EP1471054A4 - Aminoalkoholderivat oder phosphonsäurederivat und diese enthaltende medizinische zusammensetzung - Google Patents

Aminoalkoholderivat oder phosphonsäurederivat und diese enthaltende medizinische zusammensetzung

Info

Publication number
EP1471054A4
EP1471054A4 EP03701048A EP03701048A EP1471054A4 EP 1471054 A4 EP1471054 A4 EP 1471054A4 EP 03701048 A EP03701048 A EP 03701048A EP 03701048 A EP03701048 A EP 03701048A EP 1471054 A4 EP1471054 A4 EP 1471054A4
Authority
EP
European Patent Office
Prior art keywords
lower alkyl
gen
day
optionally substituted
derivative
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
EP03701048A
Other languages
English (en)
French (fr)
Other versions
EP1471054A1 (de
EP1471054B1 (de
Inventor
Takahide Nishi
Takaichi Shimozato
Futoshi Nara
Shojiro Miyazaki
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Daiichi Sankyo Co Ltd
Original Assignee
Sankyo Co Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sankyo Co Ltd filed Critical Sankyo Co Ltd
Priority to SI200331668T priority Critical patent/SI1471054T1/sl
Publication of EP1471054A1 publication Critical patent/EP1471054A1/de
Publication of EP1471054A4 publication Critical patent/EP1471054A4/de
Application granted granted Critical
Publication of EP1471054B1 publication Critical patent/EP1471054B1/de
Priority to CY20091101015T priority patent/CY1109457T1/el
Anticipated expiration legal-status Critical
Expired - Lifetime legal-status Critical Current

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    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/32—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/33—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to ring carbon atoms with substituted hydrocarbon radicals, directly attached to ring carbon atoms
    • C07D207/335—Radicals substituted by nitrogen atoms not forming part of a nitro radical
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D307/00—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom
    • C07D307/02—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings
    • C07D307/34—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members
    • C07D307/38—Heterocyclic compounds containing five-membered rings having one oxygen atom as the only ring hetero atom not condensed with other rings having two or three double bonds between ring members or between ring members and non-ring members with substituted hydrocarbon radicals attached to ring carbon atoms
    • C07D307/52—Radicals substituted by nitrogen atoms not forming part of a nitro radical
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D333/00—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom
    • C07D333/02—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings
    • C07D333/04—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom
    • C07D333/06—Heterocyclic compounds containing five-membered rings having one sulfur atom as the only ring hetero atom not condensed with other rings not substituted on the ring sulphur atom with only hydrogen atoms, hydrocarbon or substituted hydrocarbon radicals, directly attached to the ring carbon atoms
    • C07D333/14—Radicals substituted by singly bound hetero atoms other than halogen
    • C07D333/20—Radicals substituted by singly bound hetero atoms other than halogen by nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having one nitrogen atom as the only ring hetero atom
    • C07F9/572—Five-membered rings
    • C—CHEMISTRY; METALLURGY
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    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/655—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms
    • C07F9/65515—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having oxygen atoms, with or without sulfur, selenium, or tellurium atoms, as the only ring hetero atoms the oxygen atom being part of a five-membered ring
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    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
    • C07F9/6553—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having sulfur atoms, with or without selenium or tellurium atoms, as the only ring hetero atoms
    • C07F9/655345—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having sulfur atoms, with or without selenium or tellurium atoms, as the only ring hetero atoms the sulfur atom being part of a five-membered ring
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

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  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Public Health (AREA)
  • Neurology (AREA)
  • Biomedical Technology (AREA)
  • Neurosurgery (AREA)
  • Cardiology (AREA)
  • Biochemistry (AREA)
  • Diabetes (AREA)
  • Molecular Biology (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Hematology (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Dermatology (AREA)
  • Physical Education & Sports Medicine (AREA)
  • Urology & Nephrology (AREA)
  • Oncology (AREA)
  • Psychiatry (AREA)
  • Pain & Pain Management (AREA)
  • Psychology (AREA)
  • Rheumatology (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Obesity (AREA)
  • Hospice & Palliative Care (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Gastroenterology & Hepatology (AREA)
EP03701048A 2002-01-11 2003-01-09 Aminoalkoholderivat oder phosphonsäurederivat und diese enthaltende medizinische zusammensetzung Expired - Lifetime EP1471054B1 (de)

Priority Applications (2)

Application Number Priority Date Filing Date Title
SI200331668T SI1471054T1 (sl) 2002-01-11 2003-01-09 Amino alkoholni derivati ali derivati fosfoniäśne kisline in medicinski sestavki, ki vsebujejo le-te
CY20091101015T CY1109457T1 (el) 2002-01-11 2009-09-30 Παραγωγο aminoαλκοολης ή παραγωγο φωσφονικου οξεος και φαρμακευτικη συνθεση που τα περιεχει

Applications Claiming Priority (5)

Application Number Priority Date Filing Date Title
JP2002004456 2002-01-11
JP2002004484 2002-01-11
JP2002004484 2002-01-11
JP2002004456 2002-01-11
PCT/JP2003/000136 WO2003059880A1 (en) 2002-01-11 2003-01-09 Amino alcohol derivative or phosphonic acid derivative and medicinal composition containing these

Publications (3)

Publication Number Publication Date
EP1471054A1 EP1471054A1 (de) 2004-10-27
EP1471054A4 true EP1471054A4 (de) 2005-06-08
EP1471054B1 EP1471054B1 (de) 2009-07-01

Family

ID=26625490

Family Applications (1)

Application Number Title Priority Date Filing Date
EP03701048A Expired - Lifetime EP1471054B1 (de) 2002-01-11 2003-01-09 Aminoalkoholderivat oder phosphonsäurederivat und diese enthaltende medizinische zusammensetzung

Country Status (25)

Country Link
US (5) US7199150B2 (de)
EP (1) EP1471054B1 (de)
JP (1) JP4270541B2 (de)
KR (2) KR20080035702A (de)
CN (1) CN100406437C (de)
AT (1) ATE435202T1 (de)
AU (1) AU2003202495B2 (de)
BR (1) BR0306811A (de)
CA (1) CA2473461C (de)
CO (1) CO5640126A2 (de)
CY (1) CY1109457T1 (de)
DE (1) DE60328161D1 (de)
DK (1) DK1471054T3 (de)
ES (1) ES2327825T3 (de)
IL (1) IL162874A0 (de)
MX (1) MXPA04006709A (de)
NO (1) NO329134B1 (de)
NZ (1) NZ533994A (de)
PL (1) PL211954B1 (de)
PT (1) PT1471054E (de)
RU (1) RU2330839C2 (de)
SI (1) SI1471054T1 (de)
TW (1) TWI283574B (de)
WO (1) WO2003059880A1 (de)
ZA (1) ZA200406333B (de)

Families Citing this family (36)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
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US8067396B2 (en) 2011-11-29
TW200302087A (en) 2003-08-01
SI1471054T1 (sl) 2009-12-31
CN1630635A (zh) 2005-06-22
KR100836547B1 (ko) 2008-06-10
NO20043319L (no) 2004-10-05
TWI283574B (en) 2007-07-11
NZ533994A (en) 2006-10-27
US20070142335A1 (en) 2007-06-21
US20100035842A1 (en) 2010-02-11
PT1471054E (pt) 2009-09-23
JP4270541B2 (ja) 2009-06-03
CY1109457T1 (el) 2014-08-13
HK1066532A1 (en) 2005-03-24
KR20080035702A (ko) 2008-04-23
RU2330839C2 (ru) 2008-08-10
PL370790A1 (en) 2005-05-30
RU2004121143A (ru) 2006-02-27
US20070105933A1 (en) 2007-05-10
DE60328161D1 (de) 2009-08-13
EP1471054A1 (de) 2004-10-27
DK1471054T3 (da) 2009-11-09
CA2473461A1 (en) 2003-07-24
BR0306811A (pt) 2004-10-26
ATE435202T1 (de) 2009-07-15
KR20040075068A (ko) 2004-08-26
JP2003267950A (ja) 2003-09-25
IL162874A0 (en) 2005-11-20
PL211954B1 (pl) 2012-07-31
US7199150B2 (en) 2007-04-03
US20090326038A1 (en) 2009-12-31
MXPA04006709A (es) 2004-10-04
AU2003202495B2 (en) 2006-07-20
AU2003202495A1 (en) 2003-07-30
CO5640126A2 (es) 2006-05-31
CN100406437C (zh) 2008-07-30
NO329134B1 (no) 2010-08-30
US8101650B2 (en) 2012-01-24
EP1471054B1 (de) 2009-07-01
US20050043386A1 (en) 2005-02-24
ES2327825T3 (es) 2009-11-04
ZA200406333B (en) 2005-12-28
WO2003059880A1 (en) 2003-07-24
CA2473461C (en) 2011-11-01
US7638551B2 (en) 2009-12-29

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