DK2069310T3 - Sulfonylpyrazolin-1-carboxamidin-derivater som 5-HT6-antagonister - Google Patents

Sulfonylpyrazolin-1-carboxamidin-derivater som 5-HT6-antagonister

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Publication number
DK2069310T3
DK2069310T3 DK07820387.4T DK07820387T DK2069310T3 DK 2069310 T3 DK2069310 T3 DK 2069310T3 DK 07820387 T DK07820387 T DK 07820387T DK 2069310 T3 DK2069310 T3 DK 2069310T3
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Prior art keywords
sulfonylpyrazoline
antagonists
carboxamidine derivatives
carboxamidine
derivatives
Prior art date
Application number
DK07820387.4T
Other languages
English (en)
Inventor
Bakker Wouter I Iwema
Hiskias G Keizer
Van Der Martina A W Neut
Cornelis G Kruse
Van Arnold Loevezijn
Jan Zorgdrager
Original Assignee
Abbott Healthcare Products Bv
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Publication of DK2069310T3 publication Critical patent/DK2069310T3/da

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    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
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    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/41—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with two or more ring hetero atoms, at least one of which being nitrogen, e.g. tetrazole
    • A61K31/415—1,2-Diazoles
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DK07820387.4T 2006-09-22 2007-09-20 Sulfonylpyrazolin-1-carboxamidin-derivater som 5-HT6-antagonister DK2069310T3 (da)

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
US84640606P 2006-09-22 2006-09-22
EP06121087 2006-09-22
US90286507P 2007-02-23 2007-02-23
EP07102965 2007-02-23
PCT/EP2007/059944 WO2008034863A2 (en) 2006-09-22 2007-09-20 Sulfonylpyrazoline carboxamidine derivatives as 5-ht6 antagonists

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DK2069310T3 true DK2069310T3 (da) 2012-03-19

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US20080311179A1 (en) 2008-12-18
SA07280510B1 (ar) 2012-02-07
JP2010504302A (ja) 2010-02-12
HK1137992A1 (en) 2010-08-13
KR20090060356A (ko) 2009-06-11
US8722887B2 (en) 2014-05-13
AR062907A1 (es) 2008-12-17
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SI2069310T1 (sl) 2012-02-29
HRP20120215T1 (hr) 2012-04-30
CA2662484A1 (en) 2008-03-27
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EP2069310B1 (en) 2011-12-14
MY147263A (en) 2012-11-30
US20140303372A1 (en) 2014-10-09
JP5225280B2 (ja) 2013-07-03
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AU2007298987A1 (en) 2008-03-27
BRPI0716860A2 (pt) 2013-10-15
PT2069310E (pt) 2012-02-28
ES2377996T3 (es) 2012-04-04
US20100145042A1 (en) 2010-06-10
WO2008034863A3 (en) 2008-05-08
ATE537149T1 (de) 2011-12-15
CA2662484C (en) 2015-06-23
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CN101679279B (zh) 2013-11-13
WO2008034863A2 (en) 2008-03-27
AU2007298987B2 (en) 2012-10-04
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