HRP20110964T1 - PIPERIDINSKI AGONISTI GPCR-a - Google Patents

PIPERIDINSKI AGONISTI GPCR-a Download PDF

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Publication number
HRP20110964T1
HRP20110964T1 HR20110964T HRP20110964T HRP20110964T1 HR P20110964 T1 HRP20110964 T1 HR P20110964T1 HR 20110964 T HR20110964 T HR 20110964T HR P20110964 T HRP20110964 T HR P20110964T HR P20110964 T1 HRP20110964 T1 HR P20110964T1
Authority
HR
Croatia
Prior art keywords
pharmaceutically acceptable
acceptable salt
compound according
compound
image
Prior art date
Application number
HR20110964T
Other languages
English (en)
Croatian (hr)
Inventor
Sarah Bertram Lisa
Colin Thor Fyfe Matthew
Perpetua Jeevaratnam Revathy
Keily John
Andrew Swain Simon
Original Assignee
Prosidion Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from GB0700124A external-priority patent/GB0700124D0/en
Priority claimed from GB0708740A external-priority patent/GB0708740D0/en
Priority claimed from GB0719762A external-priority patent/GB0719762D0/en
Application filed by Prosidion Ltd filed Critical Prosidion Ltd
Publication of HRP20110964T1 publication Critical patent/HRP20110964T1/hr

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D413/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms
    • C07D413/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings
    • C07D413/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and oxygen atoms as the only ring hetero atoms containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A61K31/4523—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems
    • A61K31/454—Non condensed piperidines, e.g. piperocaine containing further heterocyclic ring systems containing a five-membered ring with nitrogen as a ring hetero atom, e.g. pimozide, domperidone
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/04—Anorexiants; Antiobesity agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/06—Antihyperlipidemics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P3/00—Drugs for disorders of the metabolism
    • A61P3/08—Drugs for disorders of the metabolism for glucose homeostasis
    • A61P3/10—Drugs for disorders of the metabolism for glucose homeostasis for hyperglycaemia, e.g. antidiabetics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/10—Drugs for disorders of the cardiovascular system for treating ischaemic or atherosclerotic diseases, e.g. antianginal drugs, coronary vasodilators, drugs for myocardial infarction, retinopathy, cerebrovascula insufficiency, renal arteriosclerosis
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P9/00—Drugs for disorders of the cardiovascular system
    • A61P9/12—Antihypertensives

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Diabetes (AREA)
  • Obesity (AREA)
  • Hematology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Cardiology (AREA)
  • Vascular Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Child & Adolescent Psychology (AREA)
  • Emergency Medicine (AREA)
  • Endocrinology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Peptides Or Proteins (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
HR20110964T 2007-01-04 2008-01-04 PIPERIDINSKI AGONISTI GPCR-a HRP20110964T1 (hr)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
GB0700124A GB0700124D0 (en) 2007-01-04 2007-01-04 GPCR agonists
GB0708740A GB0708740D0 (en) 2007-05-08 2007-05-08 Gpcr agonists
GB0719762A GB0719762D0 (en) 2007-10-10 2007-10-10 GPCR agonists
PCT/GB2008/050011 WO2008081205A1 (en) 2007-01-04 2008-01-04 Piperidine gpcr agonists

Publications (1)

Publication Number Publication Date
HRP20110964T1 true HRP20110964T1 (hr) 2012-01-31

Family

ID=39203222

Family Applications (1)

Application Number Title Priority Date Filing Date
HR20110964T HRP20110964T1 (hr) 2007-01-04 2008-01-04 PIPERIDINSKI AGONISTI GPCR-a

Country Status (27)

Country Link
US (1) US20100022591A1 (OSRAM)
EP (2) EP2114931B1 (OSRAM)
JP (1) JP2010514829A (OSRAM)
KR (1) KR20090104092A (OSRAM)
CN (1) CN101627036A (OSRAM)
AR (1) AR064736A1 (OSRAM)
AT (1) ATE531710T1 (OSRAM)
AU (1) AU2008203673A1 (OSRAM)
BR (1) BRPI0806468A2 (OSRAM)
CA (1) CA2674093A1 (OSRAM)
CL (1) CL2008000017A1 (OSRAM)
DK (1) DK2114931T3 (OSRAM)
EA (1) EA015805B9 (OSRAM)
ES (1) ES2376015T3 (OSRAM)
HR (1) HRP20110964T1 (OSRAM)
IL (1) IL199680A0 (OSRAM)
MA (1) MA31084B1 (OSRAM)
MX (1) MX2009007180A (OSRAM)
NZ (1) NZ578144A (OSRAM)
PE (1) PE20081849A1 (OSRAM)
PL (1) PL2114931T3 (OSRAM)
PT (1) PT2114931E (OSRAM)
RS (1) RS52168B (OSRAM)
SA (1) SA08280756B1 (OSRAM)
SI (1) SI2114931T1 (OSRAM)
TW (1) TWI380818B (OSRAM)
WO (1) WO2008081205A1 (OSRAM)

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PT2114931E (pt) 2012-01-12
EA015805B9 (ru) 2012-03-30
ES2376015T3 (es) 2012-03-08
AR064736A1 (es) 2009-04-22
BRPI0806468A2 (pt) 2011-09-27
ATE531710T1 (de) 2011-11-15
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KR20090104092A (ko) 2009-10-05
NZ578144A (en) 2011-03-31
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MX2009007180A (es) 2009-07-15
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IL199680A0 (en) 2010-04-15
MA31084B1 (fr) 2010-01-04
HK1135704A1 (en) 2010-06-11
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RS52168B (sr) 2012-08-31

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