ES8505372A1 - Un ester penem carboxilico - Google Patents
Un ester penem carboxilicoInfo
- Publication number
- ES8505372A1 ES8505372A1 ES528546A ES528546A ES8505372A1 ES 8505372 A1 ES8505372 A1 ES 8505372A1 ES 528546 A ES528546 A ES 528546A ES 528546 A ES528546 A ES 528546A ES 8505372 A1 ES8505372 A1 ES 8505372A1
- Authority
- ES
- Spain
- Prior art keywords
- antibacterial method
- oral antibacterial
- animal
- oral
- carbamoyloxymethyl
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Expired
Links
- 230000000844 anti-bacterial effect Effects 0.000 title 1
- 208000035143 Bacterial infection Diseases 0.000 abstract 1
- -1 acetoxymethyl ester Chemical class 0.000 abstract 1
- 208000022362 bacterial infectious disease Diseases 0.000 abstract 1
- 231100000252 nontoxic Toxicity 0.000 abstract 1
- 230000003000 nontoxic effect Effects 0.000 abstract 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/86—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with only atoms other than nitrogen atoms directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
- C07D499/88—Compounds with a double bond between positions 2 and 3 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
-
- A—HUMAN NECESSITIES
- A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
- A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
- A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
- A61P31/04—Antibacterial agents
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Chemical Kinetics & Catalysis (AREA)
- Life Sciences & Earth Sciences (AREA)
- General Chemical & Material Sciences (AREA)
- Medicinal Chemistry (AREA)
- Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
- Communicable Diseases (AREA)
- Pharmacology & Pharmacy (AREA)
- Oncology (AREA)
- Animal Behavior & Ethology (AREA)
- General Health & Medical Sciences (AREA)
- Public Health (AREA)
- Veterinary Medicine (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Cephalosporin Compounds (AREA)
Abstract
PROCEDIMIENTO PARA LA PREPARACION DE UN ESTER PENEM CARBOXILICO DE FORMULA GENERAL (I), EN LA QUE R REPRESENTA UN GRUPO ACETOXIMETILO, METOXIMETILO O FTALIDILO.CONSISTE EN ESTERIFICAR UN COMPUESTO DE FORMULA GENERAL (II) O UNA SAL O UN DERIVADO ESTERIFICANTE REACTIVO DEL MISMO, CON UN COMPUESTO DE FORMULA RX, EN LA QUE X ES UN ATOMO DE HALOGENO, UN GRUPO HIDROXI O UN GRUPO DE FORMULA: OSO2R2, EN LA QUE R2 ES ALQUILO INFERIOR O UN GRUPO ARILO.DE APLICACION COMO ANTIBIOTICOS UTILIZADOS COMO AGENTES TERAPEUTICOS Y PROFILACTICOS CONTRA INFECCIONES BACTERIANAS.
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| GB838300295A GB8300295D0 (en) | 1983-01-06 | 1983-01-06 | Penem esters |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| ES8505372A1 true ES8505372A1 (es) | 1985-05-16 |
| ES528546A0 ES528546A0 (es) | 1985-05-16 |
Family
ID=10535987
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| ES528546A Granted ES528546A0 (es) | 1983-01-06 | 1983-12-29 | Un ester penem carboxilico |
Country Status (31)
| Country | Link |
|---|---|
| US (1) | US5051416A (es) |
| JP (1) | JPS59134795A (es) |
| KR (1) | KR900004418B1 (es) |
| AT (1) | AT382622B (es) |
| AU (1) | AU557178B2 (es) |
| BE (1) | BE898603A (es) |
| CA (1) | CA1215042A (es) |
| CH (1) | CH659073A5 (es) |
| CS (2) | CS235996B2 (es) |
| DE (1) | DE3400090A1 (es) |
| DK (1) | DK166387C (es) |
| ES (1) | ES528546A0 (es) |
| FI (1) | FI81103C (es) |
| FR (1) | FR2539130B1 (es) |
| GB (2) | GB8300295D0 (es) |
| GR (1) | GR81730B (es) |
| HK (1) | HK74987A (es) |
| HU (1) | HU191243B (es) |
| IE (1) | IE56903B1 (es) |
| IL (1) | IL70606A (es) |
| IT (1) | IT1209490B (es) |
| NL (1) | NL8400015A (es) |
| NO (1) | NO160446C (es) |
| NZ (1) | NZ206743A (es) |
| PH (1) | PH18881A (es) |
| PT (1) | PT77922B (es) |
| SE (1) | SE458117B (es) |
| SG (1) | SG34387G (es) |
| SU (1) | SU1209031A3 (es) |
| UA (1) | UA6039A1 (es) |
| ZA (1) | ZA8457B (es) |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US5364768A (en) * | 1987-07-07 | 1994-11-15 | Farmitalia Carlo Erba S.R.L. | Process for the preparation of penems |
| GB2206578B (en) * | 1987-07-07 | 1991-07-03 | Erba Carlo Spa | Process for the preparation of penems |
| EP0937725A3 (en) | 1992-04-28 | 2004-12-01 | Tanabe Seiyaku Co., Ltd. | Method for removing the protecting group for hydroxy group |
Family Cites Families (6)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| NL7401782A (es) * | 1973-02-14 | 1974-08-16 | ||
| AU535080B2 (en) * | 1979-02-24 | 1984-03-01 | Farmitalia Carlo Erba S.R.L. | Penicillins |
| ZA80993B (en) * | 1979-02-24 | 1981-02-25 | Erba Farmitalia | -lactam-containing antibacterial agents and -lactamase inhibitors and preparation thereof |
| GB2043699B (en) * | 1979-03-03 | 1983-05-11 | Park Chem Co | Cyanide-free carburizing process and composition |
| US4482565A (en) * | 1980-02-22 | 1984-11-13 | Farmitalia Carlo Erba S.P.A. | β-Lactam-containing antibacterial agents and β-lactamase inhibitors |
| AT379399B (de) * | 1981-12-11 | 1985-12-27 | Erba Farmitalia | Verfahren zur herstellung von optisch aktiven penemen |
-
1983
- 1983-01-06 GB GB838300295A patent/GB8300295D0/en active Pending
- 1983-12-29 ES ES528546A patent/ES528546A0/es active Granted
-
1984
- 1984-01-02 FI FI840003A patent/FI81103C/fi not_active IP Right Cessation
- 1984-01-03 IL IL70606A patent/IL70606A/xx not_active IP Right Cessation
- 1984-01-03 GR GR73420A patent/GR81730B/el unknown
- 1984-01-03 FR FR8400040A patent/FR2539130B1/fr not_active Expired
- 1984-01-03 CS CS8480A patent/CS235996B2/cs unknown
- 1984-01-03 AU AU23047/84A patent/AU557178B2/en not_active Ceased
- 1984-01-03 DE DE19843400090 patent/DE3400090A1/de not_active Ceased
- 1984-01-03 NL NL8400015A patent/NL8400015A/nl not_active Application Discontinuation
- 1984-01-03 AT AT0001584A patent/AT382622B/de not_active IP Right Cessation
- 1984-01-03 IT IT8419007A patent/IT1209490B/it active
- 1984-01-03 GB GB08400043A patent/GB2133010B/en not_active Expired
- 1984-01-04 SE SE8400040A patent/SE458117B/sv not_active IP Right Cessation
- 1984-01-04 BE BE0/212151A patent/BE898603A/fr not_active IP Right Cessation
- 1984-01-04 PH PH30064A patent/PH18881A/en unknown
- 1984-01-04 PT PT77922A patent/PT77922B/pt not_active IP Right Cessation
- 1984-01-04 ZA ZA8457A patent/ZA8457B/xx unknown
- 1984-01-04 IE IE6/84A patent/IE56903B1/en not_active IP Right Cessation
- 1984-01-04 CA CA000444654A patent/CA1215042A/en not_active Expired
- 1984-01-05 KR KR1019840000014A patent/KR900004418B1/ko not_active IP Right Cessation
- 1984-01-05 SU SU843688716A patent/SU1209031A3/ru active
- 1984-01-05 DK DK005284A patent/DK166387C/da active
- 1984-01-05 JP JP59000110A patent/JPS59134795A/ja active Granted
- 1984-01-05 CH CH42/84A patent/CH659073A5/de not_active IP Right Cessation
- 1984-01-05 NO NO840035A patent/NO160446C/no unknown
- 1984-01-05 NZ NZ206743A patent/NZ206743A/en unknown
- 1984-01-05 UA UA3688716A patent/UA6039A1/uk unknown
- 1984-01-05 HU HU8437A patent/HU191243B/hu not_active IP Right Cessation
-
1987
- 1987-04-14 SG SG34387A patent/SG34387G/en unknown
- 1987-10-15 HK HK749/87A patent/HK74987A/xx not_active IP Right Cessation
-
1989
- 1989-04-03 US US07/331,853 patent/US5051416A/en not_active Expired - Fee Related
-
1991
- 1991-12-20 CS CS914150A patent/CS415091A3/cs unknown
Also Published As
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| PC1A | Transfer granted | ||
| FD1A | Patent lapsed |
Effective date: 20041004 |