DK169819B1 - Fremgangsmåde til fremstilling af 3-phenylthiazolo(3,2-a)benzimidazolderivater eller et salt deraf - Google Patents

Fremgangsmåde til fremstilling af 3-phenylthiazolo(3,2-a)benzimidazolderivater eller et salt deraf Download PDF

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Publication number
DK169819B1
DK169819B1 DK024088A DK24088A DK169819B1 DK 169819 B1 DK169819 B1 DK 169819B1 DK 024088 A DK024088 A DK 024088A DK 24088 A DK24088 A DK 24088A DK 169819 B1 DK169819 B1 DK 169819B1
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DK
Denmark
Prior art keywords
acid
water
formula
salt
reaction
Prior art date
Application number
DK024088A
Other languages
Danish (da)
English (en)
Other versions
DK24088D0 (da
DK24088A (da
Inventor
Robin Gerald Shepherd
Sie-Yearl Chai
Maynard Emanuel Lichty
Arnold Stephen Milowsky
Original Assignee
Wyeth John & Brother Ltd
American Home Prod
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Wyeth John & Brother Ltd, American Home Prod filed Critical Wyeth John & Brother Ltd
Publication of DK24088D0 publication Critical patent/DK24088D0/da
Publication of DK24088A publication Critical patent/DK24088A/da
Application granted granted Critical
Publication of DK169819B1 publication Critical patent/DK169819B1/da

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    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/02Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains two hetero rings
    • C07D513/04Ortho-condensed systems
    • CCHEMISTRY; METALLURGY
    • C07ORGANIC CHEMISTRY
    • C07DHETEROCYCLIC COMPOUNDS
    • C07D513/00Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14Ortho-condensed systems

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DK024088A 1987-01-21 1988-01-20 Fremgangsmåde til fremstilling af 3-phenylthiazolo(3,2-a)benzimidazolderivater eller et salt deraf DK169819B1 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8701228 1987-01-21
GB878701228A GB8701228D0 (en) 1987-01-21 1987-01-21 Thiazolobenzimidazoles

Publications (3)

Publication Number Publication Date
DK24088D0 DK24088D0 (da) 1988-01-20
DK24088A DK24088A (da) 1988-07-06
DK169819B1 true DK169819B1 (da) 1995-03-06

Family

ID=10610964

Family Applications (1)

Application Number Title Priority Date Filing Date
DK024088A DK169819B1 (da) 1987-01-21 1988-01-20 Fremgangsmåde til fremstilling af 3-phenylthiazolo(3,2-a)benzimidazolderivater eller et salt deraf

Country Status (16)

Country Link
US (2) US4812574A (fr)
EP (1) EP0276133B1 (fr)
JP (1) JP2555397B2 (fr)
KR (1) KR960004536B1 (fr)
AT (1) ATE86257T1 (fr)
AU (1) AU602045B2 (fr)
CA (1) CA1327042C (fr)
DE (1) DE3878700T2 (fr)
DK (1) DK169819B1 (fr)
ES (1) ES2045098T3 (fr)
GB (2) GB8701228D0 (fr)
HU (1) HU201081B (fr)
IE (1) IE61348B1 (fr)
IL (1) IL85135A (fr)
PT (1) PT86567B (fr)
ZA (1) ZA88378B (fr)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
IT1243362B (it) * 1990-07-25 1994-06-10 Pietro Monforte Sintesi di attivita' anti-hiv di 1h, 3h-tiazolo 3,4-a benzimidazoli 1-sostituiti
WO2010077295A1 (fr) * 2008-12-09 2010-07-08 King Faisal Specialist Hospital & Research Centre Hétérocycles tricycliques substitués et leurs utilisations pour traiter des tumeurs et des troubles prolifératifs
CN111116613B (zh) * 2019-12-13 2021-04-23 湘潭大学 一种多取代苯并咪唑并噻唑及衍生物及其合成方法

Family Cites Families (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR1380507A (fr) * 1963-08-28 1964-12-04 Emballages Transparents Soc D Procédé et dispositif pour la fabrication d'emballages se présentant sous forme de sachets multiples accolés ou superposés
US4214089A (en) * 1978-07-18 1980-07-22 American Home Products Corporation Thiazolo[3,2-a]benzimidazoles, imidazo [2,1-b]thiazoles, and related compounds as antineoplastic agents, and enhancers of the immune response
US4361574A (en) * 1981-10-02 1982-11-30 American Home Products Corporation Inhibitors of mammalian collagenase
US4466957A (en) * 1982-02-25 1984-08-21 American Home Products Corporation Vaccine adjuvants

Also Published As

Publication number Publication date
AU602045B2 (en) 1990-09-27
JP2555397B2 (ja) 1996-11-20
GB2200116B (en) 1991-06-12
DE3878700T2 (de) 1993-06-09
US4889936A (en) 1989-12-26
CA1327042C (fr) 1994-02-15
PT86567B (pt) 1991-12-31
KR960004536B1 (ko) 1996-04-06
DK24088D0 (da) 1988-01-20
EP0276133B1 (fr) 1993-03-03
DE3878700D1 (de) 1993-04-08
KR880009031A (ko) 1988-09-13
ZA88378B (en) 1989-09-27
GB2200116A (en) 1988-07-27
US4812574A (en) 1989-03-14
EP0276133A3 (en) 1990-03-21
IL85135A0 (en) 1988-06-30
ATE86257T1 (de) 1993-03-15
IE880143L (en) 1988-07-21
DK24088A (da) 1988-07-06
IE61348B1 (en) 1994-11-02
ES2045098T3 (es) 1994-01-16
PT86567A (en) 1988-02-01
GB8801219D0 (en) 1988-02-17
HU201081B (en) 1990-09-28
AU1037988A (en) 1988-07-28
GB8701228D0 (en) 1987-02-25
JPS63198689A (ja) 1988-08-17
IL85135A (en) 1992-07-15
EP0276133A2 (fr) 1988-07-27
HUT50835A (en) 1990-03-28

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Legal Events

Date Code Title Description
B1 Patent granted (law 1993)
PBP Patent lapsed