FI105026B - Menetelmä valmistaa terapeuttisesti aktiivisia 3,4-dihydroisokinoliinijohdannaisia - Google Patents
Menetelmä valmistaa terapeuttisesti aktiivisia 3,4-dihydroisokinoliinijohdannaisia Download PDFInfo
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- FI105026B FI105026B FI932709A FI932709A FI105026B FI 105026 B FI105026 B FI 105026B FI 932709 A FI932709 A FI 932709A FI 932709 A FI932709 A FI 932709A FI 105026 B FI105026 B FI 105026B
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Classifications
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- A61K31/475—Quinolines; Isoquinolines having an indole ring, e.g. yohimbine, reserpine, strychnine, vinblastine
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- A61K31/496—Non-condensed piperazines containing further heterocyclic rings, e.g. rifampin, thiothixene or sparfloxacin
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- A—HUMAN NECESSITIES
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- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
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- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/535—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one oxygen as the ring hetero atoms, e.g. 1,2-oxazines
- A61K31/5375—1,4-Oxazines, e.g. morpholine
- A61K31/5377—1,4-Oxazines, e.g. morpholine not condensed and containing further heterocyclic rings, e.g. timolol
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- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
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- A61K31/33—Heterocyclic compounds
- A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
- A61K31/54—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with at least one nitrogen and one sulfur as the ring hetero atoms, e.g. sulthiame
- A61K31/541—Non-condensed thiazines containing further heterocyclic rings
-
- A—HUMAN NECESSITIES
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- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P11/00—Drugs for disorders of the respiratory system
- A61P11/06—Antiasthmatics
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- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P25/00—Drugs for disorders of the nervous system
- A61P25/28—Drugs for disorders of the nervous system for treating neurodegenerative disorders of the central nervous system, e.g. nootropic agents, cognition enhancers, drugs for treating Alzheimer's disease or other forms of dementia
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P7/00—Drugs for disorders of the blood or the extracellular fluid
- A61P7/02—Antithrombotic agents; Anticoagulants; Platelet aggregation inhibitors
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P9/00—Drugs for disorders of the cardiovascular system
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- Health & Medical Sciences (AREA)
- Chemical & Material Sciences (AREA)
- Veterinary Medicine (AREA)
- Pharmacology & Pharmacy (AREA)
- Public Health (AREA)
- General Health & Medical Sciences (AREA)
- Animal Behavior & Ethology (AREA)
- Medicinal Chemistry (AREA)
- Life Sciences & Earth Sciences (AREA)
- Epidemiology (AREA)
- Organic Chemistry (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- General Chemical & Material Sciences (AREA)
- Bioinformatics & Cheminformatics (AREA)
- Engineering & Computer Science (AREA)
- Neurosurgery (AREA)
- Biomedical Technology (AREA)
- Neurology (AREA)
- Pulmonology (AREA)
- Psychiatry (AREA)
- Rheumatology (AREA)
- Hospice & Palliative Care (AREA)
- Pain & Pain Management (AREA)
- Hematology (AREA)
- Heart & Thoracic Surgery (AREA)
- Cardiology (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Diabetes (AREA)
- Plural Heterocyclic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Heterocyclic Carbon Compounds Containing A Hetero Ring Having Oxygen Or Sulfur (AREA)
- Pretreatment Of Seeds And Plants (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| DE4041482 | 1990-12-22 | ||
| DE4041482A DE4041482A1 (de) | 1990-12-22 | 1990-12-22 | Neue pharmazeutische verwendung carbocyclisch und heterocyclisch annelierter dihydropyridine |
| EP9102470 | 1991-12-20 | ||
| PCT/EP1991/002470 WO1992011010A1 (de) | 1990-12-22 | 1991-12-20 | Neue 3,4-dihydroisochinolinderivate und neue pharmazeutische verwendung carbocyclisch und heterocyclisch anellierter dihydropyridine |
Publications (3)
| Publication Number | Publication Date |
|---|---|
| FI932709A FI932709A (fi) | 1993-06-14 |
| FI932709A0 FI932709A0 (fi) | 1993-06-14 |
| FI105026B true FI105026B (fi) | 2000-05-31 |
Family
ID=6421218
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| FI932709A FI105026B (fi) | 1990-12-22 | 1993-06-14 | Menetelmä valmistaa terapeuttisesti aktiivisia 3,4-dihydroisokinoliinijohdannaisia |
Country Status (33)
| Country | Link |
|---|---|
| US (3) | US6034094A (hu) |
| EP (2) | EP0781556A1 (hu) |
| JP (1) | JP3283877B2 (hu) |
| KR (1) | KR100227953B1 (hu) |
| AT (1) | ATE177948T1 (hu) |
| AU (1) | AU666107B2 (hu) |
| BR (1) | BR1100520A (hu) |
| CA (1) | CA2098917A1 (hu) |
| CZ (3) | CZ284695A3 (hu) |
| DE (3) | DE4041482A1 (hu) |
| DK (1) | DK0563128T3 (hu) |
| ES (1) | ES2129040T3 (hu) |
| FI (1) | FI105026B (hu) |
| GR (1) | GR3030341T3 (hu) |
| HK (1) | HK1010683A1 (hu) |
| HR (1) | HRP940721B1 (hu) |
| HU (1) | HU217819B (hu) |
| ID (1) | ID16001A (hu) |
| IE (3) | IE20001043A1 (hu) |
| IL (1) | IL100450A (hu) |
| MX (1) | MX9102765A (hu) |
| NO (1) | NO179515C (hu) |
| NZ (1) | NZ241140A (hu) |
| PL (1) | PL172262B1 (hu) |
| PT (1) | PT99901B (hu) |
| RU (2) | RU2115647C1 (hu) |
| SG (1) | SG43064A1 (hu) |
| SI (1) | SI9111975B (hu) |
| SK (1) | SK281017B6 (hu) |
| TW (1) | TW283145B (hu) |
| WO (1) | WO1992011010A1 (hu) |
| YU (1) | YU48063B (hu) |
| ZA (1) | ZA9110116B (hu) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0957092A1 (de) * | 1992-06-22 | 1999-11-17 | Boehringer Ingelheim Pharma KG | Anellierte Dihydropyridine und deren Verwendung für die Herstellung von pharmazeutischen Zubereitungen |
| DE4343683A1 (de) * | 1993-12-21 | 1995-06-22 | Boehringer Ingelheim Kg | Anellierte Dihydropyridine und deren Verwendung für die Herstellung von pharmazeutischen Zubereitungen |
| PL315052A1 (en) * | 1993-12-21 | 1996-09-30 | Boehringer Ingelheim Kg | Condensed dihydropyridines, method of obtaining them, their application in producing pharmaceutic preparations and pharmaceutic preparations containing such compounds |
| GB2341318A (en) * | 1998-09-14 | 2000-03-15 | Boehringer Ingelheim Pharma | A Dihydroisoquinoline (LOE 908) and Traumatic Brain Injury. |
| AU2003215119B2 (en) * | 2002-02-11 | 2008-11-20 | Gold-T Tech, Inc. | Method for preventing thrombus formation |
| DE102004055633A1 (de) * | 2004-11-12 | 2006-05-18 | Schering Ag | 5-substituierte Chinolin- und Isochinolin-Derivate, ein Verfahren zu ihrer Herstellung und ihre Verwendung als Entzündungshemmer |
| BRPI0808737A2 (pt) * | 2007-03-15 | 2014-08-12 | Hoffmann La Roche | Malonamidas como antagonistas de orexinas. |
| CZ302637B6 (cs) * | 2010-01-05 | 2011-08-10 | Zentiva, K. S | Zpusob prípravy 6,7-dimethoxy-1-[2-(4-trifluormethylfenyl)ethyl]-3,4-dihydroisochinolinu |
| EP2420237A1 (en) | 2010-08-11 | 2012-02-22 | Ville Takio | Fluorinated derivatives of endogenous isoquinolines for use in the treatment of diseases mediated through endogenous isoquinoline pathways |
| KR101645930B1 (ko) | 2014-12-16 | 2016-08-05 | (주) 우수 | 타월 거치대 |
Family Cites Families (4)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| DE3013906A1 (de) * | 1980-04-11 | 1981-10-15 | C.H. Boehringer Sohn, 6507 Ingelheim | Substituierte (alpha) -aminocarbonyl-l-benzyl-3,4-dihydro-isochinoline, verfahren zu deren herstellung und deren verwendung |
| DE3621413A1 (de) * | 1986-06-26 | 1988-01-07 | Boehringer Ingelheim Kg | Verwendung carbocyclisch und heterocyclisch annelierter dihydropyridine als cardioprotektive mittel sowie neue heterocyclisch und carbocyclisch anellierte dihydropyridine, verfahren zu deren herstellung und zwischenstufen fuer deren herstellung |
| IL86131A0 (en) * | 1987-04-24 | 1988-11-15 | Boehringer Ingelheim Kg | Benzo-and thieno-3,4-dihydropyridine derivatives,their preparation and pharmaceutical compositions containing them |
| DE3827727A1 (de) * | 1988-08-16 | 1990-02-22 | Boehringer Ingelheim Kg | Anellierte tetrahydropyridinessigsaeurederivate, verfahren zu deren herstellung und verwendung solcher verbindungen zur kardioprotektion |
-
1990
- 1990-12-22 DE DE4041482A patent/DE4041482A1/de not_active Ceased
- 1990-12-22 DE DE9017900U patent/DE9017900U1/de not_active Expired - Lifetime
-
1991
- 1991-12-20 WO PCT/EP1991/002470 patent/WO1992011010A1/de active IP Right Grant
- 1991-12-20 KR KR1019930701908A patent/KR100227953B1/ko not_active IP Right Cessation
- 1991-12-20 IE IE20001043A patent/IE20001043A1/en unknown
- 1991-12-20 DK DK92901178T patent/DK0563128T3/da active
- 1991-12-20 CZ CZ952846A patent/CZ284695A3/cs not_active IP Right Cessation
- 1991-12-20 PT PT99901A patent/PT99901B/pt not_active IP Right Cessation
- 1991-12-20 AU AU90802/91A patent/AU666107B2/en not_active Ceased
- 1991-12-20 EP EP96119881A patent/EP0781556A1/de not_active Withdrawn
- 1991-12-20 PL PL91299674A patent/PL172262B1/pl unknown
- 1991-12-20 IE IE19990430A patent/IE990430A1/en unknown
- 1991-12-20 ES ES92901178T patent/ES2129040T3/es not_active Expired - Lifetime
- 1991-12-20 DE DE59109115T patent/DE59109115D1/de not_active Expired - Fee Related
- 1991-12-20 CA CA002098917A patent/CA2098917A1/en not_active Abandoned
- 1991-12-20 HU HU9301820A patent/HU217819B/hu not_active IP Right Cessation
- 1991-12-20 SK SK617-93A patent/SK281017B6/sk unknown
- 1991-12-20 SG SG1996003170A patent/SG43064A1/en unknown
- 1991-12-20 EP EP92901178A patent/EP0563128B1/de not_active Expired - Lifetime
- 1991-12-20 RU RU93046319A patent/RU2115647C1/ru not_active IP Right Cessation
- 1991-12-20 IL IL10045091A patent/IL100450A/xx not_active IP Right Cessation
- 1991-12-20 IE IE448691A patent/IE914486A1/en not_active Application Discontinuation
- 1991-12-20 JP JP50207392A patent/JP3283877B2/ja not_active Expired - Fee Related
- 1991-12-20 AT AT92901178T patent/ATE177948T1/de not_active IP Right Cessation
- 1991-12-20 RU RU94046320/14A patent/RU2149000C1/ru not_active IP Right Cessation
- 1991-12-20 CZ CZ19931213A patent/CZ289533B6/cs not_active IP Right Cessation
- 1991-12-23 MX MX9102765A patent/MX9102765A/es not_active IP Right Cessation
- 1991-12-23 YU YU197591A patent/YU48063B/sh unknown
- 1991-12-23 TW TW080110028A patent/TW283145B/zh active
- 1991-12-23 NZ NZ241140A patent/NZ241140A/en unknown
- 1991-12-23 SI SI9111975A patent/SI9111975B/sl unknown
- 1991-12-23 ZA ZA9110116A patent/ZA9110116B/xx unknown
-
1993
- 1993-06-14 FI FI932709A patent/FI105026B/fi active
- 1993-06-21 NO NO932279A patent/NO179515C/no unknown
-
1994
- 1994-10-21 HR HRP-1975/91A patent/HRP940721B1/xx not_active IP Right Cessation
-
1995
- 1995-06-01 US US08/458,069 patent/US6034094A/en not_active Expired - Fee Related
- 1995-06-01 US US08/456,357 patent/US5665729A/en not_active Expired - Fee Related
- 1995-06-01 US US08/456,889 patent/US5686462A/en not_active Expired - Fee Related
-
1996
- 1996-05-27 CZ CZ19961523A patent/CZ289685B6/cs not_active IP Right Cessation
-
1997
- 1997-05-13 BR BR1100520-3A patent/BR1100520A/pt active IP Right Grant
- 1997-06-13 ID IDP972024A patent/ID16001A/id unknown
-
1998
- 1998-10-21 HK HK98111437A patent/HK1010683A1/xx not_active IP Right Cessation
-
1999
- 1999-05-27 GR GR990401430T patent/GR3030341T3/el unknown
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