KR100253111B1 - Pharmaceutical compositions of alkylsulphonamides 5ht1 agonists for rectal administration - Google Patents

Pharmaceutical compositions of alkylsulphonamides 5ht1 agonists for rectal administration Download PDF

Info

Publication number
KR100253111B1
KR100253111B1 KR1019940703950A KR19940703950A KR100253111B1 KR 100253111 B1 KR100253111 B1 KR 100253111B1 KR 1019940703950 A KR1019940703950 A KR 1019940703950A KR 19940703950 A KR19940703950 A KR 19940703950A KR 100253111 B1 KR100253111 B1 KR 100253111B1
Authority
KR
South Korea
Prior art keywords
pct
rectal administration
alkylsulphonamides
agonists
pharmaceutical compositions
Prior art date
Application number
KR1019940703950A
Other languages
English (en)
Inventor
Nadine Merlet
Isabelle Richard
Isabelle Thielemans
Original Assignee
Glaxo Lab Sa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Lab Sa filed Critical Glaxo Lab Sa
Application granted granted Critical
Publication of KR100253111B1 publication Critical patent/KR100253111B1/ko

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/02—Suppositories; Bougies; Bases therefor; Ovules
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/40—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having five-membered rings with one nitrogen as the only ring hetero atom, e.g. sulpiride, succinimide, tolmetin, buflomedil
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A61K31/445—Non condensed piperidines, e.g. piperocaine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/04—Centrally acting analgesics, e.g. opioids
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/06—Antimigraine agents

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Epidemiology (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Chemical & Material Sciences (AREA)
  • Pain & Pain Management (AREA)
  • Biomedical Technology (AREA)
  • Neurology (AREA)
  • Neurosurgery (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Medicinal Preparation (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Compositions Of Macromolecular Compounds (AREA)
KR1019940703950A 1992-05-07 1994-11-05 Pharmaceutical compositions of alkylsulphonamides 5ht1 agonists for rectal administration KR100253111B1 (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB929209882A GB9209882D0 (en) 1992-05-07 1992-05-07 Compositions
PCT/EP1993/001077 WO1993021916A1 (en) 1992-05-07 1993-05-03 Pharmaceutical compositions of alkylsulphonamides 5ht1 agonists for rectal administration

Publications (1)

Publication Number Publication Date
KR100253111B1 true KR100253111B1 (en) 2000-07-01

Family

ID=10715158

Family Applications (1)

Application Number Title Priority Date Filing Date
KR1019940703950A KR100253111B1 (en) 1992-05-07 1994-11-05 Pharmaceutical compositions of alkylsulphonamides 5ht1 agonists for rectal administration

Country Status (33)

Country Link
US (1) US5705506A (ko)
EP (1) EP0639072B1 (ko)
JP (1) JPH07506570A (ko)
KR (1) KR100253111B1 (ko)
AT (1) ATE163850T1 (ko)
AU (1) AU670083B2 (ko)
BE (1) BE1007024A5 (ko)
BG (1) BG62120B1 (ko)
BR (1) BR1100108A (ko)
CA (1) CA2135179C (ko)
CH (1) CH685920A5 (ko)
CY (1) CY2039B1 (ko)
CZ (1) CZ283512B6 (ko)
DE (1) DE69317418T2 (ko)
ES (1) ES2113533T3 (ko)
FR (1) FR2690847B1 (ko)
GB (2) GB9209882D0 (ko)
GR (1) GR3026584T3 (ko)
HK (1) HK95697A (ko)
HU (2) HU227338B1 (ko)
IE (1) IE75203B1 (ko)
IL (1) IL105468A (ko)
IT (1) IT1261471B (ko)
NO (1) NO306700B1 (ko)
NZ (1) NZ252132A (ko)
OA (1) OA10109A (ko)
RO (1) RO112993B1 (ko)
RU (1) RU2118527C1 (ko)
SG (1) SG46649A1 (ko)
TW (1) TW231970B (ko)
UA (1) UA37206C2 (ko)
WO (1) WO1993021916A1 (ko)
ZA (1) ZA933178B (ko)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
WO1997044062A1 (en) * 1996-05-23 1997-11-27 Alcon Laboratories, Inc. The use of 5-ht1b/1d agonists to treat ocular pain
US7189753B1 (en) 1997-11-06 2007-03-13 Cady Roger K Preemptive prophylaxis of migraine
PT1421939E (pt) * 1998-03-26 2010-07-12 Astellas Pharma Inc Preparaã†o da libertaã†o sustentada de um composto de macrëlido como tracolimus
AU3731400A (en) * 1999-03-05 2000-09-21 Trustees Of University Technology Corporation, The Methods and compositions useful in inhibiting apoptosis
ES2524556T3 (es) 2006-10-09 2014-12-10 Charleston Laboratories, Inc. Composiciones farmacéuticas
CA2905541C (en) 2008-01-09 2020-02-11 Charleston Laboratories, Inc. Pharmaceutical compositions comprising an antiemetic and an opioid analgesic
WO2011006012A1 (en) 2009-07-08 2011-01-13 Charleston Laboratories Inc. Pharmaceutical compositions
HUE031661T2 (en) 2010-10-15 2017-07-28 Contera Pharma Aps Combinations of serotonin receptor agonists for the treatment of movement disorders
NZ700474A (en) 2012-04-18 2016-10-28 Contera Pharma Aps Orally available pharmaceutical formulation suitable for improved management of movement disorders
EP3423041A4 (en) 2016-03-04 2019-09-11 Charleston Laboratories, Inc. PHARMACEUTICAL COMPOSITIONS
CN109689036A (zh) 2016-07-11 2019-04-26 康特拉医药公司 用于治疗早晨运动不能的脉冲药物输送系统

Family Cites Families (12)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB2082175B (en) * 1980-08-12 1984-05-02 Glaxo Group Ltd Heterocyclic compounds
FR2488606A1 (fr) * 1980-08-12 1982-02-19 Glaxo Group Ltd Derives indoliques, leur preparation et leurs applications en tant que medicaments
ZW19381A1 (en) * 1980-08-12 1983-03-09 Glaxo Group Ltd Heterocyclic compounds
IT1170387B (it) * 1982-06-07 1987-06-03 Glaxo Group Ltd Composti eterociclici, procedimento per prepararli e composizioni farmaceutiche che li contengono
GB8332435D0 (en) * 1983-12-06 1984-01-11 Glaxo Group Ltd Chemical compounds
GB8419575D0 (en) * 1984-08-01 1984-09-05 Glaxo Group Ltd Chemical compounds
GB2162522B (en) * 1984-08-01 1988-02-24 Glaxo Group Ltd An indole derivative
AU584142B2 (en) * 1984-12-04 1989-05-18 Glaxo Group Limited Indole derivatives
GB8431426D0 (en) * 1984-12-13 1985-01-23 Glaxo Group Ltd Chemical compounds
DE3678805D1 (de) * 1985-11-08 1991-05-23 Glaxo Group Ltd Indolderivate.
GB2208646B (en) * 1987-08-13 1991-06-26 Glaxo Group Ltd Indole derivatives
IL114690A (en) * 1990-06-07 1997-02-18 Wellcome Found Antimigraine oxazolidinone substituted indole derivatives

Also Published As

Publication number Publication date
SG46649A1 (en) 1998-02-20
WO1993021916A1 (en) 1993-11-11
HU227338B1 (en) 2011-04-28
HK95697A (en) 1997-08-08
NO306700B1 (no) 1999-12-13
UA37206C2 (uk) 2001-05-15
GB2266665B (en) 1996-05-22
GB9209882D0 (en) 1992-06-24
HU211638A9 (en) 1995-12-28
DE69317418D1 (de) 1998-04-16
GR3026584T3 (en) 1998-07-31
HUT71418A (en) 1995-11-28
BG62120B1 (bg) 1999-03-31
CH685920A5 (fr) 1995-11-15
CZ272394A3 (en) 1995-10-18
FR2690847B1 (fr) 1995-06-09
NO944214L (no) 1994-11-07
IT1261471B (it) 1996-05-23
EP0639072B1 (en) 1998-03-11
OA10109A (en) 1996-12-18
ITRM930286A1 (it) 1994-11-06
BE1007024A5 (fr) 1995-02-21
JPH07506570A (ja) 1995-07-20
IL105468A0 (en) 1993-08-18
IE930339A1 (en) 1993-11-17
ZA933178B (en) 1994-01-10
EP0639072A1 (en) 1995-02-22
BG99167A (bg) 1995-06-30
ATE163850T1 (de) 1998-03-15
RO112993B1 (ro) 1998-03-30
CA2135179C (en) 2000-12-05
DE69317418T2 (de) 1998-07-30
CA2135179A1 (en) 1993-11-11
NO944214D0 (no) 1994-11-04
IL105468A (en) 1998-09-24
CY2039B1 (en) 1998-04-30
IE75203B1 (en) 1997-08-27
AU4064093A (en) 1993-11-29
GB2266665A (en) 1993-11-10
NZ252132A (en) 1996-09-25
FR2690847A1 (fr) 1993-11-12
AU670083B2 (en) 1996-07-04
BR1100108A (pt) 1999-12-07
US5705506A (en) 1998-01-06
TW231970B (ko) 1994-10-11
GB9309209D0 (en) 1993-06-16
RU2118527C1 (ru) 1998-09-10
ITRM930286A0 (it) 1993-05-06
CZ283512B6 (cs) 1998-04-15
ES2113533T3 (es) 1998-05-01

Similar Documents

Publication Publication Date Title
DK0641328T3 (da) Broforbundne, azabicykliske derivater som substans P-antagonister
EP0903349A3 (en) CCR-3 receptor antagonists
AP2001002129A0 (en) 5HT1 receptor agonists and metoclopramide for the treatment of migrane.
ATE331726T1 (de) Adenine-derivate
MX9702865A (es) Agentes estrogenicos.
MY117274A (en) Polycyclic amine compounds and their enantiomers,their method of preparation and pharmaceutical compositions in which they are present.
BG106142A (en) Glucocorticoid receptor modulators
ES2160949T3 (es) Derivados de fenilen-sulfonamida sustituidos en meta.
MY141384A (en) Prevention of loss and restoration of bone mass by certain prostaglandin agonists
MX9301032A (es) Compuestos farmaceuticos y procedimento para su preparacion
ZA971279B (en) Use of 5ht4 receptor antagonists for overcoming gastrointestinal effects of serotonin reuptake inhinitors
KR100253111B1 (en) Pharmaceutical compositions of alkylsulphonamides 5ht1 agonists for rectal administration
IL114598A0 (en) Triazole compounds their preparation and pharmaceutical compositions containing them
IL114600A0 (en) Thiazole and thiadiazole compounds their preparation and pharmaceutical composition containing them
EP0485431A4 (en) Partial agonists of the strychnine insensitive glycine modulatory site of the n-methyl-d-aspartate receptor complex as neuropsychopharmacological agents
GR3022615T3 (en) Pharmaceutical compositions based on ebastime or analogues thereof.
CA2448278A1 (en) Drug delivery system comprising a tetrahidroxilated estrogen for use in hormonal contraception
UA27108A1 (uk) Аhтрацикліhові глікозиди та їх фармацевтичhо прийhятhі кислотhо-адитивhі солі, спосіб їх одержаhhя, похідhі 1,6-дийод-3-оксапеhтаhу та спосіб їх одержаhhя
GR3036195T3 (en) Novel compounds
BG102229A (en) Endothelium receptor antagonists
FR2724933B1 (ko)
TW371661B (en) Novel intermediates and their use to prepare N,N'-bridged bisindolylmaleimides
HU9500175D0 (en) Pharmacologically active alpha-[tertiary-aminomethyl]-benzenemethanol derivatives
EP1051994A3 (en) 5HT1 receptor agonists and a COX-2 inhibitor for the treatment of migraine

Legal Events

Date Code Title Description
A201 Request for examination
E701 Decision to grant or registration of patent right
GRNT Written decision to grant
FPAY Annual fee payment

Payment date: 20090107

Year of fee payment: 10

LAPS Lapse due to unpaid annual fee