DK2094263T3 - 2-adamantyl-butyramidderivater som selektive 11 beta-hsd1-inhibitorer - Google Patents
2-adamantyl-butyramidderivater som selektive 11 beta-hsd1-inhibitorerInfo
- Publication number
- DK2094263T3 DK2094263T3 DK07856225.3T DK07856225T DK2094263T3 DK 2094263 T3 DK2094263 T3 DK 2094263T3 DK 07856225 T DK07856225 T DK 07856225T DK 2094263 T3 DK2094263 T3 DK 2094263T3
- Authority
- DK
- Denmark
- Prior art keywords
- adamantyl
- beta
- selective
- hsd1 inhibitors
- butyramide
- Prior art date
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- C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
- C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
- C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C07C233/04—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with carbon atoms of carboxamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton
- C07C233/06—Carboxylic acid amides having carbon atoms of carboxamide groups bound to hydrogen atoms or to acyclic carbon atoms having nitrogen atoms of carboxamide groups bound to hydrogen atoms or to carbon atoms of unsubstituted hydrocarbon radicals with carbon atoms of carboxamide groups bound to acyclic carbon atoms of an acyclic saturated carbon skeleton having the nitrogen atom of at least one of the carboxamide groups bound to a carbon atom of a ring other than a six-membered aromatic ring
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- C07D295/18—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms acylated on ring nitrogen atoms by radicals derived from carboxylic acids, or sulfur or nitrogen analogues thereof
- C07D295/182—Radicals derived from carboxylic acids
- C07D295/185—Radicals derived from carboxylic acids from aliphatic carboxylic acids
Applications Claiming Priority (2)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
EP06292011A EP1935420A1 (en) | 2006-12-21 | 2006-12-21 | 2-Adamantyl-butyramide derivatives as selective 11beta-HSD1 inhibitors |
PCT/EP2007/010124 WO2008074384A1 (en) | 2006-12-21 | 2007-11-22 | 2-ADAMANTYL-BUTYRAMIDE DERIVATIVES AS SELECTIVE 11βETA-HSD1 INHIBITORS |
Publications (1)
Publication Number | Publication Date |
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DK2094263T3 true DK2094263T3 (da) | 2013-12-02 |
Family
ID=37983344
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK07856225.3T DK2094263T3 (da) | 2006-12-21 | 2007-11-22 | 2-adamantyl-butyramidderivater som selektive 11 beta-hsd1-inhibitorer |
Country Status (12)
Country | Link |
---|---|
US (1) | US8183265B2 (da) |
EP (2) | EP1935420A1 (da) |
JP (1) | JP5546866B2 (da) |
AR (1) | AR064474A1 (da) |
AU (1) | AU2007334983B2 (da) |
CA (1) | CA2673430C (da) |
DK (1) | DK2094263T3 (da) |
ES (1) | ES2442518T3 (da) |
IL (1) | IL199112A (da) |
PL (1) | PL2094263T3 (da) |
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WO (1) | WO2008074384A1 (da) |
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2006
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2007
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- 2007-11-22 JP JP2009541801A patent/JP5546866B2/ja active Active
- 2007-11-22 EP EP07856225.3A patent/EP2094263B1/en active Active
- 2007-11-22 PT PT78562253T patent/PT2094263E/pt unknown
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PT2094263E (pt) | 2014-01-13 |
JP5546866B2 (ja) | 2014-07-09 |
IL199112A (en) | 2014-05-28 |
AU2007334983B2 (en) | 2012-08-16 |
PL2094263T3 (pl) | 2014-03-31 |
US20100022597A1 (en) | 2010-01-28 |
EP2094263A1 (en) | 2009-09-02 |
CA2673430A1 (en) | 2008-06-26 |
US8183265B2 (en) | 2012-05-22 |
EP2094263B1 (en) | 2013-10-16 |
AU2007334983A1 (en) | 2008-06-26 |
AR064474A1 (es) | 2009-04-01 |
CA2673430C (en) | 2015-06-16 |
ES2442518T3 (es) | 2014-02-12 |
EP1935420A1 (en) | 2008-06-25 |
JP2010513337A (ja) | 2010-04-30 |
WO2008074384A1 (en) | 2008-06-26 |
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