ATE163850T1 - Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen - Google Patents

Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen

Info

Publication number
ATE163850T1
ATE163850T1 AT93909884T AT93909884T ATE163850T1 AT E163850 T1 ATE163850 T1 AT E163850T1 AT 93909884 T AT93909884 T AT 93909884T AT 93909884 T AT93909884 T AT 93909884T AT E163850 T1 ATE163850 T1 AT E163850T1
Authority
AT
Austria
Prior art keywords
pct
rectal administration
agonistic
pharmaceutical compositions
sec
Prior art date
Application number
AT93909884T
Other languages
English (en)
Inventor
Nadine Merlet
Isabelle Richard
Isabelle Thielemans
Original Assignee
Glaxo Wellcome Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Wellcome Lab filed Critical Glaxo Wellcome Lab
Application granted granted Critical
Publication of ATE163850T1 publication Critical patent/ATE163850T1/de

Links

Classifications

    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00Medicinal preparations characterised by special physical form
    • A61K9/02Suppositories; Bougies; Bases therefor; Ovules
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61KPREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00Medicinal preparations containing organic active ingredients
    • A61K31/33Heterocyclic compounds
    • A61K31/395Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445Non condensed piperidines, e.g. piperocaine
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/04Centrally acting analgesics, e.g. opioids
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00Drugs for disorders of the nervous system
    • A61P25/06Antimigraine agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
AT93909884T 1992-05-07 1993-05-03 Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen ATE163850T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929209882A GB9209882D0 (en) 1992-05-07 1992-05-07 Compositions

Publications (1)

Publication Number Publication Date
ATE163850T1 true ATE163850T1 (de) 1998-03-15

Family

ID=10715158

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93909884T ATE163850T1 (de) 1992-05-07 1993-05-03 Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen

Country Status (33)

Country Link
US (1) US5705506A (de)
EP (1) EP0639072B1 (de)
JP (1) JPH07506570A (de)
KR (1) KR100253111B1 (de)
AT (1) ATE163850T1 (de)
AU (1) AU670083B2 (de)
BE (1) BE1007024A5 (de)
BG (1) BG62120B1 (de)
BR (1) BR1100108A (de)
CA (1) CA2135179C (de)
CH (1) CH685920A5 (de)
CY (1) CY2039B1 (de)
CZ (1) CZ283512B6 (de)
DE (1) DE69317418T2 (de)
ES (1) ES2113533T3 (de)
FR (1) FR2690847B1 (de)
GB (2) GB9209882D0 (de)
GR (1) GR3026584T3 (de)
HK (1) HK95697A (de)
HU (2) HU227338B1 (de)
IE (1) IE75203B1 (de)
IL (1) IL105468A (de)
IT (1) IT1261471B (de)
NO (1) NO306700B1 (de)
NZ (1) NZ252132A (de)
OA (1) OA10109A (de)
RO (1) RO112993B1 (de)
RU (1) RU2118527C1 (de)
SG (1) SG46649A1 (de)
TW (1) TW231970B (de)
UA (1) UA37206C2 (de)
WO (1) WO1993021916A1 (de)
ZA (1) ZA933178B (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997044062A1 (en) * 1996-05-23 1997-11-27 Alcon Laboratories, Inc. The use of 5-ht1b/1d agonists to treat ocular pain
US7189753B1 (en) 1997-11-06 2007-03-13 Cady Roger K Preemptive prophylaxis of migraine
ATE464900T1 (de) * 1998-03-26 2010-05-15 Astellas Pharma Inc Retardpräparat mit makroliden wie tacrolimus
AU3731400A (en) * 1999-03-05 2000-09-21 Trustees Of University Technology Corporation, The Methods and compositions useful in inhibiting apoptosis
EP2813144A1 (de) 2006-10-09 2014-12-17 Charleston Laboratories, Inc. Analgetische Zusammensetzungen enthaltend ein Antihistamin
ES2620672T3 (es) 2008-01-09 2017-06-29 Charleston Laboratories, Inc. Comprimidos de doble capa que comprenden oxicodona y prometazina
WO2011006012A1 (en) 2009-07-08 2011-01-13 Charleston Laboratories Inc. Pharmaceutical compositions
BR112013009004B1 (pt) 2010-10-15 2022-05-10 Contera Pharma Aps Uso de composição farmacêutica ou kit de partes compreendendo combinações de agonistas dereceptor de serotonina
BR112014025907B1 (pt) 2012-04-18 2023-02-14 Contera Pharma Aps Formulação farmacêutica disponível para administração por via oral adequada para manejo aprimorado de transtornos do movimento
EP3423041A4 (de) 2016-03-04 2019-09-11 Charleston Laboratories, Inc. Pharmazeutische zusammensetzungen
WO2018011181A1 (en) 2016-07-11 2018-01-18 Contera Pharma Aps Pulsatile drug delivery system for treating morning akinesia

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2082175B (en) * 1980-08-12 1984-05-02 Glaxo Group Ltd Heterocyclic compounds
ZW19381A1 (en) * 1980-08-12 1983-03-09 Glaxo Group Ltd Heterocyclic compounds
AU550010B2 (en) * 1980-08-12 1986-02-27 Glaxo Group Limited 5-tryptaminoacetamides, carbamates and ureas
GR79215B (de) * 1982-06-07 1984-10-22 Glaxo Group Ltd
HU196752B (en) * 1983-12-06 1989-01-30 Glaxo Group Ltd Process for production of medical compositions containing indole-derivatives and these compounds
GB2162522B (en) * 1984-08-01 1988-02-24 Glaxo Group Ltd An indole derivative
GB8419575D0 (en) * 1984-08-01 1984-09-05 Glaxo Group Ltd Chemical compounds
GB2168973B (en) * 1984-12-04 1988-02-03 Glaxo Group Ltd Indole derivatives
GB8431426D0 (en) * 1984-12-13 1985-01-23 Glaxo Group Ltd Chemical compounds
DE3678805D1 (de) * 1985-11-08 1991-05-23 Glaxo Group Ltd Indolderivate.
US4997841A (en) * 1987-08-13 1991-03-05 Glaxo Group Limited Indole derivatives
CA2064815C (en) * 1990-06-07 1999-11-16 Alan Duncan Robertson Therapeutic heterocyclic compounds

Also Published As

Publication number Publication date
CY2039B1 (en) 1998-04-30
RU2118527C1 (ru) 1998-09-10
GB9209882D0 (en) 1992-06-24
IE930339A1 (en) 1993-11-17
CH685920A5 (fr) 1995-11-15
EP0639072B1 (de) 1998-03-11
NO944214L (no) 1994-11-07
ES2113533T3 (es) 1998-05-01
AU670083B2 (en) 1996-07-04
HU227338B1 (en) 2011-04-28
ITRM930286A1 (it) 1994-11-06
WO1993021916A1 (en) 1993-11-11
DE69317418T2 (de) 1998-07-30
SG46649A1 (en) 1998-02-20
CZ283512B6 (cs) 1998-04-15
FR2690847A1 (fr) 1993-11-12
GB2266665B (en) 1996-05-22
KR100253111B1 (en) 2000-07-01
HUT71418A (en) 1995-11-28
FR2690847B1 (fr) 1995-06-09
OA10109A (en) 1996-12-18
GB9309209D0 (en) 1993-06-16
CA2135179C (en) 2000-12-05
DE69317418D1 (de) 1998-04-16
GR3026584T3 (en) 1998-07-31
EP0639072A1 (de) 1995-02-22
US5705506A (en) 1998-01-06
NO306700B1 (no) 1999-12-13
BR1100108A (pt) 1999-12-07
BG99167A (bg) 1995-06-30
NZ252132A (en) 1996-09-25
IL105468A0 (en) 1993-08-18
JPH07506570A (ja) 1995-07-20
TW231970B (de) 1994-10-11
CZ272394A3 (en) 1995-10-18
UA37206C2 (uk) 2001-05-15
ZA933178B (en) 1994-01-10
IL105468A (en) 1998-09-24
CA2135179A1 (en) 1993-11-11
NO944214D0 (no) 1994-11-04
IT1261471B (it) 1996-05-23
RO112993B1 (ro) 1998-03-30
AU4064093A (en) 1993-11-29
BG62120B1 (bg) 1999-03-31
IE75203B1 (en) 1997-08-27
GB2266665A (en) 1993-11-10
BE1007024A5 (fr) 1995-02-21
HU211638A9 (en) 1995-12-28
HK95697A (en) 1997-08-08
ITRM930286A0 (it) 1993-05-06

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UEP Publication of translation of european patent specification