ZA921875B - New esters of bi- and tricyclic amino alcohols, their preparation and their use in pharmaceutical compositions - Google Patents

New esters of bi- and tricyclic amino alcohols, their preparation and their use in pharmaceutical compositions

Info

Publication number
ZA921875B
ZA921875B ZA921875A ZA921875A ZA921875B ZA 921875 B ZA921875 B ZA 921875B ZA 921875 A ZA921875 A ZA 921875A ZA 921875 A ZA921875 A ZA 921875A ZA 921875 B ZA921875 B ZA 921875B
Authority
ZA
South Africa
Prior art keywords
pharmaceutical compositions
preparation
amino alcohols
new esters
tricyclic amino
Prior art date
Application number
ZA921875A
Other languages
English (en)
Inventor
Rolf Banholzer
Rudolf Bauer
Richard Reichl
Original Assignee
Boehringer Ingelheim Int
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Int filed Critical Boehringer Ingelheim Int
Publication of ZA921875B publication Critical patent/ZA921875B/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/02—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof
    • C07D451/04—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing not further condensed 8-azabicyclo [3.2.1] octane or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane; Cyclic acetals thereof with hetero atoms directly attached in position 3 of the 8-azabicyclo [3.2.1] octane or in position 7 of the 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring system
    • C07D451/06—Oxygen atoms
    • C07D451/10—Oxygen atoms acylated by aliphatic or araliphatic carboxylic acids, e.g. atropine, scopolamine
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P11/00—Drugs for disorders of the respiratory system
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P25/00—Drugs for disorders of the nervous system
    • A61P25/02—Drugs for disorders of the nervous system for peripheral neuropathies
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D451/00—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof
    • C07D451/14—Heterocyclic compounds containing 8-azabicyclo [3.2.1] octane, 9-azabicyclo [3.3.1] nonane, or 3-oxa-9-azatricyclo [3.3.1.0<2,4>] nonane ring systems, e.g. tropane or granatane alkaloids, scopolamine; Cyclic acetals thereof containing 9-azabicyclo [3.3.1] nonane ring systems, e.g. granatane, 2-aza-adamantane; Cyclic acetals thereof

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Animal Behavior & Ethology (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Steroid Compounds (AREA)
  • Medicinal Preparation (AREA)
ZA921875A 1991-03-15 1992-03-13 New esters of bi- and tricyclic amino alcohols, their preparation and their use in pharmaceutical compositions ZA921875B (en)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE4108393A DE4108393A1 (de) 1991-03-15 1991-03-15 Neue ester bi- und tricyclischer aminoalkohole, ihre herstellung und ihre verwendung in arzneimitteln

Publications (1)

Publication Number Publication Date
ZA921875B true ZA921875B (en) 1993-09-13

Family

ID=6427349

Family Applications (1)

Application Number Title Priority Date Filing Date
ZA921875A ZA921875B (en) 1991-03-15 1992-03-13 New esters of bi- and tricyclic amino alcohols, their preparation and their use in pharmaceutical compositions

Country Status (26)

Country Link
US (1) US5654314A (xx)
EP (1) EP0579615B1 (xx)
JP (1) JP3352684B2 (xx)
KR (1) KR100307274B1 (xx)
AT (1) ATE202778T1 (xx)
AU (1) AU662128B2 (xx)
CA (1) CA2105575C (xx)
CZ (1) CZ281509B6 (xx)
DE (2) DE4108393A1 (xx)
DK (1) DK0579615T3 (xx)
ES (1) ES2160577T3 (xx)
FI (1) FI120235B (xx)
GR (1) GR3036792T3 (xx)
HU (1) HU224210B1 (xx)
IE (1) IE920815A1 (xx)
IL (1) IL101225A (xx)
MX (1) MX9201139A (xx)
NO (1) NO304266B1 (xx)
NZ (1) NZ241961A (xx)
PL (1) PL179673B1 (xx)
PT (1) PT100234B (xx)
SG (1) SG43037A1 (xx)
SK (1) SK281511B6 (xx)
UA (1) UA29406C2 (xx)
WO (1) WO1992016528A1 (xx)
ZA (1) ZA921875B (xx)

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US20030229227A1 (en) * 2002-03-16 2003-12-11 Boehringer Ingelheim Pharma Gmbh & Co. Kg New difurylglycolic acid esters, processes for the preparation thereof as well as the use thereof as pharmaceutical compositions
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US7244415B2 (en) * 2002-03-28 2007-07-17 Boehringer Ingelheim Pharma Gmbh & Co. Kg HFA suspension formulations of an anhydrate
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Also Published As

Publication number Publication date
DE4108393A1 (de) 1992-09-17
NO933274D0 (no) 1993-09-14
ES2160577T3 (es) 2001-11-16
JPH06505718A (ja) 1994-06-30
CZ191793A3 (en) 1994-05-18
NZ241961A (en) 1995-07-26
PT100234B (pt) 1999-06-30
AU1345792A (en) 1992-10-21
FI934000A0 (fi) 1993-09-13
CZ281509B6 (cs) 1996-10-16
SK94993A3 (en) 1994-04-06
IL101225A (en) 1996-05-14
ATE202778T1 (de) 2001-07-15
DK0579615T3 (da) 2001-09-17
JP3352684B2 (ja) 2002-12-03
HUT65132A (en) 1994-04-28
EP0579615A1 (de) 1994-01-26
WO1992016528A1 (de) 1992-10-01
PT100234A (pt) 1993-07-30
HU9302611D0 (en) 1993-12-28
UA29406C2 (uk) 2000-11-15
SK281511B6 (sk) 2001-04-09
CA2105575A1 (en) 1992-09-16
SG43037A1 (en) 1997-10-17
PL179673B1 (pl) 2000-10-31
HU224210B1 (hu) 2005-06-28
AU662128B2 (en) 1995-08-24
IE920815A1 (en) 1992-09-23
IL101225A0 (en) 1992-11-15
NO304266B1 (no) 1998-11-23
KR100307274B1 (ko) 2001-12-05
FI934000A (fi) 1993-09-13
EP0579615B1 (de) 2001-07-04
GR3036792T3 (en) 2002-01-31
US5654314A (en) 1997-08-05
CA2105575C (en) 2000-04-25
DE59209907D1 (de) 2001-08-09
FI120235B (fi) 2009-08-14
NO933274L (no) 1993-11-12
MX9201139A (es) 1992-10-01

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