ES8601686A1 - Un procedimiento para preparar una composicion solida de liberacion rapida a base de un compuesto de dihidropiridina a. - Google Patents

Un procedimiento para preparar una composicion solida de liberacion rapida a base de un compuesto de dihidropiridina a.

Info

Publication number
ES8601686A1
ES8601686A1 ES535019A ES535019A ES8601686A1 ES 8601686 A1 ES8601686 A1 ES 8601686A1 ES 535019 A ES535019 A ES 535019A ES 535019 A ES535019 A ES 535019A ES 8601686 A1 ES8601686 A1 ES 8601686A1
Authority
ES
Spain
Prior art keywords
dihydropyridine
compound
procedure
quick release
preparing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
ES535019A
Other languages
English (en)
Spanish (es)
Other versions
ES535019A0 (es
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Fujisawa Pharmaceutical Co Ltd
Original Assignee
Fujisawa Pharmaceutical Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Fujisawa Pharmaceutical Co Ltd filed Critical Fujisawa Pharmaceutical Co Ltd
Publication of ES535019A0 publication Critical patent/ES535019A0/es
Publication of ES8601686A1 publication Critical patent/ES8601686A1/es
Expired legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/20—Pills, tablets, discs, rods
    • A61K9/28—Dragees; Coated pills or tablets, e.g. with film or compression coating
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/44—Non condensed pyridines; Hydrogenated derivatives thereof
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K9/00—Medicinal preparations characterised by special physical form
    • A61K9/14—Particulate form, e.g. powders, Processes for size reducing of pure drugs or the resulting products, Pure drug nanoparticles
    • A61K9/141—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers
    • A61K9/146—Intimate drug-carrier mixtures characterised by the carrier, e.g. ordered mixtures, adsorbates, solid solutions, eutectica, co-dried, co-solubilised, co-kneaded, co-milled, co-ground products, co-precipitates, co-evaporates, co-extrudates, co-melts; Drug nanoparticles with adsorbed surface modifiers with organic macromolecular compounds

Landscapes

  • Health & Medical Sciences (AREA)
  • Epidemiology (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Medicinal Preparation (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
ES535019A 1983-08-11 1984-08-09 Un procedimiento para preparar una composicion solida de liberacion rapida a base de un compuesto de dihidropiridina a. Expired ES8601686A1 (es)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
JP58147871A JPS6038322A (ja) 1983-08-11 1983-08-11 ジヒドロピリジンａ物質含有易溶性固形製剤

Publications (2)

Publication Number Publication Date
ES535019A0 ES535019A0 (es) 1985-11-01
ES8601686A1 true ES8601686A1 (es) 1985-11-01

Family

ID=15440116

Family Applications (1)

Application Number Title Priority Date Filing Date
ES535019A Expired ES8601686A1 (es) 1983-08-11 1984-08-09 Un procedimiento para preparar una composicion solida de liberacion rapida a base de un compuesto de dihidropiridina a.

Country Status (24)

Country Link
US (1) US4654206A (https=)
EP (1) EP0137198B1 (https=)
JP (1) JPS6038322A (https=)
KR (1) KR910003559B1 (https=)
AT (1) AT382779B (https=)
AU (1) AU564506B2 (https=)
BE (1) BE900348A (https=)
CA (1) CA1228815A (https=)
CH (1) CH660967A5 (https=)
DE (1) DE3484259D1 (https=)
DK (1) DK164020C (https=)
ES (1) ES8601686A1 (https=)
FI (1) FI83839C (https=)
FR (1) FR2550444B1 (https=)
GB (1) GB2145332B (https=)
GR (1) GR80004B (https=)
HK (1) HK6688A (https=)
IE (1) IE57757B1 (https=)
IL (1) IL72565A (https=)
IT (1) IT1183062B (https=)
MY (1) MY100042A (https=)
PH (1) PH21551A (https=)
SG (1) SG73087G (https=)
ZA (1) ZA845844B (https=)

Families Citing this family (30)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE3424553A1 (de) * 1984-07-04 1986-01-09 Bayer Ag, 5090 Leverkusen Feste arzneizubereitungen mit dihydropyridinen und verfahren zu ihrer herstellung
GB8608080D0 (en) * 1986-04-02 1986-05-08 Fujisawa Pharmaceutical Co Solid dispersion composition
EP0281200B1 (en) * 1987-03-02 1994-01-19 Yamanouchi Europe B.V. Pharmaceutical composition, pharmaceutical granulate and process for their preparation
DE3720757A1 (de) * 1987-06-24 1989-01-05 Bayer Ag Dhp-manteltablette
US5045553A (en) * 1987-06-24 1991-09-03 Fujisawa Pharmaceutical Company, Ltd. Pharmaceutical composition for percutaneous drug absorption and percutaneous drug absorption promoter
NO883326L (no) * 1987-08-11 1989-02-13 Bayer Ag Dhp-retard-tilberedning.
JPH02206A (ja) * 1987-11-11 1990-01-05 Fujisawa Pharmaceut Co Ltd エキシホンと水溶性高分子化合物とを含有することを特徴とする新規製剤
DE3877331T2 (de) * 1987-11-11 1993-05-27 Pharmascience Lab Exifon und ein wasserloesliches polymer enthaltende pharmazeutische zubereitung.
FR2640137A1 (fr) * 1988-12-08 1990-06-15 Texinfine Sa Systemes transporteurs de principes actifs lipophiles et leur procede d'obtention
JPH0347124A (ja) * 1989-04-20 1991-02-28 Fujisawa Pharmaceut Co Ltd 経口吸収用製剤
WO1991007385A1 (en) * 1989-11-18 1991-05-30 Schering Agrochemicals Limited Preparation of propenoic acid derivatives
JP3110794B2 (ja) * 1991-06-05 2000-11-20 ユーシービージャパン株式会社 １，４−ジヒドロピリジン誘導体を含有する製剤
US5340591A (en) * 1992-01-24 1994-08-23 Fujisawa Pharmaceutical Co., Ltd. Method of producing a solid dispersion of the sparingly water-soluble drug, nilvadipine
IL104192A (en) * 1992-02-17 1998-01-04 Siegfried Ag Pharma Pharmaceutical dosage forms having prolonged release rate of zero order of the active ingredient
EP0557244B1 (en) * 1992-02-17 1996-03-13 Siegfried Pharma AG Dosage forms having prolonged active-ingredient release
DE4316537A1 (de) * 1993-05-18 1994-11-24 Basf Ag Zubereitungen in Form fester Lösungen
US5871776A (en) * 1995-01-31 1999-02-16 Mehta; Atul M. Controlled-release nifedipine
DE19511131A1 (de) * 1995-03-27 1996-10-02 Basf Ag Mechanisch stabile feste Wirkstoffzubereitungsformen
TW487582B (en) * 1995-08-11 2002-05-21 Nissan Chemical Ind Ltd Method for converting sparingly water-soluble medical substance to amorphous state
WO1997034601A1 (fr) * 1996-03-18 1997-09-25 Eisai Co., Ltd. Compositions medicamenteuses a solubilite amelioree
HN1998000115A (es) * 1997-08-21 1999-06-02 Warner Lambert Co Formas de dosificación farmacéuticas sólidas
US6555139B2 (en) 1999-06-28 2003-04-29 Wockhardt Europe Limited Preparation of micron-size pharmaceutical particles by microfluidization
JP2003146878A (ja) * 2002-11-22 2003-05-21 Sawai Pharmaceutical Co Ltd ニルバジピン含有易溶性固形製剤およびその製造法
CA2525970C (en) * 2003-05-15 2011-03-22 Roskamp Research, Llc Use of nilvadipine for reducing amyloid deposition, amyloid neurotoxicity and microgliosis
TWI346114B (en) * 2003-09-29 2011-08-01 Method for stabilization of diarylvinylene compounds
CA2546115C (en) 2003-11-14 2013-01-08 Ajinomoto Co., Inc. Solid dispersions or solid dispersion pharmaceutical preparations of phenylalanine derivatives
US20100093810A1 (en) * 2007-10-05 2010-04-15 Alzheimer's Institute Of America, Inc. Pharmaceutical Compositions for Reducing Amyloid Deposition, Amyloid Neurotoxicity, and Microgliosis
TWI500422B (zh) * 2007-10-05 2015-09-21 Alzheimer S Inst Of America Inc 以（－）－尼代地平（ｎｉｌｖａｄｉｐｉｎｅ）對映異構物減低類澱粉沉積、類澱粉神經毒性及微神經膠細胞增生之方法
WO2013122260A1 (en) * 2012-02-15 2013-08-22 Takeda Pharmaceutical Company Limited Tablet
AU2017324406A1 (en) * 2016-09-07 2019-05-02 Saniona A/S Tesofensine compositions

Family Cites Families (13)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3852421A (en) * 1970-03-23 1974-12-03 Shinetsu Chemical Co Excipient and shaped medicaments prepared therewith
GB1593261A (en) * 1976-07-23 1981-07-15 Inveresk Res Int Controlled release suppository
GB1579818A (en) * 1977-06-07 1980-11-26 Yamanouchi Pharma Co Ltd Nifedipine-containing solid preparation composition
CA1117117A (en) * 1978-10-10 1982-01-26 Fujisawa Pharmaceutical Co., Ltd. 2-methyl-dihydropyridine compound, processes for preparation thereof and pharmaceutical composition comprising the same
DE3013839A1 (de) * 1979-04-13 1980-10-30 Freunt Ind Co Ltd Verfahren zur herstellung einer aktivierten pharmazeutischen zusammensetzung
CA1146866A (en) * 1979-07-05 1983-05-24 Yamanouchi Pharmaceutical Co. Ltd. Process for the production of sustained release pharmaceutical composition of solid medical material
US4259314A (en) * 1979-12-10 1981-03-31 Hans Lowey Method and composition for the preparation of controlled long-acting pharmaceuticals
JPS5668619A (en) * 1980-10-09 1981-06-09 Yamanouchi Pharmaceut Co Ltd Nifedipine-containing solid composition
JPS5877811A (ja) * 1981-11-04 1983-05-11 Kanebo Ltd 安定な易吸収性ニフエジピン製剤の製法
US4369172A (en) * 1981-12-18 1983-01-18 Forest Laboratories Inc. Prolonged release therapeutic compositions based on hydroxypropylmethylcellulose
JPS58109412A (ja) * 1981-12-23 1983-06-29 Toa Eiyou Kagaku Kogyo Kk ニフエジピン固形製剤
US4389393A (en) * 1982-03-26 1983-06-21 Forest Laboratories, Inc. Sustained release therapeutic compositions based on high molecular weight hydroxypropylmethylcellulose
DE3307422A1 (de) * 1983-03-03 1984-09-06 Bayer Ag, 5090 Leverkusen Fluessigzubereitungen von dihydropyridinen, ein verfahren zu ihrer herstellung, sowie ihre verwendung bei der bekaempfung von erkrankungen

Also Published As

Publication number Publication date
FR2550444B1 (fr) 1988-09-16
DK164020C (da) 1992-09-28
IE841974L (en) 1985-02-11
AT382779B (de) 1987-04-10
IL72565A0 (en) 1984-11-30
CA1228815A (en) 1987-11-03
JPS6038322A (ja) 1985-02-27
GB2145332A (en) 1985-03-27
MY100042A (en) 1989-06-29
DK388884D0 (da) 1984-08-10
KR850001691A (ko) 1985-04-01
ES535019A0 (es) 1985-11-01
EP0137198B1 (en) 1991-03-13
PH21551A (en) 1987-12-11
FR2550444A1 (fr) 1985-02-15
KR910003559B1 (ko) 1991-06-05
EP0137198A3 (en) 1986-10-01
US4654206A (en) 1987-03-31
AU3130684A (en) 1985-02-14
EP0137198A2 (en) 1985-04-17
IL72565A (en) 1988-01-31
FI83839B (fi) 1991-05-31
DK388884A (da) 1985-02-12
CH660967A5 (de) 1987-06-30
SG73087G (en) 1988-03-04
BE900348A (fr) 1985-02-11
FI843083A0 (fi) 1984-08-06
ATA251584A (de) 1986-09-15
GB8419815D0 (en) 1984-09-05
DK164020B (da) 1992-05-04
IT8422294A0 (it) 1984-08-09
DE3484259D1 (de) 1991-04-18
IE57757B1 (en) 1993-03-24
IT1183062B (it) 1987-10-05
HK6688A (en) 1988-01-29
GR80004B (en) 1984-11-30
AU564506B2 (en) 1987-08-13
FI843083L (fi) 1985-02-12
FI83839C (fi) 1991-09-10
JPH0412245B2 (https=) 1992-03-04
GB2145332B (en) 1987-03-25
ZA845844B (en) 1985-05-29

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Legal Events

Date Code Title Description
FD1A Patent lapsed

Effective date: 20050705