ATE163850T1 - Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen - Google Patents

Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen

Info

Publication number
ATE163850T1
ATE163850T1 AT93909884T AT93909884T ATE163850T1 AT E163850 T1 ATE163850 T1 AT E163850T1 AT 93909884 T AT93909884 T AT 93909884T AT 93909884 T AT93909884 T AT 93909884T AT E163850 T1 ATE163850 T1 AT E163850T1
Authority
AT
Austria
Prior art keywords
pct
rectal administration
agonistic
pharmaceutical compositions
sec
Prior art date
Application number
AT93909884T
Other languages
English (en)
Inventor
Nadine Merlet
Isabelle Richard
Isabelle Thielemans
Original Assignee
Glaxo Wellcome Lab
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Wellcome Lab filed Critical Glaxo Wellcome Lab
Application granted granted Critical
Publication of ATE163850T1 publication Critical patent/ATE163850T1/de

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Organic Chemistry (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Engineering & Computer Science (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Indole Compounds (AREA)
AT93909884T 1992-05-07 1993-05-03 Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen ATE163850T1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB929209882A GB9209882D0 (en) 1992-05-07 1992-05-07 Compositions

Publications (1)

Publication Number Publication Date
ATE163850T1 true ATE163850T1 (de) 1998-03-15

Family

ID=10715158

Family Applications (1)

Application Number Title Priority Date Filing Date
AT93909884T ATE163850T1 (de) 1992-05-07 1993-05-03 Pharmazeutische zusammensetzungen von 5ht1 agonistischen alkyl sulphonamidenfür rektale verabreichungen

Country Status (33)

Country Link
US (1) US5705506A (de)
EP (1) EP0639072B1 (de)
JP (1) JPH07506570A (de)
KR (1) KR100253111B1 (de)
AT (1) ATE163850T1 (de)
AU (1) AU670083B2 (de)
BE (1) BE1007024A5 (de)
BG (1) BG62120B1 (de)
BR (1) BR1100108A (de)
CA (1) CA2135179C (de)
CH (1) CH685920A5 (de)
CY (1) CY2039B1 (de)
CZ (1) CZ283512B6 (de)
DE (1) DE69317418T2 (de)
ES (1) ES2113533T3 (de)
FR (1) FR2690847B1 (de)
GB (2) GB9209882D0 (de)
GR (1) GR3026584T3 (de)
HK (1) HK95697A (de)
HU (2) HU227338B1 (de)
IE (1) IE75203B1 (de)
IL (1) IL105468A (de)
IT (1) IT1261471B (de)
NO (1) NO306700B1 (de)
NZ (1) NZ252132A (de)
OA (1) OA10109A (de)
RO (1) RO112993B1 (de)
RU (1) RU2118527C1 (de)
SG (1) SG46649A1 (de)
TW (1) TW231970B (de)
UA (1) UA37206C2 (de)
WO (1) WO1993021916A1 (de)
ZA (1) ZA933178B (de)

Families Citing this family (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997044062A1 (en) * 1996-05-23 1997-11-27 Alcon Laboratories, Inc. The use of 5-ht1b/1d agonists to treat ocular pain
US7189753B1 (en) 1997-11-06 2007-03-13 Cady Roger K Preemptive prophylaxis of migraine
KR100440553B1 (ko) * 1998-03-26 2004-07-15 후지사와 야꾸힝 고교 가부시키가이샤 서방성 제제
AU3731400A (en) * 1999-03-05 2000-09-21 Trustees Of University Technology Corporation, The Methods and compositions useful in inhibiting apoptosis
AR056690A1 (es) * 2005-10-14 2007-10-17 Athersys Inc Derivados de indol como inhibidores de indol como inhibidores del receptor 3 de histamina para el tartamiento de trastornos del sueno y cognitivos obesidad y otros trastornos de snc
EP2813144A1 (de) 2006-10-09 2014-12-17 Charleston Laboratories, Inc. Analgetische Zusammensetzungen enthaltend ein Antihistamin
EP3090743A1 (de) 2008-01-09 2016-11-09 Charleston Laboratories, Inc. Pharmazeutische zusammensetzungen
CA2767576C (en) 2009-07-08 2020-03-10 Charleston Laboratories Inc. Pharmaceutical compositions comprising an antiemetic and an opioid analgesic
CA2813648C (en) 2010-10-15 2019-06-25 Concit Pharma Aps Combinations of serotonin receptor agonists for treatment of movement disorders
SG11201406690SA (en) 2012-04-18 2014-11-27 Contera Pharma Aps Orally available pharmaceutical formulation suitable for improved management of movement disorders
EP3423041A4 (de) 2016-03-04 2019-09-11 Charleston Laboratories, Inc. Pharmazeutische zusammensetzungen
CN109689036A (zh) 2016-07-11 2019-04-26 康特拉医药公司 用于治疗早晨运动不能的脉冲药物输送系统

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2082175B (en) * 1980-08-12 1984-05-02 Glaxo Group Ltd Heterocyclic compounds
ZW19381A1 (en) * 1980-08-12 1983-03-09 Glaxo Group Ltd Heterocyclic compounds
FR2488606A1 (fr) * 1980-08-12 1982-02-19 Glaxo Group Ltd Derives indoliques, leur preparation et leurs applications en tant que medicaments
GR79215B (de) * 1982-06-07 1984-10-22 Glaxo Group Ltd
GB8332435D0 (en) * 1983-12-06 1984-01-11 Glaxo Group Ltd Chemical compounds
GB8419575D0 (en) * 1984-08-01 1984-09-05 Glaxo Group Ltd Chemical compounds
GB2162522B (en) * 1984-08-01 1988-02-24 Glaxo Group Ltd An indole derivative
SE8505715L (sv) * 1984-12-04 1986-06-05 Glaxo Group Ltd Indolderivat
GB8431426D0 (en) * 1984-12-13 1985-01-23 Glaxo Group Ltd Chemical compounds
DE3678805D1 (de) * 1985-11-08 1991-05-23 Glaxo Group Ltd Indolderivate.
IL87437A0 (en) * 1987-08-13 1989-01-31 Glaxo Group Ltd Indole derivatives,their preparation and pharmaceutical compositions containing them
SI9111010B (sl) * 1990-06-07 2005-02-28 Astrazeneca Ab 3,5-disubstituirani indolni derivati kot "5-HT1-podobni" receptorski agonisti

Also Published As

Publication number Publication date
NO944214D0 (no) 1994-11-04
FR2690847A1 (fr) 1993-11-12
DE69317418T2 (de) 1998-07-30
IL105468A (en) 1998-09-24
CZ283512B6 (cs) 1998-04-15
BR1100108A (pt) 1999-12-07
IL105468A0 (en) 1993-08-18
WO1993021916A1 (en) 1993-11-11
ZA933178B (en) 1994-01-10
TW231970B (de) 1994-10-11
OA10109A (en) 1996-12-18
EP0639072A1 (de) 1995-02-22
GR3026584T3 (en) 1998-07-31
JPH07506570A (ja) 1995-07-20
CA2135179C (en) 2000-12-05
AU670083B2 (en) 1996-07-04
GB2266665B (en) 1996-05-22
SG46649A1 (en) 1998-02-20
CZ272394A3 (en) 1995-10-18
NO306700B1 (no) 1999-12-13
RO112993B1 (ro) 1998-03-30
BG62120B1 (bg) 1999-03-31
HK95697A (en) 1997-08-08
IT1261471B (it) 1996-05-23
FR2690847B1 (fr) 1995-06-09
HU227338B1 (en) 2011-04-28
NZ252132A (en) 1996-09-25
ITRM930286A1 (it) 1994-11-06
AU4064093A (en) 1993-11-29
EP0639072B1 (de) 1998-03-11
GB2266665A (en) 1993-11-10
IE75203B1 (en) 1997-08-27
US5705506A (en) 1998-01-06
BE1007024A5 (fr) 1995-02-21
CH685920A5 (fr) 1995-11-15
BG99167A (bg) 1995-06-30
GB9309209D0 (en) 1993-06-16
NO944214L (no) 1994-11-07
ITRM930286A0 (it) 1993-05-06
RU2118527C1 (ru) 1998-09-10
IE930339A1 (en) 1993-11-17
HUT71418A (en) 1995-11-28
HU211638A9 (en) 1995-12-28
CY2039B1 (en) 1998-04-30
GB9209882D0 (en) 1992-06-24
ES2113533T3 (es) 1998-05-01
CA2135179A1 (en) 1993-11-11
DE69317418D1 (de) 1998-04-16
UA37206C2 (uk) 2001-05-15
KR100253111B1 (en) 2000-07-01

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