EA004403B1 - Производные пиразолотриазинов, фармацевтические композиции, содержащие их, способы лечения - Google Patents
Производные пиразолотриазинов, фармацевтические композиции, содержащие их, способы лечения Download PDFInfo
- Publication number
- EA004403B1 EA004403B1 EA199900158A EA199900158A EA004403B1 EA 004403 B1 EA004403 B1 EA 004403B1 EA 199900158 A EA199900158 A EA 199900158A EA 199900158 A EA199900158 A EA 199900158A EA 004403 B1 EA004403 B1 EA 004403B1
- Authority
- EA
- Eurasian Patent Office
- Prior art keywords
- denotes
- compound
- formula
- stands
- ome
- Prior art date
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- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Plural Heterocyclic Compounds (AREA)
- Polymers With Sulfur, Phosphorus Or Metals In The Main Chain (AREA)
- Macromolecular Compounds Obtained By Forming Nitrogen-Containing Linkages In General (AREA)
- Agricultural Chemicals And Associated Chemicals (AREA)
- Detergent Compositions (AREA)
- Coloring (AREA)
Applications Claiming Priority (4)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| US68604796A | 1996-07-24 | 1996-07-24 | |
| US2329096P | 1996-07-24 | 1996-07-24 | |
| PCT/US1997/013072 WO1998003510A1 (fr) | 1996-07-24 | 1997-07-23 | Azolo triazines et pyrimidines |
| US08/899,242 US6124289A (en) | 1996-07-24 | 1997-07-23 | Azolo triazines and pyrimidines |
Publications (2)
| Publication Number | Publication Date |
|---|---|
| EA199900158A1 EA199900158A1 (ru) | 1999-10-28 |
| EA004403B1 true EA004403B1 (ru) | 2004-04-29 |
Family
ID=27362048
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| EA199900158A EA004403B1 (ru) | 1996-07-24 | 1997-07-23 | Производные пиразолотриазинов, фармацевтические композиции, содержащие их, способы лечения |
Country Status (15)
| Country | Link |
|---|---|
| JP (2) | JP4704521B2 (fr) |
| CN (3) | CN1104432C (fr) |
| AR (1) | AR049583A2 (fr) |
| BR (1) | BR9710544A (fr) |
| CA (1) | CA2259583C (fr) |
| CZ (1) | CZ299451B6 (fr) |
| EA (1) | EA004403B1 (fr) |
| EE (1) | EE04316B1 (fr) |
| HR (1) | HRP970413A2 (fr) |
| IL (4) | IL127871A0 (fr) |
| NO (1) | NO315610B3 (fr) |
| NZ (1) | NZ333777A (fr) |
| PL (1) | PL195762B1 (fr) |
| SI (1) | SI9720045B (fr) |
| SK (1) | SK286461B6 (fr) |
Families Citing this family (10)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| WO2002072202A1 (fr) * | 2001-03-13 | 2002-09-19 | Bristol-Myers Squibb Pharma Company | 4-(2-butylamino)-2,7-dimethyl-8-(2-methyl-6-methoxypyrid-3-yl) pyrazolo-[1,5-a]-1,3,5-triazine, ses enantiomeres et sels pharmaceutiquement acceptables en tant que ligands du recepteur de la corticoliberine |
| WO2004110454A1 (fr) * | 2003-06-13 | 2004-12-23 | Ishihara Sangyo Kaisha, Ltd. | Composition de traitement ou de prevention de maladies necessitant l'administration d'un agoniste du recepteur a2a de l'adenosine |
| US7329662B2 (en) * | 2003-10-03 | 2008-02-12 | Hoffmann-La Roche Inc. | Pyrazolo-pyridine |
| GB0519957D0 (en) * | 2005-09-30 | 2005-11-09 | Sb Pharmco Inc | Chemical compound |
| DK2094709T3 (da) * | 2006-09-20 | 2010-12-06 | Lilly Co Eli | Thiazol-pyrazolopyrimidiner som CRF1-receptorantagonister |
| CN103694242B (zh) * | 2013-12-10 | 2016-01-06 | 昆明翔昊科技有限公司 | 吡唑并嘧啶类化合物及其药物组合物和其在制药中的应用 |
| EP3628005A4 (fr) | 2017-08-14 | 2021-01-20 | Spruce Biosciences, Inc. | Antagonistes du récepteur du facteur de libération de la corticotropine |
| CN112479956A (zh) * | 2019-07-30 | 2021-03-12 | 杭州阿诺生物医药科技有限公司 | 一种用于制备腺苷受体抑制剂中间体的方法 |
| WO2022036123A1 (fr) | 2020-08-12 | 2022-02-17 | Spruce Biosciences, Inc. | Procédés et compositions pour traiter le syndrome des ovaires polykystiques |
| US11708372B2 (en) | 2021-11-19 | 2023-07-25 | Spruce Biosciences, Inc. | Crystalline composition of tildacerfont and methods of use and preparation thereof |
Family Cites Families (7)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| US3995039A (en) * | 1975-05-27 | 1976-11-30 | Merck & Co., Inc. | Pyrazolo [1,5-a] [1,3,5] triazines |
| JPS6157587A (ja) * | 1984-08-29 | 1986-03-24 | Shionogi & Co Ltd | 縮合複素環誘導体および抗潰瘍剤 |
| US4824834A (en) * | 1986-10-31 | 1989-04-25 | Otsuka Pharmaceutical Company, Limited | Pyrazolotriazine compounds |
| JP2691317B2 (ja) * | 1989-08-25 | 1997-12-17 | 株式会社大塚製薬工場 | ４―ヒドロキシ―８―（３―低級アルコキシ―４―フェニルスルフィニルフェニル）ピラゾロ〔１，５―ａ〕―１，３，５―トリアジン光学活性体の塩類及びその製造方法 |
| US5420128A (en) * | 1990-10-09 | 1995-05-30 | Otsuka Pharmaceutical Co., Ltd. | Pyrimidine derivatives, method of manufacturing the same, and androgen inhibitor |
| DE69130683T2 (de) * | 1991-04-22 | 1999-05-06 | Otsuka Pharmaceutical Factory, Inc., Naruto, Tokushima | PYRAZOLO[1,5-a]PYRIMIDINDERIVATE UND SIE ENTHALTENDE ANTIINFLAMMATORISCHE MITTEL |
| US5356897A (en) * | 1991-09-09 | 1994-10-18 | Fujisawa Pharmaceutical Co., Ltd. | 3-(heteroaryl)-pyrazololi[1,5-a]pyrimidines |
-
1997
- 1997-07-23 CZ CZ0018499A patent/CZ299451B6/cs not_active IP Right Cessation
- 1997-07-23 NZ NZ333777A patent/NZ333777A/en not_active IP Right Cessation
- 1997-07-23 BR BR9710544A patent/BR9710544A/pt not_active IP Right Cessation
- 1997-07-23 EA EA199900158A patent/EA004403B1/ru not_active IP Right Cessation
- 1997-07-23 JP JP50723398A patent/JP4704521B2/ja not_active Expired - Fee Related
- 1997-07-23 EE EEP199900019A patent/EE04316B1/xx unknown
- 1997-07-23 IL IL12787197A patent/IL127871A0/xx unknown
- 1997-07-23 PL PL97331523A patent/PL195762B1/pl unknown
- 1997-07-23 SK SK97-99A patent/SK286461B6/sk not_active IP Right Cessation
- 1997-07-23 CA CA002259583A patent/CA2259583C/fr not_active Expired - Lifetime
- 1997-07-23 SI SI9720045A patent/SI9720045B/sl active Search and Examination
- 1997-07-23 CN CN97196525A patent/CN1104432C/zh not_active Expired - Lifetime
- 1997-07-24 HR HRP970413 patent/HRP970413A2/hr not_active Application Discontinuation
-
1998
- 1998-12-30 IL IL127871A patent/IL127871A/en not_active IP Right Cessation
-
1999
- 1999-01-21 NO NO19990264A patent/NO315610B3/no not_active IP Right Cessation
-
2001
- 2001-05-30 CN CN 01120849 patent/CN1250223C/zh not_active Expired - Lifetime
-
2002
- 2002-04-25 CN CN 02118589 patent/CN1388126A/zh active Pending
- 2002-06-11 IL IL150163A patent/IL150163A/en not_active IP Right Cessation
-
2004
- 2004-07-23 JP JP2004216483A patent/JP4194539B2/ja not_active Expired - Fee Related
- 2004-10-12 IL IL164513A patent/IL164513A/en not_active IP Right Cessation
-
2005
- 2005-07-11 AR ARP050102868A patent/AR049583A2/es not_active Application Discontinuation
Also Published As
| Publication number | Publication date |
|---|---|
| NZ333777A (en) | 2000-07-28 |
| HRP970413A2 (en) | 1998-10-31 |
| IL164513A0 (en) | 2005-12-18 |
| CN1250223C (zh) | 2006-04-12 |
| CZ18499A3 (cs) | 1999-11-17 |
| IL127871A (en) | 2010-04-29 |
| JP2005097257A (ja) | 2005-04-14 |
| IL127871A0 (en) | 1999-10-28 |
| SK9799A3 (sk) | 2005-04-01 |
| EE04316B1 (et) | 2004-06-15 |
| NO315610B1 (no) | 2003-09-29 |
| SI9720045A (sl) | 1999-10-31 |
| EA199900158A1 (ru) | 1999-10-28 |
| NO990264L (no) | 1999-03-10 |
| CN1327793A (zh) | 2001-12-26 |
| CZ299451B6 (cs) | 2008-07-30 |
| CN1225637A (zh) | 1999-08-11 |
| JP4194539B2 (ja) | 2008-12-10 |
| SI9720045B (sl) | 2008-02-29 |
| NO315610B3 (no) | 2003-09-29 |
| EE9900019A (et) | 1999-08-16 |
| JP2002513382A (ja) | 2002-05-08 |
| AR049583A2 (es) | 2006-08-16 |
| SK286461B6 (sk) | 2008-10-07 |
| IL164513A (en) | 2010-04-29 |
| NO990264D0 (no) | 1999-01-21 |
| PL195762B1 (pl) | 2007-10-31 |
| CN1388126A (zh) | 2003-01-01 |
| IL150163A (en) | 2010-12-30 |
| BR9710544A (pt) | 1999-08-17 |
| CN1104432C (zh) | 2003-04-02 |
| PL331523A1 (en) | 1999-07-19 |
| JP4704521B2 (ja) | 2011-06-15 |
| CA2259583A1 (fr) | 1998-01-29 |
| CA2259583C (fr) | 2009-11-17 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| MK4A | Patent expired |
Designated state(s): AM AZ BY KZ KG MD TJ TM RU |