69502939T2 (https=)
DK (1) DK0746317T3 (https=)
ES (1) ES2118584T3 (https=)
FI (1) FI117923B (https=)
FR (1) FR10C0056I2 (https=)
HK (1) HK1008417A1 (https=)
HU (1) HU225051B1 (https=)
LU (1) LU91751I2 (https=)
NO (2) NO308772B1 (https=)
NZ (1) NZ282394A (https=)
PL (1) PL180465B1 (https=)
RU (1) RU2139051C1 (https=)
WO (1) WO1995023600A1 (https=)

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Also Published As

Publication number Publication date
JP4616810B2 (ja) 2011-01-19
WO1995023600A1 (en) 1995-09-08
ATE167057T1 (de) 1998-06-15
CA2182981A1 (en) 1995-09-08
RU2139051C1 (ru) 1999-10-10
NO308772B1 (no) 2000-10-30
NZ282394A (en) 1997-12-19
EP0746317B1 (en) 1998-06-10
CN1079670C (zh) 2002-02-27
KR100330942B1 (ko) 2002-11-16
FI117923B (fi) 2007-04-30
JP2006342178A (ja) 2006-12-21
PL180465B1 (pl) 2001-02-28
BR1100625A (pt) 1999-12-28
PL316080A1 (en) 1996-12-23
CA2182981C (en) 2006-10-17
HUT76319A (en) 1997-08-28
CN1143320A (zh) 1997-02-19
FI963398L (fi) 1996-08-30
DE69502939T2 (de) 1998-10-22
CZ284633B6 (cs) 1999-01-13
AU692530B2 (en) 1998-06-11
US5763476A (en) 1998-06-09
CZ254196A3 (en) 1997-10-15
JP4099224B2 (ja) 2008-06-11
FI963398A0 (fi) 1996-08-30
LU91751I2 (fr) 2011-01-04
DE69502939D1 (de) 1998-07-16
JPH09509674A (ja) 1997-09-30
HU9602383D0 (en) 1996-10-28
DE122010000050I2 (de) 2011-07-21
DK0746317T3 (da) 1999-03-22
NO963639D0 (no) 1996-08-30
AU1947895A (en) 1995-09-18
HK1008417A1 (en) 1999-05-07
NO963639L (no) 1996-10-30
DE122010000050I1 (de) 2011-05-05
ES2118584T3 (es) 1998-09-16
FR10C0056I2 (https=) 2011-11-25
NO2010024I1 (no) 2011-01-03
BR9506924A (pt) 1997-09-30
EP0746317A1 (en) 1996-12-11
FR10C0056I1 (https=) 2011-01-28
NO2010024I2 (no) 2012-04-10
MX9603713A (es) 1997-12-31

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