KR100330942B1 - 설하또는협측투여용약학조성물 - Google Patents

설하또는협측투여용약학조성물 Download PDF

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Publication number
KR100330942B1
KR100330942B1 KR1019960704774A KR19960704774A KR100330942B1 KR 100330942 B1 KR100330942 B1 KR 100330942B1 KR 1019960704774 A KR1019960704774 A KR 1019960704774A KR 19960704774 A KR19960704774 A KR 19960704774A KR 100330942 B1 KR100330942 B1 KR 100330942B1
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KR
South Korea
Prior art keywords
sublingual
oxepino
tetrahydro
chloro
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired - Lifetime
Application number
KR1019960704774A
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English (en)
Korean (ko)
Inventor
페트루스 카를라 델브레씨네 레오나르두스
후베르투스 비에린가 요한네스
Original Assignee
악조 노벨 엔.브이.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
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First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=8216678&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=KR100330942(B1) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Application filed by 악조 노벨 엔.브이. filed Critical 악조 노벨 엔.브이.
Application granted granted Critical
Publication of KR100330942B1 publication Critical patent/KR100330942B1/ko
Assigned to 오르가논 아일랜드 리미티드 reassignment 오르가논 아일랜드 리미티드 권리의 전부이전등록 Assignors: 악조 노벨 엔.브이.
Assigned to 엔.브이.오가논 reassignment 엔.브이.오가논 권리의 전부이전등록 Assignors: 오르가논 아일랜드 리미티드
Assigned to 엠에스디 오스 비.브이. reassignment 엠에스디 오스 비.브이. 권리의 전부이전등록 Assignors: 엔.브이.오가논
Assigned to 머크 샤프 앤 도메 비.브이. reassignment 머크 샤프 앤 도메 비.브이. 권리의 전부이전등록 Assignors: 엠에스디 오스 비.브이.
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A61K31/407—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil condensed with other heterocyclic ring systems, e.g. ketorolac, physostigmine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/006—Oral mucosa, e.g. mucoadhesive forms, sublingual droplets; Buccal patches or films; Buccal sprays
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/2095—Tabletting processes
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/18—Antipsychotics, i.e. neuroleptics; Drugs for mania or schizophrenia
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/22—Anxiolytics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0053—Mouth and digestive tract, i.e. intraoral and peroral administration
    • A61K9/0056—Mouth soluble or dispersible forms; Suckable, eatable, chewable coherent forms; Forms rapidly disintegrating in the mouth; Lozenges; Lollipops; Bite capsules; Baked products; Baits or other oral forms for animals

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Neurosurgery (AREA)
  • Biomedical Technology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Neurology (AREA)
  • Physiology (AREA)
  • Nutrition Science (AREA)
  • Psychiatry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
KR1019960704774A 1994-03-02 1995-03-01 설하또는협측투여용약학조성물 Expired - Lifetime KR100330942B1 (ko)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
EP94200521.6 1994-03-02
EP94200521 1994-03-02
PCT/EP1995/000765 WO1995023600A1 (en) 1994-03-02 1995-03-01 Sublingual or buccal pharmaceutical composition

Publications (1)

Publication Number Publication Date
KR100330942B1 true KR100330942B1 (ko) 2002-11-16

Family

ID=8216678

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019960704774A Expired - Lifetime KR100330942B1 (ko) 1994-03-02 1995-03-01 설하또는협측투여용약학조성물

Country Status (23)

Country Link
US (1) US5763476A (https=)
EP (1) EP0746317B1 (https=)
JP (2) JP4099224B2 (https=)
KR (1) KR100330942B1 (https=)
CN (1) CN1079670C (https=)
AT (1) ATE167057T1 (https=)
AU (1) AU692530B2 (https=)
BR (2) BR9506924A (https=)
CA (1) CA2182981C (https=)
CZ (1) CZ284633B6 (https=)
DE (2) DE69502939T2 (https=)
DK (1) DK0746317T3 (https=)
ES (1) ES2118584T3 (https=)
FI (1) FI117923B (https=)
FR (1) FR10C0056I2 (https=)
HK (1) HK1008417A1 (https=)
HU (1) HU225051B1 (https=)
LU (1) LU91751I2 (https=)
NO (2) NO308772B1 (https=)
NZ (1) NZ282394A (https=)
PL (1) PL180465B1 (https=)
RU (1) RU2139051C1 (https=)
WO (1) WO1995023600A1 (https=)

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EP1710245B1 (en) * 2005-04-07 2007-08-22 N.V. Organon Crystal form of asenapine maleate
US7741358B2 (en) 2005-04-14 2010-06-22 N.V. Organon Crystal form of asenapine maleate
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Also Published As

Publication number Publication date
JP4616810B2 (ja) 2011-01-19
WO1995023600A1 (en) 1995-09-08
ATE167057T1 (de) 1998-06-15
CA2182981A1 (en) 1995-09-08
RU2139051C1 (ru) 1999-10-10
NO308772B1 (no) 2000-10-30
NZ282394A (en) 1997-12-19
EP0746317B1 (en) 1998-06-10
CN1079670C (zh) 2002-02-27
FI117923B (fi) 2007-04-30
JP2006342178A (ja) 2006-12-21
PL180465B1 (pl) 2001-02-28
BR1100625A (pt) 1999-12-28
PL316080A1 (en) 1996-12-23
CA2182981C (en) 2006-10-17
HUT76319A (en) 1997-08-28
CN1143320A (zh) 1997-02-19
FI963398L (fi) 1996-08-30
DE69502939T2 (de) 1998-10-22
CZ284633B6 (cs) 1999-01-13
AU692530B2 (en) 1998-06-11
US5763476A (en) 1998-06-09
HU225051B1 (en) 2006-05-29
CZ254196A3 (en) 1997-10-15
JP4099224B2 (ja) 2008-06-11
FI963398A0 (fi) 1996-08-30
LU91751I2 (fr) 2011-01-04
DE69502939D1 (de) 1998-07-16
JPH09509674A (ja) 1997-09-30
HU9602383D0 (en) 1996-10-28
DE122010000050I2 (de) 2011-07-21
DK0746317T3 (da) 1999-03-22
NO963639D0 (no) 1996-08-30
AU1947895A (en) 1995-09-18
HK1008417A1 (en) 1999-05-07
NO963639L (no) 1996-10-30
DE122010000050I1 (de) 2011-05-05
ES2118584T3 (es) 1998-09-16
FR10C0056I2 (https=) 2011-11-25
NO2010024I1 (no) 2011-01-03
BR9506924A (pt) 1997-09-30
EP0746317A1 (en) 1996-12-11
FR10C0056I1 (https=) 2011-01-28
NO2010024I2 (no) 2012-04-10
MX9603713A (es) 1997-12-31

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