HRP20120215T1 - Derivati sulfonil-pirazolinil-1-karboksamidina kao 5-ht6-antagonista - Google Patents

Derivati sulfonil-pirazolinil-1-karboksamidina kao 5-ht6-antagonista Download PDF

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HRP20120215T1
HRP20120215T1 HR20120215T HRP20120215T HRP20120215T1 HR P20120215 T1 HRP20120215 T1 HR P20120215T1 HR 20120215 T HR20120215 T HR 20120215T HR P20120215 T HRP20120215 T HR P20120215T HR P20120215 T1 HRP20120215 T1 HR P20120215T1
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HR20120215T
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I. Iwema Bakker Wouter
G. Keizer Hiskias
A.W. Van Der Neut Martina
G. Kruse Cornelis
Van Loevezijn Arnold
Zorgdrager Jan
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Abbott Healthcare Products B.V.
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Publication of HRP20120215T1 publication Critical patent/HRP20120215T1/hr

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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/0012—Galenical forms characterised by the site of application
    • A61K9/0019—Injectable compositions; Intramuscular, intravenous, arterial, subcutaneous administration; Compositions to be administered through the skin in an invasive manner
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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
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  • Plural Heterocyclic Compounds (AREA)
HR20120215T 2006-09-22 2012-03-06 Derivati sulfonil-pirazolinil-1-karboksamidina kao 5-ht6-antagonista HRP20120215T1 (hr)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US846406A 2006-09-22 2006-09-22
EP06121087 2006-09-22
US90286507P 2007-02-23 2007-02-23
EP07102965 2007-02-23
PCT/EP2007/059944 WO2008034863A2 (en) 2006-09-22 2007-09-20 Sulfonylpyrazoline carboxamidine derivatives as 5-ht6 antagonists

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AR070898A1 (es) 2008-03-18 2010-05-12 Solvay Pharm Bv Derivados de arilsulfonil pirazolin carboxamidina como antagonistas de 5-ht6
AR079935A1 (es) 2010-01-29 2012-02-29 Abbott Healthcare Products Bv Sintesis de derivados de pirazolin carboxamidina sustituida
WO2013055386A2 (en) * 2011-10-03 2013-04-18 The University Of Utah Research Foundation Application of 5-ht6 receptor antagonists for the alleviation of cognitive deficits of down syndrome
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ES2674476T3 (es) 2013-07-25 2018-07-02 Uniwersytet Jagiellonski Derivados de pirroloquinolina como antagonistas de 5-HT6, método de preparación y uso de los mismos
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