DOP2009000240A - Compuestos triciclicos que contienen nitrogeno como agentes antibacterianos - Google Patents

Compuestos triciclicos que contienen nitrogeno como agentes antibacterianos

Info

Publication number
DOP2009000240A
DOP2009000240A DO2009000240A DO2009000240A DOP2009000240A DO P2009000240 A DOP2009000240 A DO P2009000240A DO 2009000240 A DO2009000240 A DO 2009000240A DO 2009000240 A DO2009000240 A DO 2009000240A DO P2009000240 A DOP2009000240 A DO P2009000240A
Authority
DO
Dominican Republic
Prior art keywords
antibacterial agents
compounds containing
containing nitrogen
tricycle
tricycle compounds
Prior art date
Application number
DO2009000240A
Other languages
English (en)
Spanish (es)
Inventor
David Egan Davies
David Thomas Davies
Llaria Giordano
Alan Joseph Hennessy
Neil David Pearson
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Family has litigation
First worldwide family litigation filed litigation Critical https://patents.darts-ip.com/?family=39580226&utm_source=google_patent&utm_medium=platform_link&utm_campaign=public_patent_search&patent=DOP2009000240(A) "Global patent litigation dataset” by Darts-ip is licensed under a Creative Commons Attribution 4.0 International License.
Priority claimed from GB0707705A external-priority patent/GB0707705D0/en
Priority claimed from GB0720569A external-priority patent/GB0720569D0/en
Priority claimed from GB0805311A external-priority patent/GB0805311D0/en
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of DOP2009000240A publication Critical patent/DOP2009000240A/es

Links

Classifications

    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D471/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains three hetero rings
    • C07D471/16Peri-condensed systems
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04Antibacterial agents
    • A61P31/06Antibacterial agents for tuberculosis
    • AHUMAN NECESSITIES
    • A61MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61PSPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/12Antivirals
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D487/00Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/12Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains three hetero rings
    • C07D487/16Peri-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D519/00Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Communicable Diseases (AREA)
  • Veterinary Medicine (AREA)
  • Animal Behavior & Ethology (AREA)
  • Oncology (AREA)
  • Public Health (AREA)
  • Pulmonology (AREA)
  • Virology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Agricultural Chemicals And Associated Chemicals (AREA)
  • Medicines Containing Material From Animals Or Micro-Organisms (AREA)
DO2009000240A 2007-04-20 2009-10-09 Compuestos triciclicos que contienen nitrogeno como agentes antibacterianos DOP2009000240A (es)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
GB0707705A GB0707705D0 (en) 2007-04-20 2007-04-20 Compounds
GB0720569A GB0720569D0 (en) 2007-10-19 2007-10-19 Compounds
GB0805311A GB0805311D0 (en) 2008-03-20 2008-03-20 Compounds

Publications (1)

Publication Number Publication Date
DOP2009000240A true DOP2009000240A (es) 2009-12-31

Family

ID=39580226

Family Applications (1)

Application Number Title Priority Date Filing Date
DO2009000240A DOP2009000240A (es) 2007-04-20 2009-10-09 Compuestos triciclicos que contienen nitrogeno como agentes antibacterianos

Country Status (31)

Country Link
US (1) US8389524B2 (enExample)
EP (1) EP2137196B1 (enExample)
JP (1) JP5389013B2 (enExample)
KR (1) KR101567096B1 (enExample)
CN (1) CN101687887B (enExample)
AR (1) AR066111A1 (enExample)
AT (1) ATE483717T1 (enExample)
AU (1) AU2008240764C1 (enExample)
BR (1) BRPI0810064B8 (enExample)
CA (1) CA2684659C (enExample)
CL (1) CL2008001122A1 (enExample)
CO (1) CO6251368A2 (enExample)
CR (2) CR11123A (enExample)
CY (1) CY1111248T1 (enExample)
DE (1) DE602008002912D1 (enExample)
DK (1) DK2137196T3 (enExample)
DO (1) DOP2009000240A (enExample)
EA (1) EA015821B1 (enExample)
HR (1) HRP20100574T1 (enExample)
IL (1) IL201204A0 (enExample)
MA (1) MA31324B1 (enExample)
MX (1) MX2009011317A (enExample)
MY (1) MY149347A (enExample)
NZ (1) NZ579877A (enExample)
PE (1) PE20090274A1 (enExample)
PL (1) PL2137196T3 (enExample)
PT (1) PT2137196E (enExample)
SI (1) SI2137196T1 (enExample)
TW (1) TWI431006B (enExample)
UY (1) UY31038A1 (enExample)
WO (1) WO2008128942A1 (enExample)

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WO2009050236A1 (de) 2007-10-19 2009-04-23 Boehringer Ingelheim International Gmbh Neue piperazino-dihydrothienopyrimidin-derivate
WO2009050248A1 (de) 2007-10-19 2009-04-23 Boehringer Ingelheim International Gmbh Substituierte piperidino-dihydrothienopyrimidine
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WO2009141399A1 (en) * 2008-05-23 2009-11-26 Glaxo Group Limited Tricyclic nitrogen containing compounds and their use as antibacterials
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US9802954B2 (en) 2011-08-24 2017-10-31 Boehringer Ingelheim International Gmbh Piperidino-dihydrothienopyrimidine sulfoxides and their use for treating COPD and asthma
US20130059866A1 (en) 2011-08-24 2013-03-07 Boehringer Ingelheim International Gmbh Novel piperidino-dihydrothienopyrimidine sulfoxides and their use for treating copd and asthma
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EP3612513A4 (en) 2017-04-17 2020-09-30 Ohio State Innovation Foundation TYPE II TOPOISOMERASE INHIBITORS AND METHOD OF MANUFACTURING AND USING THEREOF
JP2022528890A (ja) * 2019-04-03 2022-06-16 グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッド 細菌性尿路感染症の治療に使用するためのゲポチダシン
ES2981617T3 (es) 2019-07-05 2024-10-09 Glaxosmithkline Intellectual Property Dev Combinación para el tratamiento de infecciones provocadas por Mycoplasma genitalium
JP2023528560A (ja) 2020-04-02 2023-07-05 グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッド ゲポチダシンを用いて淋菌感染症を治療するためのレジメン
EP4143188A1 (en) * 2020-04-29 2023-03-08 GlaxoSmithKline Intellectual Property Development Limited Crystalline forms of gepotidacin
CN111494241B (zh) * 2020-06-01 2023-03-24 湖北洁世达环保科技有限公司 一种纸巾柔润保湿液
WO2022167515A1 (en) 2021-02-05 2022-08-11 Glaxosmithkline Intellectual Property Development Limited Oral solid dose formulations
JP2025502442A (ja) 2022-01-21 2025-01-24 グラクソスミスクライン、インテレクチュアル、プロパティー、ディベロップメント、リミテッド Staphylococcus saprophyticusによって引き起こされる感染症の処置における使用のためのゲポチダシンおよびバンコマイシン
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Also Published As

Publication number Publication date
BRPI0810064A2 (pt) 2019-08-27
WO2008128942A1 (en) 2008-10-30
EA015821B1 (ru) 2011-12-30
IL201204A0 (en) 2010-05-17
ATE483717T1 (de) 2010-10-15
JP5389013B2 (ja) 2014-01-15
EP2137196A1 (en) 2009-12-30
AU2008240764B2 (en) 2011-04-07
EA200970987A1 (ru) 2010-04-30
CN101687887A (zh) 2010-03-31
US20100137282A1 (en) 2010-06-03
KR20100017133A (ko) 2010-02-16
PT2137196E (pt) 2010-12-16
NZ579877A (en) 2011-09-30
CO6251368A2 (es) 2011-02-21
CA2684659C (en) 2015-11-24
TWI431006B (zh) 2014-03-21
CN101687887B (zh) 2012-08-29
AU2008240764C1 (en) 2011-10-20
AR066111A1 (es) 2009-07-22
HK1138000A1 (en) 2010-08-13
KR101567096B1 (ko) 2015-11-06
CA2684659A1 (en) 2008-10-30
AU2008240764A1 (en) 2008-10-30
CL2008001122A1 (es) 2008-10-24
TW200848420A (en) 2008-12-16
UY31038A1 (es) 2008-11-28
CR11123A (es) 2010-03-08
CR20150586A (es) 2016-04-04
CY1111248T1 (el) 2015-06-11
BRPI0810064B1 (pt) 2021-03-30
HRP20100574T1 (hr) 2010-12-31
SI2137196T1 (sl) 2011-01-31
JP2010524884A (ja) 2010-07-22
PL2137196T3 (pl) 2011-03-31
DE602008002912D1 (de) 2010-11-18
EP2137196B1 (en) 2010-10-06
DK2137196T3 (da) 2011-01-10
MX2009011317A (es) 2009-11-05
MA31324B1 (fr) 2010-04-01
MY149347A (en) 2013-08-30
BRPI0810064B8 (pt) 2021-05-25
PE20090274A1 (es) 2009-04-03
US8389524B2 (en) 2013-03-05

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