DK2699553T3 - Substituerede diaminocarboxamid- og diaminocarbonitrilpyrimidiner, sammensætninger deraf og fremgangsmåder til behandling dermed - Google Patents

Substituerede diaminocarboxamid- og diaminocarbonitrilpyrimidiner, sammensætninger deraf og fremgangsmåder til behandling dermed Download PDF

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DK2699553T3
DK2699553T3 DK12718524.7T DK12718524T DK2699553T3 DK 2699553 T3 DK2699553 T3 DK 2699553T3 DK 12718524 T DK12718524 T DK 12718524T DK 2699553 T3 DK2699553 T3 DK 2699553T3
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compositions
processes
treatment
diaminocarboxamide
substituted
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DK12718524.7T
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Danish (da)
English (en)
Inventor
Brydon L Bennett
Paul Erdman
Robert Hilgraf
Laurie Ann Lebrun
Meg Mccarrick
Stephen Norris
David A Paisner
Marianne Sloss
William J Romanow
Yoshitaka Satoh
Jayashree Tikhe
Won Hyung Yoon
Jan Elsner
Mehran F Moghaddam
Mark A Nagy
Maria Mercedes Delgado
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Signal Pharm Llc
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    • C07D239/02—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings
    • C07D239/24—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members
    • C07D239/28—Heterocyclic compounds containing 1,3-diazine or hydrogenated 1,3-diazine rings not condensed with other rings having three or more double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to ring carbon atoms
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    • C07D239/48—Two nitrogen atoms
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    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
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DK12718524.7T 2011-04-22 2012-04-20 Substituerede diaminocarboxamid- og diaminocarbonitrilpyrimidiner, sammensætninger deraf og fremgangsmåder til behandling dermed DK2699553T3 (da)

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US201161478076P 2011-04-22 2011-04-22
US201161555339P 2011-11-03 2011-11-03
PCT/US2012/034349 WO2012145569A1 (en) 2011-04-22 2012-04-20 Substituted diaminocarboxamide and diaminocarbonitrile pyrimidines, compositions thereof, and methods of treatment therewith

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DK2699553T3 true DK2699553T3 (da) 2024-01-29

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CN (5) CN105001165B (enExample)
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EC (1) ECSP13012985A (enExample)
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JP2023179797A (ja) 2023-12-19
CA2829264C (en) 2020-04-07
RU2625309C2 (ru) 2017-07-13
UA120740C2 (uk) 2020-02-10
CL2013003025A1 (es) 2014-05-30
CN106946795A (zh) 2017-07-14
RU2017121958A (ru) 2019-01-29
US20230116093A1 (en) 2023-04-13
CN106946795B (zh) 2020-06-02
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IL245792B (en) 2018-03-29
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EP2699553A1 (en) 2014-02-26
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US20180305322A1 (en) 2018-10-25

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