FI120235B - Uusien terapeuttisesti aktiivisten bi- ja trisyklisten aminoalkoholien estereiden valmistusmenetelmä - Google Patents

Uusien terapeuttisesti aktiivisten bi- ja trisyklisten aminoalkoholien estereiden valmistusmenetelmä Download PDF

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Publication number
FI120235B
FI120235B FI934000A FI934000A FI120235B FI 120235 B FI120235 B FI 120235B FI 934000 A FI934000 A FI 934000A FI 934000 A FI934000 A FI 934000A FI 120235 B FI120235 B FI 120235B
Authority
FI
Finland
Prior art keywords
tropanyl
thienyl
eller
methyl
methobromide
Prior art date
Application number
FI934000A
Other languages
English (en)
Finnish (fi)
Swedish (sv)
Other versions
FI934000A0 (fi
FI934000A (fi
Inventor
Rolf Banholzer
Richard Reichl
Rudolf Bauer
Original Assignee
Boehringer Ingelheim Kg
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
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Publication date
Application filed by Boehringer Ingelheim Kg filed Critical Boehringer Ingelheim Kg
Publication of FI934000A0 publication Critical patent/FI934000A0/fi
Publication of FI934000A publication Critical patent/FI934000A/fi
Application granted granted Critical
Publication of FI120235B publication Critical patent/FI120235B/fi

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/14—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing 9-azabicyclo [3.3.1] nonane ring systems, e.g. granatane, 2-aza-adamantane; Cyclic acetals thereof

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
FI934000A 1991-03-15 1993-09-13 Uusien terapeuttisesti aktiivisten bi- ja trisyklisten aminoalkoholien estereiden valmistusmenetelmä FI120235B (fi)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
DE4108393 1991-03-15
DE4108393A DE4108393A1 (de) 1991-03-15 1991-03-15 Neue ester bi- und tricyclischer aminoalkohole, ihre herstellung und ihre verwendung in arzneimitteln
EP9200489 1992-03-05
PCT/EP1992/000489 WO1992016528A1 (fr) 1991-03-15 1992-03-05 Esters nouveaux d'amino-alcools bicycliques et tricycliques, leur preparation et leur utilisation dans des medicaments

Publications (3)

Publication Number Publication Date
FI934000A0 FI934000A0 (fi) 1993-09-13
FI934000A FI934000A (fi) 1993-09-13
FI120235B true FI120235B (fi) 2009-08-14

Family

ID=6427349

Family Applications (1)

Application Number Title Priority Date Filing Date
FI934000A FI120235B (fi) 1991-03-15 1993-09-13 Uusien terapeuttisesti aktiivisten bi- ja trisyklisten aminoalkoholien estereiden valmistusmenetelmä

Country Status (26)

Country Link
US (1) US5654314A (fr)
EP (1) EP0579615B1 (fr)
JP (1) JP3352684B2 (fr)
KR (1) KR100307274B1 (fr)
AT (1) ATE202778T1 (fr)
AU (1) AU662128B2 (fr)
CA (1) CA2105575C (fr)
CZ (1) CZ281509B6 (fr)
DE (2) DE4108393A1 (fr)
DK (1) DK0579615T3 (fr)
ES (1) ES2160577T3 (fr)
FI (1) FI120235B (fr)
GR (1) GR3036792T3 (fr)
HU (1) HU224210B1 (fr)
IE (1) IE920815A1 (fr)
IL (1) IL101225A (fr)
MX (1) MX9201139A (fr)
NO (1) NO304266B1 (fr)
NZ (1) NZ241961A (fr)
PL (1) PL179673B1 (fr)
PT (1) PT100234B (fr)
SG (1) SG43037A1 (fr)
SK (1) SK281511B6 (fr)
UA (1) UA29406C2 (fr)
WO (1) WO1992016528A1 (fr)
ZA (1) ZA921875B (fr)

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Also Published As

Publication number Publication date
FI934000A0 (fi) 1993-09-13
CZ281509B6 (cs) 1996-10-16
WO1992016528A1 (fr) 1992-10-01
IL101225A (en) 1996-05-14
NO933274L (no) 1993-11-12
JPH06505718A (ja) 1994-06-30
HUT65132A (en) 1994-04-28
ES2160577T3 (es) 2001-11-16
NO304266B1 (no) 1998-11-23
KR100307274B1 (ko) 2001-12-05
PT100234A (pt) 1993-07-30
SG43037A1 (en) 1997-10-17
SK281511B6 (sk) 2001-04-09
JP3352684B2 (ja) 2002-12-03
NO933274D0 (no) 1993-09-14
AU662128B2 (en) 1995-08-24
EP0579615A1 (fr) 1994-01-26
ZA921875B (en) 1993-09-13
DE4108393A1 (de) 1992-09-17
EP0579615B1 (fr) 2001-07-04
UA29406C2 (uk) 2000-11-15
IE920815A1 (en) 1992-09-23
CA2105575C (fr) 2000-04-25
SK94993A3 (en) 1994-04-06
CZ191793A3 (en) 1994-05-18
NZ241961A (en) 1995-07-26
IL101225A0 (en) 1992-11-15
DE59209907D1 (de) 2001-08-09
FI934000A (fi) 1993-09-13
DK0579615T3 (da) 2001-09-17
PL179673B1 (pl) 2000-10-31
AU1345792A (en) 1992-10-21
HU9302611D0 (en) 1993-12-28
GR3036792T3 (en) 2002-01-31
ATE202778T1 (de) 2001-07-15
HU224210B1 (hu) 2005-06-28
PT100234B (pt) 1999-06-30
US5654314A (en) 1997-08-05
CA2105575A1 (fr) 1992-09-16
MX9201139A (es) 1992-10-01

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