HK1170221A1 - Azetidinyl diamides as monoacylglycerol lipase inhibitors - Google Patents

Azetidinyl diamides as monoacylglycerol lipase inhibitors

Info

Publication number
HK1170221A1
HK1170221A1 HK12110778.3A HK12110778A HK1170221A1 HK 1170221 A1 HK1170221 A1 HK 1170221A1 HK 12110778 A HK12110778 A HK 12110778A HK 1170221 A1 HK1170221 A1 HK 1170221A1
Authority
HK
Hong Kong
Prior art keywords
lipase inhibitors
monoacylglycerol lipase
diamides
azetidinyl
azetidinyl diamides
Prior art date
Application number
HK12110778.3A
Other languages
English (en)
Chinese (zh)
Inventor
Haiyan Bian
Kristen M Chevalier
Peter J Connolly
Christopher M Flores
Shu-Chen Lin
Li Liu
John Mabus
Mark J Macielag
Donnell Mark E Mc
Philip M Pitis
Sui-Po Zhang
Yue-Mei Zhang
Bin Zhu
Jose Clemente
Original Assignee
Janssen Pharmaceutica Nv
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Janssen Pharmaceutica Nv filed Critical Janssen Pharmaceutica Nv
Publication of HK1170221A1 publication Critical patent/HK1170221A1/xx

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    • C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
    • C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
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HK12110778.3A 2009-04-22 2012-10-29 Azetidinyl diamides as monoacylglycerol lipase inhibitors HK1170221A1 (en)

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US17165809P 2009-04-22 2009-04-22
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PCT/US2010/032049 WO2010124086A1 (en) 2009-04-22 2010-04-22 Azetidinyl diamides as monoacylglycerol lipase inhibitors

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KR (8) KR20120034616A (ko)
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WO2010011493A1 (en) 2008-07-21 2010-01-28 Novartis Ag Silicone-containing polymeric materals with hydrolyzable groups
EP2421848A1 (en) * 2009-04-22 2012-02-29 Janssen Pharmaceutica N.V. Azetidinyl diamides as monoacylglycerol lipase inhibitors
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US20130102585A1 (en) 2013-04-25
WO2010124086A1 (en) 2010-10-28
KR20110137834A (ko) 2011-12-23
RU2011147230A (ru) 2013-05-27
TW201103930A (en) 2011-02-01
CN102459167B (zh) 2015-04-01
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US20130123233A1 (en) 2013-05-16
KR20120034617A (ko) 2012-04-12
CA2759713A1 (en) 2010-10-28
WO2010124102A1 (en) 2010-10-28
IL215775A0 (en) 2012-01-31
BRPI1014885A2 (pt) 2016-04-19
JP2012524802A (ja) 2012-10-18
US20110015170A1 (en) 2011-01-20
US8445477B2 (en) 2013-05-21
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JP2012524804A (ja) 2012-10-18
US20100331300A1 (en) 2010-12-30
HRP20140295T1 (hr) 2014-04-25
BRPI1014281A2 (pt) 2019-09-24
KR20120035146A (ko) 2012-04-13
ES2455744T3 (es) 2014-04-16
AU2010238732A1 (en) 2011-11-10
CN102459166A (zh) 2012-05-16

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