CR9930A - Compuestos - Google Patents

Compuestos

Info

Publication number
CR9930A
CR9930A CR9930A CR9930A CR9930A CR 9930 A CR9930 A CR 9930A CR 9930 A CR9930 A CR 9930A CR 9930 A CR9930 A CR 9930A CR 9930 A CR9930 A CR 9930A
Authority
CR
Costa Rica
Prior art keywords
compounds
antibacterials
compounds containing
containing tricyclic
tricyclic nitrogen
Prior art date
Application number
CR9930A
Other languages
English (en)
Inventor
Nathalie Cailleau
David Thomas Davies
Joel Michael Esken
Alan Joseph Hennessy
Sukumar Senthil Kumar Kusalakumari
Roger Edward Markwell
Timothy James Miles
Neil David Pearson
Original Assignee
Glaxo Group Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Glaxo Group Ltd filed Critical Glaxo Group Ltd
Publication of CR9930A publication Critical patent/CR9930A/es

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D471/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00
    • C07D471/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, at least one ring being a six-membered ring with one nitrogen atom, not provided for by groups C07D451/00 - C07D463/00 in which the condensed system contains two hetero rings
    • C07D471/06—Peri-condensed systems
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/435—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom
    • A61K31/4353—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems
    • A61K31/436—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with one nitrogen as the only ring hetero atom ortho- or peri-condensed with heterocyclic ring systems the heterocyclic ring system containing a six-membered ring having oxygen as a ring hetero atom, e.g. rapamycin
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P31/00—Antiinfectives, i.e. antibiotics, antiseptics, chemotherapeutics
    • A61P31/04—Antibacterial agents
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D519/00—Heterocyclic compounds containing more than one system of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring system not provided for in groups C07D453/00 or C07D455/00

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • General Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • General Chemical & Material Sciences (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Oncology (AREA)
  • Communicable Diseases (AREA)
  • Epidemiology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)

Abstract

Compuestos que contienen nitrogeno triciclico y sus usos como antibacterianos.
CR9930A 2005-10-21 2008-04-25 Compuestos CR9930A (es)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US72897505P 2005-10-21 2005-10-21
US82659006P 2006-09-22 2006-09-22

Publications (1)

Publication Number Publication Date
CR9930A true CR9930A (es) 2008-07-29

Family

ID=38256822

Family Applications (1)

Application Number Title Priority Date Filing Date
CR9930A CR9930A (es) 2005-10-21 2008-04-25 Compuestos

Country Status (27)

Country Link
US (2) US20080221110A1 (es)
EP (1) EP1954697B1 (es)
JP (1) JP2009512695A (es)
KR (1) KR20080064173A (es)
AR (1) AR057981A1 (es)
AT (1) ATE458737T1 (es)
AU (1) AU2006335042A1 (es)
BR (1) BRPI0617467A2 (es)
CA (1) CA2626641A1 (es)
CR (1) CR9930A (es)
CY (1) CY1110137T1 (es)
DE (1) DE602006012535D1 (es)
DK (1) DK1954697T3 (es)
EA (1) EA200801128A1 (es)
ES (1) ES2340531T3 (es)
HK (1) HK1118546A1 (es)
HR (1) HRP20100194T8 (es)
IL (1) IL190803A0 (es)
MA (1) MA29873B1 (es)
NO (1) NO20082191L (es)
NZ (1) NZ567315A (es)
PE (1) PE20070793A1 (es)
PL (1) PL1954697T3 (es)
PT (1) PT1954697E (es)
SI (1) SI1954697T1 (es)
TW (1) TW200736263A (es)
WO (1) WO2007081597A2 (es)

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ATE481406T1 (de) 2006-04-06 2010-10-15 Glaxo Group Ltd Pyrrolochinoxalinonderivate als antibakterielle mittel
GB0608263D0 (en) 2006-04-26 2006-06-07 Glaxo Group Ltd Compounds
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GB0705672D0 (en) * 2007-03-23 2007-05-02 Glaxo Group Ltd Compounds
CL2008001002A1 (es) 2007-04-11 2008-10-17 Actelion Pharmaceuticals Ltd Compuestos derivados de oxazolidinona; composicion farmaceutica que comprende a dichos compuestos; y su uso para preparar un medicamento para tratar una infeccion bacteriana.
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TW200940551A (en) 2008-02-20 2009-10-01 Actelion Pharmaceuticals Ltd Azatricyclic antibiotic compounds
US8012961B2 (en) 2008-04-15 2011-09-06 Actelion Pharmaceutical Ltd. Tricyclic antibiotics
JP2011529960A (ja) 2008-08-04 2011-12-15 アクテリオン ファーマシューティカルズ リミテッド 三環式アルキルアミノメチルオキサゾリジノン誘導体
EP2344495B1 (en) 2008-10-07 2014-12-31 Actelion Pharmaceuticals Ltd. Tricyclic oxazolidinone antibiotic compounds
JP2012505866A (ja) * 2008-10-17 2012-03-08 グラクソ グループ リミテッド 抗菌剤として使用される三環式窒素化合物
TWI426076B (zh) 2008-12-12 2014-02-11 Actelion Pharmaceuticals Ltd ５－胺基－２－（１－羥基－乙基）－四氫哌喃衍生物
JP5653935B2 (ja) 2009-01-15 2015-01-14 グラクソ グループ リミテッドＧｌａｘｏ Ｇｒｏｕｐ Ｌｉｍｉｔｅｄ 抗菌薬として有用なナフチリジン―２（１ｈ）−オン化合物
WO2013038374A1 (en) 2011-09-16 2013-03-21 Actelion Pharmaceuticals Ltd Process for manufacturing a synthetic intermediate
JP2014533747A (ja) 2011-11-30 2014-12-15 アクテリオン ファーマシューティカルズ リミテッドＡｃｔｅｌｉｏｎ Ｐｈａｒｍａｃｅｕｔｉｃａｌｓ Ｌｔｄ ３，７−二置換オクタヒドロ−２Ｈ−ピリド［４，３−ｅ］［１，３］オキサジン−２−オン抗生物質
ES2759303T3 (es) 2014-08-22 2020-05-08 Glaxosmithkline Ip Dev Ltd Compuestos tricíclicos que contienen nitrógeno para tratar infección por Neisseria gonorrhoeae
BR112019017522B1 (pt) 2017-02-28 2023-11-28 Mitsui Chemicals Agro, Inc Métodos para o controle de doenças de planta mediante a sua aplicação
CA3063037A1 (en) * 2017-05-10 2018-11-15 Albajuna Therapeutics, S.L. Fc-fusion protein derivatives with high dual hiv antiviral and immunomodulatory activity
IL293340A (en) 2019-12-02 2022-07-01 Storm Therapeutics Ltd Polyheterocyclic compounds as mettl3 inhibitors
CA3164134A1 (en) 2019-12-06 2021-06-10 Vertex Pharmaceuticals Incorporated Substituted tetrahydrofurans as modulators of sodium channels

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ATE481406T1 (de) * 2006-04-06 2010-10-15 Glaxo Group Ltd Pyrrolochinoxalinonderivate als antibakterielle mittel
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Also Published As

Publication number Publication date
US20080221110A1 (en) 2008-09-11
SI1954697T1 (sl) 2010-05-31
EP1954697B1 (en) 2010-02-24
HRP20100194T1 (hr) 2010-05-31
HRP20100194T8 (en) 2010-06-30
WO2007081597A3 (en) 2008-06-12
ES2340531T3 (es) 2010-06-04
EP1954697A2 (en) 2008-08-13
CA2626641A1 (en) 2007-07-19
PT1954697E (pt) 2010-05-17
AR057981A1 (es) 2008-01-09
ATE458737T1 (de) 2010-03-15
JP2009512695A (ja) 2009-03-26
EA200801128A1 (ru) 2008-10-30
MA29873B1 (fr) 2008-10-03
NZ567315A (en) 2011-01-28
DE602006012535D1 (de) 2010-04-08
NO20082191L (no) 2008-07-16
KR20080064173A (ko) 2008-07-08
US20080280892A1 (en) 2008-11-13
BRPI0617467A2 (pt) 2011-07-26
CY1110137T1 (el) 2015-01-14
WO2007081597A2 (en) 2007-07-19
PL1954697T3 (pl) 2010-07-30
AU2006335042A1 (en) 2007-07-19
HK1118546A1 (en) 2009-02-13
PE20070793A1 (es) 2007-08-23
DK1954697T3 (da) 2010-06-14
IL190803A0 (en) 2008-12-29
TW200736263A (en) 2007-10-01

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Legal Events

Date Code Title Description
FA Abandonment or withdrawal (granting procedure)