HK95697A - 5-HT1-like receptor agonist for rectal administration - Google Patents

5-HT1-like receptor agonist for rectal administration

Info

Publication number
HK95697A
HK95697A HK95697A HK95697A HK95697A HK 95697 A HK95697 A HK 95697A HK 95697 A HK95697 A HK 95697A HK 95697 A HK95697 A HK 95697A HK 95697 A HK95697 A HK 95697A
Authority
HK
Hong Kong
Prior art keywords
pct
receptor agonist
rectal administration
sec
date
Prior art date
Application number
HK95697A
Other languages
English (en)
Inventor
Nadine Merlet
Isabelle Richard
Isabelle Thielemans
Original Assignee
Glaxo Wellcome Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Wellcome Lab filed Critical Glaxo Wellcome Lab
Publication of HK95697A publication Critical patent/HK95697A/xx

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
HK95697A 1992-05-07 1997-06-26 5-HT1-like receptor agonist for rectal administration HK95697A (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929209882A GB9209882D0 (en) 1992-05-07 1992-05-07 Compositions

Publications (1)

Publication Number Publication Date
HK95697A true HK95697A (en) 1997-08-08

Family

ID=10715158

Family Applications (1)

Application Number Title Priority Date Filing Date
HK95697A HK95697A (en) 1992-05-07 1997-06-26 5-HT1-like receptor agonist for rectal administration

Country Status (33)

Country Link
US (1) US5705506A (bg)
EP (1) EP0639072B1 (bg)
JP (1) JPH07506570A (bg)
KR (1) KR100253111B1 (bg)
AT (1) ATE163850T1 (bg)
AU (1) AU670083B2 (bg)
BE (1) BE1007024A5 (bg)
BG (1) BG62120B1 (bg)
BR (1) BR1100108A (bg)
CA (1) CA2135179C (bg)
CH (1) CH685920A5 (bg)
CY (1) CY2039B1 (bg)
CZ (1) CZ283512B6 (bg)
DE (1) DE69317418T2 (bg)
ES (1) ES2113533T3 (bg)
FR (1) FR2690847B1 (bg)
GB (2) GB9209882D0 (bg)
GR (1) GR3026584T3 (bg)
HK (1) HK95697A (bg)
HU (2) HU227338B1 (bg)
IE (1) IE75203B1 (bg)
IL (1) IL105468A (bg)
IT (1) IT1261471B (bg)
NO (1) NO306700B1 (bg)
NZ (1) NZ252132A (bg)
OA (1) OA10109A (bg)
RO (1) RO112993B1 (bg)
RU (1) RU2118527C1 (bg)
SG (1) SG46649A1 (bg)
TW (1) TW231970B (bg)
UA (1) UA37206C2 (bg)
WO (1) WO1993021916A1 (bg)
ZA (1) ZA933178B (bg)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
AU2434297A (en) * 1996-05-23 1997-12-09 Alcon Laboratories, Inc. The use of 5-ht1b/1d agonists to treat ocular pain
US7189753B1 (en) 1997-11-06 2007-03-13 Cady Roger K Preemptive prophylaxis of migraine
ES2367294T3 (es) * 1998-03-26 2011-11-02 Astellas Pharma Inc. Preparación de liberación sostenida de un compuesto macrólido como tacrolimus.
WO2000051624A2 (en) * 1999-03-05 2000-09-08 The Trustees Of University Technology Corporation Methods and compositions useful in inhibiting apoptosis
PL2124556T3 (pl) 2006-10-09 2015-02-27 Charleston Laboratories Inc Kompozycje farmaceutyczne
JP5714910B2 (ja) 2008-01-09 2015-05-07 チャールストン ラボラトリーズ，インコーポレイテッド 薬学的組成物
WO2011006012A1 (en) 2009-07-08 2011-01-13 Charleston Laboratories Inc. Pharmaceutical compositions
KR101825972B1 (ko) 2010-10-15 2018-02-06 콘테라 파르마 에이피에스 운동 장애 치료를 위한 세로토닌 수용체 작용제의 조합
US10561618B2 (en) 2012-04-18 2020-02-18 Contera Pharma Aps Orally available pharmaceutical formulation suitable for improved management of movement disorders
JP2019507181A (ja) 2016-03-04 2019-03-14 チャールストン ラボラトリーズ，インコーポレイテッド 医薬組成物
KR102443161B1 (ko) 2016-07-11 2022-09-14 콘테라 파르마 에이/에스 아침 운동 불능을 치료하기 위한 박동성 약물 전달 시스템

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1171450B (it) * 1980-08-12 1987-06-10 Glaxo Group Ltd Composti eterociclici indolici, procedimento per produrli e composizioni farmaceutiche che li contengono
ZW19381A1 (en) * 1980-08-12 1983-03-09 Glaxo Group Ltd Heterocyclic compounds
GB2082175B (en) * 1980-08-12 1984-05-02 Glaxo Group Ltd Heterocyclic compounds
GR79215B (bg) * 1982-06-07 1984-10-22 Glaxo Group Ltd
GB8332435D0 (en) * 1983-12-06 1984-01-11 Glaxo Group Ltd Chemical compounds
GB2162522B (en) * 1984-08-01 1988-02-24 Glaxo Group Ltd An indole derivative
GB8419575D0 (en) * 1984-08-01 1984-09-05 Glaxo Group Ltd Chemical compounds
FR2574077A1 (fr) * 1984-12-04 1986-06-06 Glaxo Group Ltd Derives d'indoles, leur preparation et les compositions pharmaceutiques les contenant
GB8431426D0 (en) * 1984-12-13 1985-01-23 Glaxo Group Ltd Chemical compounds
DE3678805D1 (de) * 1985-11-08 1991-05-23 Glaxo Group Ltd Indolderivate.
PT88255B (pt) * 1987-08-13 1995-03-01 Glaxo Group Ltd Processo para a preparacao de derivados do indole
PT97888B (pt) * 1990-06-07 1998-12-31 Zeneca Ltd Processo para a preparacao de compostos heterociclicos derivados de indol e de composicoes farmaceuticas que os contem

Also Published As

Publication number Publication date
US5705506A (en) 1998-01-06
BG62120B1 (bg) 1999-03-31
BE1007024A5 (fr) 1995-02-21
NZ252132A (en) 1996-09-25
IE75203B1 (en) 1997-08-27
NO306700B1 (no) 1999-12-13
GB2266665A (en) 1993-11-10
FR2690847B1 (fr) 1995-06-09
RO112993B1 (ro) 1998-03-30
ITRM930286A1 (it) 1994-11-06
IT1261471B (it) 1996-05-23
CZ283512B6 (cs) 1998-04-15
NO944214L (no) 1994-11-07
DE69317418D1 (de) 1998-04-16
CY2039B1 (en) 1998-04-30
HUT71418A (en) 1995-11-28
AU670083B2 (en) 1996-07-04
OA10109A (en) 1996-12-18
HU227338B1 (en) 2011-04-28
CA2135179A1 (en) 1993-11-11
BG99167A (bg) 1995-06-30
EP0639072A1 (en) 1995-02-22
SG46649A1 (en) 1998-02-20
FR2690847A1 (fr) 1993-11-12
HU211638A9 (en) 1995-12-28
TW231970B (bg) 1994-10-11
GB9209882D0 (en) 1992-06-24
GR3026584T3 (en) 1998-07-31
RU2118527C1 (ru) 1998-09-10
JPH07506570A (ja) 1995-07-20
EP0639072B1 (en) 1998-03-11
BR1100108A (pt) 1999-12-07
ATE163850T1 (de) 1998-03-15
IE930339A1 (en) 1993-11-17
CA2135179C (en) 2000-12-05
ITRM930286A0 (it) 1993-05-06
WO1993021916A1 (en) 1993-11-11
ES2113533T3 (es) 1998-05-01
CH685920A5 (fr) 1995-11-15
IL105468A0 (en) 1993-08-18
CZ272394A3 (en) 1995-10-18
NO944214D0 (no) 1994-11-04
DE69317418T2 (de) 1998-07-30
UA37206C2 (uk) 2001-05-15
ZA933178B (en) 1994-01-10
GB2266665B (en) 1996-05-22
AU4064093A (en) 1993-11-29
KR100253111B1 (en) 2000-07-01
IL105468A (en) 1998-09-24
GB9309209D0 (en) 1993-06-16

Similar Documents

Publication Publication Date Title
IL127244A (en) Substituted amines, methods of their preparation and pharmaceutical compositions containing them
EP0903349A3 (en) CCR-3 receptor antagonists
ES2160949T3 (es) Derivados de fenilen-sulfonamida sustituidos en meta.
CA2366268A1 (en) Pharmaceutical compositions for cns and other disorders
DK0641328T3 (da) Broforbundne, azabicykliske derivater som substans P-antagonister
MX9301032A (es) Compuestos farmaceuticos y procedimento para su preparacion
BG105534A (bg) 5ht1 средство и метод за лечение на мигрена
ZA971279B (en) Use of 5ht4 receptor antagonists for overcoming gastrointestinal effects of serotonin reuptake inhinitors
MX9505065A (es) Composicion farmaceutica, aplicable oralmente.
GB2266665B (en) 5-HT1-like receptor agonist for rectal administration
MX9505064A (es) Composicion farmaceutica, aplicable oralmente.
ZA922297B (en) Crystalline tiababine monohydrate,its preparation and use
WO2000000198A8 (en) Piperidine derivatives having effects on serotonin related systems
NO944781D0 (no) 2,5-diokso-2,5-dihydro-1H-benz(b)azepiner som NMDA-reseptor-antagonister
PL350568A1 (en) N-(2-phenyl-4-aminobutyl)-1-naphtamides as antagonists of neurokinin 1 receptors
AU7681198A (en) Novel compounds
BG102229A (bg) Антагонисти на ендотелинови рецептори
TW371661B (en) Novel intermediates and their use to prepare N,N'-bridged bisindolylmaleimides
HU9500175D0 (en) Pharmacologically active alpha-[tertiary-aminomethyl]-benzenemethanol derivatives
ATE162946T1 (de) Pharmazeutische zusammensetzungen enthaltend contignasterol-verbindungen
UA30798A (uk) Спосіб пролонгованої терапії онкологічних хворих

Legal Events

Date Code Title Description
PF Patent in force
PC Patent ceased (i.e. patent has lapsed due to the failure to pay the renewal fee)

Effective date: 20090505