BRPI1014281A2 - azetidinil diamidas como inibidores da monoacilglicerol lipase - Google Patents
azetidinil diamidas como inibidores da monoacilglicerol lipaseInfo
- Publication number
- BRPI1014281A2 BRPI1014281A2 BRPI1014281A BRPI1014281A BRPI1014281A2 BR PI1014281 A2 BRPI1014281 A2 BR PI1014281A2 BR PI1014281 A BRPI1014281 A BR PI1014281A BR PI1014281 A BRPI1014281 A BR PI1014281A BR PI1014281 A2 BRPI1014281 A2 BR PI1014281A2
- Authority
- BR
- Brazil
- Prior art keywords
- lipase inhibitors
- monoacylglycerol lipase
- diamides
- azetidinyl
- azetidinyl diamides
- Prior art date
Links
Classifications
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/04—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
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- C07—ORGANIC CHEMISTRY
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- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/10—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing aromatic rings
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- C07D205/02—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings
- C07D205/04—Heterocyclic compounds containing four-membered rings with one nitrogen atom as the only ring hetero atom not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
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- C07D409/06—Heterocyclic compounds containing two or more hetero rings, at least one ring having sulfur atoms as the only ring hetero atoms containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
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- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
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- C—CHEMISTRY; METALLURGY
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- C07D491/00—Heterocyclic compounds containing in the condensed ring system both one or more rings having oxygen atoms as the only ring hetero atoms and one or more rings having nitrogen atoms as the only ring hetero atoms, not provided for by groups C07D451/00 - C07D459/00, C07D463/00, C07D477/00 or C07D489/00
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Applications Claiming Priority (3)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
US17164909P | 2009-04-22 | 2009-04-22 | |
US17165809P | 2009-04-22 | 2009-04-22 | |
PCT/US2010/032092 WO2010124116A1 (en) | 2009-04-22 | 2010-04-22 | Azetidinyl diamides as monoacylglycerol lipase inhibitors |
Publications (1)
Publication Number | Publication Date |
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BRPI1014281A2 true BRPI1014281A2 (pt) | 2019-09-24 |
Family
ID=42208680
Family Applications (8)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI1014876A BRPI1014876A2 (pt) | 2009-04-22 | 2010-04-22 | "diamidas de azetidinila como inibidores de monoacilglicerol lipase." |
BRPI1014885A BRPI1014885A8 (pt) | 2009-04-22 | 2010-04-22 | "azetidinil diamidas como inibidores de monoacilglicerol lipase." |
BRPI1015238A BRPI1015238A2 (pt) | 2009-04-22 | 2010-04-22 | diamidas de azetidilina como inibidores de monoaciglicerol lipase |
BRPI1014284A BRPI1014284A2 (pt) | 2009-04-22 | 2010-04-22 | azetidinil diamidas como inibidores da monoacilglicerol lipase |
BRPI1013540-5A BRPI1013540A2 (pt) | 2009-04-22 | 2010-04-22 | azetidinil diamidas como inibidores de monoacilglicerol lipases |
BRPI1013538A BRPI1013538A2 (pt) | 2009-04-22 | 2010-04-22 | azetidinil diamidas como inibidores de monoacilglicerol lipase |
BRPI1014281A BRPI1014281A2 (pt) | 2009-04-22 | 2010-04-22 | azetidinil diamidas como inibidores da monoacilglicerol lipase |
BRPI1013545A BRPI1013545A2 (pt) | 2009-04-22 | 2010-04-22 | azetidinil diamidas como inibidores de monoacilglicerol lipase |
Family Applications Before (6)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI1014876A BRPI1014876A2 (pt) | 2009-04-22 | 2010-04-22 | "diamidas de azetidinila como inibidores de monoacilglicerol lipase." |
BRPI1014885A BRPI1014885A8 (pt) | 2009-04-22 | 2010-04-22 | "azetidinil diamidas como inibidores de monoacilglicerol lipase." |
BRPI1015238A BRPI1015238A2 (pt) | 2009-04-22 | 2010-04-22 | diamidas de azetidilina como inibidores de monoaciglicerol lipase |
BRPI1014284A BRPI1014284A2 (pt) | 2009-04-22 | 2010-04-22 | azetidinil diamidas como inibidores da monoacilglicerol lipase |
BRPI1013540-5A BRPI1013540A2 (pt) | 2009-04-22 | 2010-04-22 | azetidinil diamidas como inibidores de monoacilglicerol lipases |
BRPI1013538A BRPI1013538A2 (pt) | 2009-04-22 | 2010-04-22 | azetidinil diamidas como inibidores de monoacilglicerol lipase |
Family Applications After (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
BRPI1013545A BRPI1013545A2 (pt) | 2009-04-22 | 2010-04-22 | azetidinil diamidas como inibidores de monoacilglicerol lipase |
Country Status (22)
Country | Link |
---|---|
US (16) | US8362000B2 (pt) |
EP (8) | EP2421848A1 (pt) |
JP (8) | JP5733840B2 (pt) |
KR (8) | KR101705697B1 (pt) |
CN (8) | CN102459228A (pt) |
AR (8) | AR076381A1 (pt) |
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2012
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2013
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2014
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Free format text: EM VIRTUDE DO ARQUIVAMENTO PUBLICADO NA RPI 2543 DE 01-10-2019 E CONSIDERANDO AUSENCIA DE MANIFESTACAO DENTRO DOS PRAZOS LEGAIS, INFORMO QUE CABE SER MANTIDO O ARQUIVAMENTO DO PEDIDO DE PATENTE, CONFORME O DISPOSTO NO ARTIGO 12, DA RESOLUCAO 113/2013. |