EE03401B1 - Antibiootilist aktiivsust omavad erütromütsiini A 9-O-oksiimi derivaadid - Google Patents

Antibiootilist aktiivsust omavad erütromütsiini A 9-O-oksiimi derivaadid

Info

Publication number
EE03401B1
EE03401B1 EE9700124A EE9700124A EE03401B1 EE 03401 B1 EE03401 B1 EE 03401B1 EE 9700124 A EE9700124 A EE 9700124A EE 9700124 A EE9700124 A EE 9700124A EE 03401 B1 EE03401 B1 EE 03401B1
Authority
EE
Estonia
Prior art keywords
erythromycin
antibiotic activity
oxime derivatives
oxime
derivatives
Prior art date
Application number
EE9700124A
Other languages
English (en)
Estonian (et)
Other versions
EE9700124A (et
Inventor
Pellacini Franco
Schioppacassi Giovanna
Albini Enrico
Botta Daniela
Romagnano Stefano
Santangelo Francesco
Original Assignee
Zambon Group S.P.A.
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Zambon Group S.P.A. filed Critical Zambon Group S.P.A.
Publication of EE9700124A publication Critical patent/EE9700124A/xx
Publication of EE03401B1 publication Critical patent/EE03401B1/xx

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H17/00—Compounds containing heterocyclic radicals directly attached to hetero atoms of saccharide radicals
    • C07H17/04—Heterocyclic radicals containing only oxygen as ring hetero atoms
    • C07H17/08—Hetero rings containing eight or more ring members, e.g. erythromycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P33/00—Antiparasitic agents
    • A61P33/02—Antiprotozoals, e.g. for leishmaniasis, trichomoniasis, toxoplasmosis
    • Y—GENERAL TAGGING OF NEW TECHNOLOGICAL DEVELOPMENTS; GENERAL TAGGING OF CROSS-SECTIONAL TECHNOLOGIES SPANNING OVER SEVERAL SECTIONS OF THE IPC; TECHNICAL SUBJECTS COVERED BY FORMER USPC CROSS-REFERENCE ART COLLECTIONS [XRACs] AND DIGESTS
    • Y02—TECHNOLOGIES OR APPLICATIONS FOR MITIGATION OR ADAPTATION AGAINST CLIMATE CHANGE
    • Y02A—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE
    • Y02A50/00—TECHNOLOGIES FOR ADAPTATION TO CLIMATE CHANGE in human health protection, e.g. against extreme weather
    • Y02A50/30—Against vector-borne diseases, e.g. mosquito-borne, fly-borne, tick-borne or waterborne diseases whose impact is exacerbated by climate change

Landscapes

  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • General Chemical & Material Sciences (AREA)
  • Genetics & Genomics (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Animal Behavior & Ethology (AREA)
  • Molecular Biology (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Biochemistry (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Tropical Medicine & Parasitology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
EE9700124A 1994-12-13 1995-12-07 Antibiootilist aktiivsust omavad erütromütsiini A 9-O-oksiimi derivaadid EE03401B1 (et)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
IT94MI002496A IT1276901B1 (it) 1994-12-13 1994-12-13 Derivati dell'eritromicina a 9-0-ossina dotati di attivita' antibiotica
PCT/EP1995/004815 WO1996018633A1 (en) 1994-12-13 1995-12-07 Erythromycin a 9-0-oxime derivatives endowed with antibiotic activity

Publications (2)

Publication Number Publication Date
EE9700124A EE9700124A (et) 1997-12-15
EE03401B1 true EE03401B1 (et) 2001-04-16

Family

ID=11369979

Family Applications (1)

Application Number Title Priority Date Filing Date
EE9700124A EE03401B1 (et) 1994-12-13 1995-12-07 Antibiootilist aktiivsust omavad erütromütsiini A 9-O-oksiimi derivaadid

Country Status (35)

Country Link
US (1) US5847092A (de)
EP (1) EP0797579B1 (de)
JP (1) JPH10510520A (de)
KR (1) KR100367559B1 (de)
CN (1) CN1046535C (de)
AP (1) AP739A (de)
AT (1) ATE190620T1 (de)
AU (1) AU690791B2 (de)
BG (1) BG63261B1 (de)
BR (1) BR9510015A (de)
CA (1) CA2207029A1 (de)
CZ (1) CZ289943B6 (de)
DE (1) DE69515694T2 (de)
DK (1) DK0797579T3 (de)
EE (1) EE03401B1 (de)
ES (1) ES2144154T3 (de)
FI (1) FI972493A (de)
GE (1) GEP20012391B (de)
GR (1) GR3033622T3 (de)
HU (1) HU220631B1 (de)
IT (1) IT1276901B1 (de)
LT (1) LT4276B (de)
LV (1) LV11898B (de)
MD (1) MD1788G2 (de)
NO (1) NO309816B1 (de)
NZ (1) NZ297446A (de)
OA (1) OA10491A (de)
PL (1) PL182053B1 (de)
PT (1) PT797579E (de)
RO (1) RO116282B1 (de)
RU (1) RU2152951C1 (de)
SI (1) SI9520124A (de)
TJ (1) TJ306B (de)
UA (1) UA48958C2 (de)
WO (1) WO1996018633A1 (de)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1290447B1 (it) 1997-03-28 1998-12-03 Zambon Spa Derivati 1,3-ossatiolanici ad attivita' antivirale
IT1301967B1 (it) * 1998-07-30 2000-07-20 Zambon Spa Derivato di eritromicina ad attivita' antibiotica
IT1301968B1 (it) * 1998-07-30 2000-07-20 Zambon Spa Derivati di eritromicina ad attivita' antibiotica
IT1306205B1 (it) * 1999-01-15 2001-05-30 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.
US6638908B1 (en) 2000-08-09 2003-10-28 Yale University Crystals of the large ribosomal subunit
US6947844B2 (en) 2000-08-09 2005-09-20 Yale University Modulators of ribosomal function and identification thereof
IL151012A0 (en) 2001-08-03 2003-02-12 Ribosomes Structure And Protei Ribosomes structure and protein synthesis inhibitors
US6952650B2 (en) 2001-08-03 2005-10-04 Yale University Modulators of ribosomal function and identification thereof
ITMI20021726A1 (it) 2002-08-01 2004-02-02 Zambon Spa Macrolidi ad attivita' antiinfiammatoria.
TW200420573A (en) 2002-09-26 2004-10-16 Rib X Pharmaceuticals Inc Bifunctional heterocyclic compounds and methods of making and using same
US8202843B2 (en) 2004-02-27 2012-06-19 Rib-X Pharmaceuticals, Inc. Macrocyclic compounds and methods of making and using the same

Family Cites Families (6)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2473525A1 (fr) * 1980-01-11 1981-07-17 Roussel Uclaf Nouvelles oximes derivees de l'erythromycine, leur procede de preparation et leur application comme medicaments
GB8521402D0 (en) 1985-08-28 1985-10-02 Beecham Group Plc Chemical compounds
US4740502A (en) * 1986-06-20 1988-04-26 Abbott Laboratories Semisynthetic erythromycin antibiotics
DK90788A (da) 1987-02-24 1988-08-25 Beecham Group Plc Erythromycinderivater
US5302705A (en) * 1989-10-07 1994-04-12 Taisho Pharmaceutical Co., Ltd. 6-O-methylerythromycin a oxime derivatives
IL99995A (en) * 1990-11-21 1997-11-20 Roussel Uclaf Erythromycin derivatives, their preparation and pharmaceutical compositions containing them

Also Published As

Publication number Publication date
BG101570A (en) 1998-02-27
LV11898B (en) 1998-03-20
BR9510015A (pt) 1997-10-28
AU690791B2 (en) 1998-04-30
AP739A (en) 1999-03-24
CA2207029A1 (en) 1996-06-20
CN1169727A (zh) 1998-01-07
KR100367559B1 (ko) 2003-04-21
FI972493A0 (fi) 1997-06-12
MD1788F2 (en) 2001-11-30
MD1788G2 (ro) 2002-05-31
RO116282B1 (ro) 2000-12-29
EE9700124A (et) 1997-12-15
NZ297446A (en) 1999-06-29
US5847092A (en) 1998-12-08
GEP20012391B (en) 2001-03-25
BG63261B1 (bg) 2001-07-31
MD970243A (en) 1999-05-31
RU2152951C1 (ru) 2000-07-20
PL182053B1 (pl) 2001-10-31
EP0797579A1 (de) 1997-10-01
PL320688A1 (en) 1997-10-27
CZ178697A3 (en) 1997-12-17
TJ306B (en) 2001-08-06
SI9520124A (sl) 1998-04-30
ATE190620T1 (de) 2000-04-15
JPH10510520A (ja) 1998-10-13
CZ289943B6 (cs) 2002-04-17
MX9704253A (es) 1997-09-30
HU220631B1 (hu) 2002-03-28
UA48958C2 (uk) 2002-09-16
NO309816B1 (no) 2001-04-02
PT797579E (pt) 2000-08-31
GR3033622T3 (en) 2000-10-31
DE69515694D1 (de) 2000-04-20
DE69515694T2 (de) 2000-10-26
DK0797579T3 (da) 2000-06-05
NO972702D0 (no) 1997-06-12
LT4276B (lt) 1998-01-26
EP0797579B1 (de) 2000-03-15
ES2144154T3 (es) 2000-06-01
ITMI942496A0 (it) 1994-12-13
LV11898A (lv) 1997-12-20
AP9700989A0 (en) 1997-07-31
HUT77126A (hu) 1998-03-02
IT1276901B1 (it) 1997-11-03
WO1996018633A1 (en) 1996-06-20
NO972702L (no) 1997-08-13
AU4260396A (en) 1996-07-03
ITMI942496A1 (it) 1996-06-13
CN1046535C (zh) 1999-11-17
FI972493A (fi) 1997-06-12
OA10491A (en) 2002-04-10
LT97116A (en) 1997-10-27

Similar Documents

Publication Publication Date Title
LV11739A (lv) Eritromicina atvasinajumi iegusanas panemiens un pielietojums
ATE310742T1 (de) C-4ß-SUBSTITUTIERTE MACROLID-DERIVATE
IS5251A (is) 9-oxím erýþrómýsín afleiður
LV11547A (lv) Makrolidi ar imunodepresantu aktivitati
PT788511E (pt) Hexapeptidos ciclicos com actividade antibiotica
NO993876D0 (no) 3'-N-oksid, 3'-N-dimetylamin, 9-oksim erytromycin A derivater
IL129946A0 (en) Erythromycin a derivatives
NO980016D0 (no) Makrolider
DE69821009D1 (de) 6,9-verbrückte erythromycin-derivate
PT1025114E (pt) Derivados de eritromicina-cetolido 6-o-substituido 3'-n-modificados possuindo actividade antibacteriana
ATE210666T1 (de) Cephalosporinantibiotika
ATE239750T1 (de) 6,11-verbrückte erythromycinderivate
FI102508B3 (fi) Vuodejärjestelmä
EE03401B1 (et) Antibiootilist aktiivsust omavad erütromütsiini A 9-O-oksiimi derivaadid
NO934264L (no) Antibiotiske forbindelser
ZA989835B (en) Erythromycin a derivatives
ZA989830B (en) Erythromycin a derivatives
AU6421398A (en) Erythromycin a derivatives
ZA981572B (en) Erythromycin a derivatives
IL115312A0 (en) Antibiotic macrolides
PT984975E (pt) Derivados de eritromicina multiciclicos
LV10450A (lv) O-heteroaril- O-alkilheteroaril- O-alkenilheteroaril- un O-alkinilheteroaril- makrolidi
SI1100806T1 (en) Erythromycin derivative with antibiotic activity
AU9645998A (en) Erythromycin a derivatives
ZA951845B (en) Acid-stabile erythromycin derivatives

Legal Events

Date Code Title Description
KB4A Valid patent at the end of a year

Effective date: 20021231

KB4A Valid patent at the end of a year

Effective date: 20031231

KB4A Valid patent at the end of a year

Effective date: 20041231

KB4A Valid patent at the end of a year

Effective date: 20051231

MM4A Lapsed by not paying the annual fees

Effective date: 20051207