EE03608B1 - Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid - Google Patents

Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid

Info

Publication number
EE03608B1
EE03608B1 EE9700315A EE9700315A EE03608B1 EE 03608 B1 EE03608 B1 EE 03608B1 EE 9700315 A EE9700315 A EE 9700315A EE 9700315 A EE9700315 A EE 9700315A EE 03608 B1 EE03608 B1 EE 03608B1
Authority
EE
Estonia
Prior art keywords
taxoids
preparation
pharmaceutical compositions
compositions containing
pharmaceutical
Prior art date
Application number
EE9700315A
Other languages
English (en)
Estonian (et)
Other versions
EE9700315A (et
Inventor
Bouchard Herv
Bourzat Jean-Dominique
Commer�on Alain
Original Assignee
Rh�Ne-Poulenc Rorer S.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Priority claimed from FR9503545A external-priority patent/FR2732340B1/fr
Priority claimed from FR9515381A external-priority patent/FR2742754B1/fr
Application filed by Rh�Ne-Poulenc Rorer S.A. filed Critical Rh�Ne-Poulenc Rorer S.A.
Publication of EE9700315A publication Critical patent/EE9700315A/xx
Publication of EE03608B1 publication Critical patent/EE03608B1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D305/00—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms
    • C07D305/14—Heterocyclic compounds containing four-membered rings having one oxygen atom as the only ring hetero atoms condensed with carbocyclic rings or ring systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/335—Heterocyclic compounds having oxygen as the only ring hetero atom, e.g. fungichromin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A61P35/02—Antineoplastic agents specific for leukemia
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02P—CLIMATE CHANGE MITIGATION TECHNOLOGIES IN THE PRODUCTION OR PROCESSING OF GOODS
    • Y02P20/00—Technologies relating to chemical industry
    • Y02P20/50—Improvements relating to the production of bulk chemicals
    • Y02P20/55—Design of synthesis routes, e.g. reducing the use of auxiliary or protecting groups

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Hematology (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Epoxy Compounds (AREA)
  • Medicines Containing Plant Substances (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
EE9700315A 1995-03-27 1996-03-25 Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid EE03608B1 (et)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
FR9503545A FR2732340B1 (fr) 1995-03-27 1995-03-27 Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent
FR9515381A FR2742754B1 (fr) 1995-12-22 1995-12-22 Procede de preparation de taxoides
PCT/FR1996/000440 WO1996030355A1 (fr) 1995-03-27 1996-03-25 Nouveaux taxoides, leur preparation et les compositions pharmaceutiques qui les contiennent

Publications (2)

Publication Number Publication Date
EE9700315A EE9700315A (et) 1998-06-15
EE03608B1 true EE03608B1 (et) 2002-02-15

Family

ID=26231838

Family Applications (2)

Application Number Title Priority Date Filing Date
EE9700315A EE03608B1 (et) 1995-03-27 1996-03-25 Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid
EE9700323A EE03609B1 (et) 1995-03-27 1996-03-25 Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid

Family Applications After (1)

Application Number Title Priority Date Filing Date
EE9700323A EE03609B1 (et) 1995-03-27 1996-03-25 Taksoidid, meetod nende valmistamiseks ja neid sisaldavad farmatseutilised kompositsioonid

Country Status (41)

Country Link
US (3) US5889043A (ko)
EP (2) EP0817779B1 (ko)
JP (2) JP2941951B2 (ko)
KR (2) KR100485309B1 (ko)
CN (2) CN1213042C (ko)
AP (2) AP785A (ko)
AR (1) AR001440A1 (ko)
AT (2) ATE188471T1 (ko)
AU (2) AU703278B2 (ko)
BG (2) BG63121B1 (ko)
BR (2) BR9607929A (ko)
CA (2) CA2214321C (ko)
CO (1) CO4700576A1 (ko)
CZ (2) CZ287468B6 (ko)
DE (2) DE69604653T2 (ko)
DK (2) DK0817779T3 (ko)
DZ (1) DZ2009A1 (ko)
EA (2) EA000567B1 (ko)
EE (2) EE03608B1 (ko)
ES (2) ES2140075T3 (ko)
GE (2) GEP20002211B (ko)
GR (2) GR3031526T3 (ko)
HU (2) HU223732B1 (ko)
IL (1) IL117636A (ko)
IS (2) IS2058B (ko)
MA (1) MA23823A1 (ko)
MY (1) MY121225A (ko)
NO (2) NO316379B1 (ko)
NZ (2) NZ304901A (ko)
OA (2) OA10513A (ko)
PE (1) PE51097A1 (ko)
PL (2) PL188284B1 (ko)
PT (1) PT817779E (ko)
RO (2) RO115878B1 (ko)
SK (2) SK281927B6 (ko)
TN (1) TNSN96043A1 (ko)
TR (2) TR199701040T1 (ko)
TW (1) TW394765B (ko)
UY (2) UY24192A1 (ko)
WO (2) WO1996030356A1 (ko)
ZA (1) ZA962399B (ko)

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US6495579B1 (en) 1996-12-02 2002-12-17 Angiotech Pharmaceuticals, Inc. Method for treating multiple sclerosis
US5811452A (en) * 1997-01-08 1998-09-22 The Research Foundation Of State University Of New York Taxoid reversal agents for drug-resistance in cancer chemotherapy and pharmaceutical compositions thereof
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US6346543B1 (en) * 1998-08-17 2002-02-12 Aventis Pharma S.A. Use of a taxoid to treat abnormal cell proliferation in the brain
EP0982027A1 (en) * 1998-08-17 2000-03-01 Aventis Pharma S.A. Taxoid derivatives for treating abnormal cell proliferation of the brain
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EP0982028A1 (en) * 1998-08-20 2000-03-01 Aventis Pharma S.A. New use of taxoid derivatives
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US6664275B2 (en) * 2000-02-02 2003-12-16 Fsu Research Foundation, Inc. C10 heterosubstituted acetate taxanes
US6649632B2 (en) 2000-02-02 2003-11-18 Fsu Research Foundation, Inc. C10 ester substituted taxanes
US8147816B2 (en) * 2000-08-16 2012-04-03 Encore Health, Llc Presbyopia treatment by lens alteration
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AU2001290636A1 (en) * 2000-09-22 2002-04-02 Bristol-Myers Squibb Company Method for reducing toxicity of combined chemotherapies
US6593334B1 (en) 2002-05-02 2003-07-15 The University Of North Carolina At Chapel Hill Camptothecin-taxoid conjugates as antimitotic and antitumor agents
CN102516417B (zh) 2002-09-06 2014-12-10 天蓝制药公司 用于传递治疗剂的以环糊精为基础的聚合物
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SV2006002010A (es) * 2004-02-13 2006-08-23 Univ Florida State Res Found Taxanos sustituidos con esteres de ciclopentilo en c10
GT200500025A (es) * 2004-02-13 2005-09-30 Taxanos sustituidos con esteres de ciclopentilo en c10
JP2008530122A (ja) * 2005-02-14 2008-08-07 フロリダ・ステイト・ユニバーシティ・リサーチ・ファウンデイション・インコーポレイテッド Ｃ１０シクロプロピルエステル置換タキサン組成物
RS52438B (en) * 2005-03-31 2013-02-28 Accord Healthcare Inc. PREPARATION OF 9-DIHYDRO-13-ACETYLBACCATINE TAXAN III
US8207358B2 (en) * 2005-11-04 2012-06-26 Accord Healthcare Ltd. Methods for the preparation of taxanes using chiral auxiliaries
US7847111B2 (en) * 2006-06-19 2010-12-07 Canada Inc. Semi-synthetic route for the preparation of paclitaxel, docetaxel, and 10-deacetylbaccatin III from 9-dihydro-13-acetylbaccatin III
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TWI526437B (zh) * 2011-09-09 2016-03-21 台灣神隆股份有限公司 卡巴他賽之結晶型
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CN102408397B (zh) 2011-10-19 2014-08-20 上海贝美医药科技有限公司 紫杉烷类衍生物及其制备方法
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CN104650012A (zh) * 2013-11-22 2015-05-27 天士力控股集团有限公司 一种紫杉烷类化合物
CN104086514A (zh) * 2014-06-19 2014-10-08 上海应用技术学院 紫杉醇衍生物及其制备方法
PL3258931T3 (pl) 2015-02-17 2020-12-28 Erasmus University Medical Center Rotterdam Zastosowanie kabazitakselu w leczeniu nowotworu złośliwego prostaty
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Also Published As

Publication number Publication date
RO115878B1 (ro) 2000-07-28
DE69604653T2 (de) 2000-05-31
TW394765B (en) 2000-06-21
US20020038038A1 (en) 2002-03-28
MA23823A1 (fr) 1996-10-01
NO316607B1 (no) 2004-03-08
AU711227B2 (en) 1999-10-07
DZ2009A1 (fr) 2002-10-23
CA2214321A1 (fr) 1996-10-03
AU5278196A (en) 1996-10-16
JP2941951B2 (ja) 1999-08-30
CZ303297A3 (cs) 1998-01-14
HUP9801204A3 (en) 2000-12-28
HU223666B1 (hu) 2004-11-29
UY24370A1 (es) 2001-10-25
NO973922D0 (no) 1997-08-26
HU223732B1 (hu) 2004-12-28
BG101918A (en) 1998-10-30
DE69606028T2 (de) 2000-08-10
PE51097A1 (es) 1997-12-22
HUP9801201A2 (hu) 2000-05-28
IS4567A (is) 1997-09-23
DE69606028D1 (de) 2000-02-10
HUP9801204A1 (hu) 2000-05-28
EA000567B1 (ru) 1999-12-29
EA199700269A1 (ru) 1998-04-30
EP0817779B1 (fr) 2000-01-05
HUP9801201A3 (en) 2000-12-28
EP0817780A1 (fr) 1998-01-14
DK0817779T3 (da) 2000-06-19
KR100297196B1 (ko) 2001-11-22
AR001440A1 (es) 1997-10-22
CZ287468B6 (en) 2000-12-13
EE9700323A (et) 1998-06-15
RO115877B1 (ro) 2000-07-28
GEP20002188B (en) 2000-07-25
NZ304900A (en) 1998-09-24
EA199700270A1 (ru) 1998-02-26
ATE188471T1 (de) 2000-01-15
NO973923D0 (no) 1997-08-26
OA10513A (fr) 2002-04-22
PL188284B1 (pl) 2005-01-31
BG101917A (en) 1998-10-30
SK130197A3 (en) 1998-04-08
EE03609B1 (et) 2002-02-15
MY121225A (en) 2006-01-28
PL322465A1 (en) 1998-02-02
BR9607930A (pt) 1998-06-02
US6387946B1 (en) 2002-05-14
MX9706568A (es) 1997-11-29
AU5278096A (en) 1996-10-16
IL117636A0 (en) 1996-07-23
AU703278B2 (en) 1999-03-25
CZ287326B6 (en) 2000-10-11
SK130297A3 (en) 1998-03-04
US6331635B1 (en) 2001-12-18
PL188987B1 (pl) 2005-05-31
TR199701040T1 (xx) 1998-01-21
EE9700315A (et) 1998-06-15
ES2140075T3 (es) 2000-02-16
CZ303097A3 (cs) 1998-01-14
CN1179775A (zh) 1998-04-22
JPH11500141A (ja) 1999-01-06
CA2214319A1 (fr) 1996-10-03
ATE185562T1 (de) 1999-10-15
NO973923L (no) 1997-08-26
DK0817780T3 (da) 2000-03-27
NO316379B1 (no) 2004-01-19
GR3032316T3 (en) 2000-04-27
IS2056B (is) 2005-10-14
KR19980703287A (ko) 1998-10-15
CN1152870C (zh) 2004-06-09
WO1996030355A1 (fr) 1996-10-03
ZA962399B (en) 1996-10-01
AP753A (en) 1999-07-21
CN1179776A (zh) 1998-04-22
BG63121B1 (bg) 2001-04-30
TNSN96043A1 (fr) 2005-03-15
US5889043A (en) 1999-03-30
EP0817779A1 (fr) 1998-01-14
CA2214319C (fr) 2004-02-17
BG63009B1 (bg) 2001-01-31
IL117636A (en) 2004-08-31
KR19980703357A (ko) 1998-10-15
SK281927B6 (sk) 2001-09-11
IS2058B (is) 2005-10-14
AP9701090A0 (en) 1997-10-31
TR199701042T1 (xx) 1998-01-21
MX9706278A (es) 1997-10-31
AP9701093A0 (en) 1997-10-31
CO4700576A1 (es) 1998-12-29
NZ304901A (en) 1998-12-23
PL322499A1 (en) 1998-02-02
AP785A (en) 1999-11-26
GR3031526T3 (en) 2000-01-31
EA000709B1 (ru) 2000-02-28
EP0817780B1 (fr) 1999-10-13
WO1996030356A1 (fr) 1996-10-03
GEP20002211B (en) 2000-08-25
IS4536A (is) 1997-07-31
SK281928B6 (sk) 2001-09-11
UY24192A1 (es) 1996-06-14
PT817779E (pt) 2000-04-28
CN1213042C (zh) 2005-08-03
JPH11502531A (ja) 1999-03-02
JP3790826B2 (ja) 2006-06-28
ES2143187T3 (es) 2000-05-01
DE69604653D1 (de) 1999-11-18
NO973922L (no) 1997-08-26
BR9607929A (pt) 1998-06-02
OA10514A (fr) 2002-04-22
KR100485309B1 (ko) 2005-10-12
CA2214321C (fr) 2008-01-22

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