FI57255C - Foerfarande foer framstaellning av farmakologiskt vaerdefulla 1-alkyl-2-nitro-5-vinyl-imidazoler - Google Patents

Foerfarande foer framstaellning av farmakologiskt vaerdefulla 1-alkyl-2-nitro-5-vinyl-imidazoler Download PDF

Info

Publication number
FI57255C
FI57255C FI1864/72A FI186472A FI57255C FI 57255 C FI57255 C FI 57255C FI 1864/72 A FI1864/72 A FI 1864/72A FI 186472 A FI186472 A FI 186472A FI 57255 C FI57255 C FI 57255C
Authority
FI
Finland
Prior art keywords
nitro
alkyl
vinyl
imidazoler
framework
Prior art date
Application number
FI1864/72A
Other languages
English (en)
Finnish (fi)
Other versions
FI57255B (fi
Inventor
Bruno Cavalleri
Giancarlo Lancini
Original Assignee
Lepetit Spa
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Lepetit Spa filed Critical Lepetit Spa
Application granted granted Critical
Publication of FI57255B publication Critical patent/FI57255B/fi
Publication of FI57255C publication Critical patent/FI57255C/fi

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/04—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings directly linked by a ring-member-to-ring-member bond
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D233/00—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings
    • C07D233/54—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members
    • C07D233/66—Heterocyclic compounds containing 1,3-diazole or hydrogenated 1,3-diazole rings, not condensed with other rings having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D233/91—Nitro radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
FI1864/72A 1971-07-30 1972-06-30 Foerfarande foer framstaellning av farmakologiskt vaerdefulla 1-alkyl-2-nitro-5-vinyl-imidazoler FI57255C (fi)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT4297871 1971-07-30
IT4297871 1971-07-30

Publications (2)

Publication Number Publication Date
FI57255B FI57255B (fi) 1980-03-31
FI57255C true FI57255C (fi) 1980-07-10

Family

ID=11254772

Family Applications (1)

Application Number Title Priority Date Filing Date
FI1864/72A FI57255C (fi) 1971-07-30 1972-06-30 Foerfarande foer framstaellning av farmakologiskt vaerdefulla 1-alkyl-2-nitro-5-vinyl-imidazoler

Country Status (27)

Country Link
US (1) US3954789A (xx)
JP (2) JPS528832B1 (xx)
AR (4) AR199084A1 (xx)
AT (3) AT316545B (xx)
AU (1) AU462723B2 (xx)
BE (1) BE785024A (xx)
CA (1) CA997340A (xx)
CH (4) CH574933A5 (xx)
CS (1) CS180585B2 (xx)
DD (2) DD99996A5 (xx)
DE (2) DE2229248C3 (xx)
DK (1) DK154295C (xx)
ES (3) ES405343A1 (xx)
FI (1) FI57255C (xx)
FR (1) FR2148073B1 (xx)
GB (1) GB1362444A (xx)
HU (2) HU164926B (xx)
IE (1) IE36530B1 (xx)
IL (1) IL39880A (xx)
LU (1) LU65816A1 (xx)
NL (2) NL148602B (xx)
NO (2) NO135592C (xx)
PL (4) PL85190B1 (xx)
RO (6) RO61517A (xx)
SE (3) SE417711B (xx)
SU (4) SU466684A3 (xx)
ZA (1) ZA724723B (xx)

Families Citing this family (9)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1480192A (en) * 1975-01-15 1977-07-20 Lepetit Spa 1-methyl-2-nitro-imidazole-5-methanol derivatives
GB1526451A (en) * 1976-01-27 1978-09-27 Lepetit Spa Alpha,alpha,1-trimethyl-2-nitroimidazole-5-methanol derivatives
US4218460A (en) * 1976-09-29 1980-08-19 Basf Aktiengesellschaft Nitroimidazoles
US4199592A (en) * 1978-08-29 1980-04-22 E. I. Du Pont De Nemours And Company Antiinflammatory 4,5-diaryl-2-nitroimidazoles
ZW24982A1 (en) * 1981-11-30 1983-06-15 Hoffmann La Roche 2-nitroimidazoles
JPH10338673A (ja) * 1997-06-04 1998-12-22 Nippon Bayeragrochem Kk イソニコチン酸ヒドラジド誘導体および有害生物防除剤
ZA200507752B (en) 2003-03-28 2007-01-31 Threshold Pharmaceuticals Inc Compositions and methods for treating cancer
PL1896040T3 (pl) 2005-06-29 2012-12-31 Threshold Pharmaceuticals Inc Proleki alkilatora fosforoamidowego
US8552048B2 (en) 2006-12-26 2013-10-08 Threshold Pharmaceuticals, Inc. Phosphoramidate alkylator prodrugs for the treatment of cancer

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
NL124627C (xx) * 1964-08-12
NL143227B (nl) * 1968-11-15 1974-09-16 Lepetit Spa Werkwijze ter bereiding van imidazoolderivaten met bactericide werking.
US3583985A (en) * 1969-04-09 1971-06-08 Richardson Merrell Inc Nitroimidazolyl nitrones
US3711495A (en) * 1970-01-07 1973-01-16 Merck & Co Inc Isoxazalin-3-yl-substituted-5-nitroimidazoles

Also Published As

Publication number Publication date
CH574933A5 (xx) 1976-04-30
RO61517A (xx) 1976-12-15
DE2229248C3 (de) 1980-03-27
DE2229248A1 (de) 1973-02-15
SU463263A3 (ru) 1975-03-05
AR193999A1 (es) 1973-06-12
SE7503080L (xx) 1975-03-18
NL148602B (nl) 1976-02-16
SE392615B (sv) 1977-04-04
RO63049A (fr) 1978-07-15
RO62787A (xx) 1977-08-15
AR193885A1 (es) 1973-05-31
DE2229223C3 (de) 1975-12-18
AU4422872A (en) 1974-01-10
DK154295B (da) 1988-10-31
SU466684A3 (ru) 1975-04-05
HU164926B (xx) 1974-05-28
CH572040A5 (xx) 1976-01-30
FR2148073B1 (xx) 1975-11-28
DE2229223B2 (de) 1975-05-07
SE417711B (sv) 1981-04-06
CS180585B2 (en) 1978-01-31
NO135592C (xx) 1977-04-27
IL39880A (en) 1976-04-30
PL82980B1 (xx) 1975-12-31
AT316545B (de) 1974-07-10
DE2229223A1 (de) 1973-02-15
BE785024A (fr) 1972-10-16
PL87673B1 (xx) 1976-07-31
NL149491B (nl) 1976-05-17
NL7210340A (xx) 1973-02-01
SU581863A3 (ru) 1977-11-25
DD99995A5 (xx) 1973-09-05
PL84350B1 (xx) 1976-03-31
RO63047A (fr) 1978-05-15
AR199084A1 (es) 1974-08-08
DK154295C (da) 1989-03-28
ES418921A1 (es) 1976-10-16
AT323736B (de) 1975-07-25
NO135591C (xx) 1977-04-27
AU462723B2 (en) 1975-07-03
DE2229248B2 (de) 1979-07-26
ZA724723B (en) 1973-04-25
HU167622B (xx) 1975-11-28
AR199680A1 (es) 1974-09-23
GB1362444A (en) 1974-08-07
NO135592B (xx) 1977-01-17
PL85190B1 (xx) 1976-04-30
LU65816A1 (xx) 1972-11-29
ES405341A1 (es) 1975-07-01
US3954789A (en) 1976-05-04
IL39880A0 (en) 1972-09-28
SE417200B (sv) 1981-03-02
IE36530B1 (en) 1976-11-24
RO63048A (fr) 1978-05-15
NO135591B (xx) 1977-01-17
RO63453A (fr) 1978-06-15
CA997340A (en) 1976-09-21
JPS5038111B1 (xx) 1975-12-06
AT315164B (de) 1974-05-10
FI57255B (fi) 1980-03-31
CH574934A5 (xx) 1976-04-30
JPS528832B1 (xx) 1977-03-11
DD99996A5 (xx) 1973-09-05
CH580596A5 (xx) 1976-10-15
ES405343A1 (es) 1975-07-16
IE36530L (en) 1973-01-30
FR2148073A1 (xx) 1973-03-11
NL7210339A (xx) 1973-02-01
SU567404A3 (ru) 1977-07-30

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