DK160612C - Analogifremgangsmaade til fremstilling af ved begge n-atomer cyclopenta-, cyclohexa- og cyclohepta-annelerede pyrazol- og pyridazinderivater - Google Patents
Analogifremgangsmaade til fremstilling af ved begge n-atomer cyclopenta-, cyclohexa- og cyclohepta-annelerede pyrazol- og pyridazinderivaterInfo
- Publication number
- DK160612C DK160612C DK194783A DK194783A DK160612C DK 160612 C DK160612 C DK 160612C DK 194783 A DK194783 A DK 194783A DK 194783 A DK194783 A DK 194783A DK 160612 C DK160612 C DK 160612C
- Authority
- DK
- Denmark
- Prior art keywords
- analyed
- cyclohexa
- cyclohepta
- cyclopenta
- pyrazole
- Prior art date
Links
- WTKZEGDFNFYCGP-UHFFFAOYSA-N Pyrazole Chemical compound C=1C=NNC=1 WTKZEGDFNFYCGP-UHFFFAOYSA-N 0.000 title 1
- PBMFSQRYOILNGV-UHFFFAOYSA-N pyridazine Chemical class C1=CC=NN=C1 PBMFSQRYOILNGV-UHFFFAOYSA-N 0.000 title 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
- C07D209/44—Iso-indoles; Hydrogenated iso-indoles
- C07D209/48—Iso-indoles; Hydrogenated iso-indoles with oxygen atoms in positions 1 and 3, e.g. phthalimide
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D231/00—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings
- C07D231/02—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings
- C07D231/04—Heterocyclic compounds containing 1,2-diazole or hydrogenated 1,2-diazole rings not condensed with other rings having no double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D237/00—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings
- C07D237/02—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings
- C07D237/04—Heterocyclic compounds containing 1,2-diazine or hydrogenated 1,2-diazine rings not condensed with other rings having less than three double bonds between ring members or between ring members and non-ring members
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D403/00—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00
- C07D403/02—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings
- C07D403/06—Heterocyclic compounds containing two or more hetero rings, having nitrogen atoms as the only ring hetero atoms, not provided for by group C07D401/00 containing two hetero rings linked by a carbon chain containing only aliphatic carbon atoms
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
- C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
- C07D487/04—Ortho-condensed systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/3804—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)] not used, see subgroups
- C07F9/3886—Acids containing the structure -C(=X)-P(=X)(XH)2 or NC-P(=X)(XH)2, (X = O, S, Se)
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/28—Phosphorus compounds with one or more P—C bonds
- C07F9/38—Phosphonic acids [RP(=O)(OH)2]; Thiophosphonic acids ; [RP(=X1)(X2H)2(X1, X2 are each independently O, S or Se)]
- C07F9/40—Esters thereof
- C07F9/4071—Esters thereof the ester moiety containing a substituent or a structure which is considered as characteristic
- C07F9/409—Compounds containing the structure P(=X)-X-acyl, P(=X) -X-heteroatom, P(=X)-X-CN (X = O, S, Se)
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/645—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom having two nitrogen atoms as the only ring hetero atoms
- C07F9/6509—Six-membered rings
- C07F9/650905—Six-membered rings having the nitrogen atoms in the positions 1 and 2
- C07F9/650947—Six-membered rings having the nitrogen atoms in the positions 1 and 2 condensed with carbocyclic rings or carbocyclic ring systems
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
- C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
- C07F9/02—Phosphorus compounds
- C07F9/547—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom
- C07F9/6561—Heterocyclic compounds, e.g. containing phosphorus as a ring hetero atom containing systems of two or more relevant hetero rings condensed among themselves or condensed with a common carbocyclic ring or ring system, with or without other non-condensed hetero rings
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07K—PEPTIDES
- C07K5/00—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof
- C07K5/04—Peptides containing up to four amino acids in a fully defined sequence; Derivatives thereof containing only normal peptide links
- C07K5/06—Dipeptides
- C07K5/06139—Dipeptides with the first amino acid being heterocyclic
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Health & Medical Sciences (AREA)
- Life Sciences & Earth Sciences (AREA)
- Biochemistry (AREA)
- General Health & Medical Sciences (AREA)
- Molecular Biology (AREA)
- Crystallography & Structural Chemistry (AREA)
- Biophysics (AREA)
- Genetics & Genomics (AREA)
- Medicinal Chemistry (AREA)
- Proteomics, Peptides & Aminoacids (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
- Nitrogen Condensed Heterocyclic Rings (AREA)
- Indole Compounds (AREA)
Applications Claiming Priority (4)
Application Number | Priority Date | Filing Date | Title |
---|---|---|---|
GB8213850 | 1982-05-12 | ||
GB8213850 | 1982-05-12 | ||
GB08305505A GB2128984B (en) | 1982-05-12 | 1983-02-28 | Diaza-bicyclic compounds |
GB8305505 | 1983-02-28 |
Publications (4)
Publication Number | Publication Date |
---|---|
DK194783D0 DK194783D0 (da) | 1983-05-02 |
DK194783A DK194783A (da) | 1983-11-13 |
DK160612B DK160612B (da) | 1991-04-02 |
DK160612C true DK160612C (da) | 1991-09-23 |
Family
ID=26282820
Family Applications (1)
Application Number | Title | Priority Date | Filing Date |
---|---|---|---|
DK194783A DK160612C (da) | 1982-05-12 | 1983-05-02 | Analogifremgangsmaade til fremstilling af ved begge n-atomer cyclopenta-, cyclohexa- og cyclohepta-annelerede pyrazol- og pyridazinderivater |
Country Status (32)
Country | Link |
---|---|
US (3) | US4512924A (ko) |
EP (1) | EP0094095B1 (ko) |
KR (1) | KR890002106B1 (ko) |
AR (1) | AR240940A1 (ko) |
AU (1) | AU567873B2 (ko) |
BG (1) | BG61123B2 (ko) |
CA (1) | CA1234568A (ko) |
CS (2) | CS249128B2 (ko) |
CU (1) | CU21532A3 (ko) |
DE (2) | DE3317290A1 (ko) |
DK (1) | DK160612C (ko) |
DO (1) | DOP1983004163A (ko) |
DZ (1) | DZ540A1 (ko) |
ES (6) | ES522291A0 (ko) |
FI (1) | FI77244C (ko) |
FR (1) | FR2531956B1 (ko) |
GB (1) | GB2128984B (ko) |
GR (1) | GR77462B (ko) |
HK (1) | HK91692A (ko) |
HU (3) | HU199842B (ko) |
IE (1) | IE56480B1 (ko) |
IL (1) | IL68620A (ko) |
IT (1) | IT1212738B (ko) |
LU (2) | LU84803A1 (ko) |
MC (1) | MC1515A1 (ko) |
MY (1) | MY102889A (ko) |
NL (2) | NL8301640A (ko) |
NO (1) | NO160368C (ko) |
PT (1) | PT76681B (ko) |
SE (1) | SE461792B (ko) |
SG (1) | SG81192G (ko) |
ZW (1) | ZW9883A1 (ko) |
Families Citing this family (102)
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US4902707A (en) * | 1985-04-30 | 1990-02-20 | Eli Lilly And Company | Bicyclic pyrazolidinones, compositions and use |
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IL58849A (en) * | 1978-12-11 | 1983-03-31 | Merck & Co Inc | Carboxyalkyl dipeptides and derivatives thereof,their preparation and pharmaceutical compositions containing them |
IL60617A0 (en) * | 1979-07-23 | 1980-09-16 | Sparamedica Ag | Triazolopyridazine derivative,their preparation and pharmaceutical compositions containing them |
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EP0042100A1 (de) * | 1980-06-13 | 1981-12-23 | F. HOFFMANN-LA ROCHE & CO. Aktiengesellschaft | Pyrazolopyridazin-Derivate, Zwischenprodukte und Verfahren zu deren Herstellung, sowie diese enthaltende Arzneimittel |
DE3169261D1 (en) * | 1980-09-10 | 1985-04-18 | Beecham Group Plc | Aryl diazabicyclyl amides, a process for their preparation and use |
GB2128984B (en) * | 1982-05-12 | 1985-05-22 | Hoffmann La Roche | Diaza-bicyclic compounds |
-
1983
- 1983-02-28 GB GB08305505A patent/GB2128984B/en not_active Expired
- 1983-04-29 CA CA000427095A patent/CA1234568A/en not_active Expired
- 1983-04-29 ZW ZW98/83A patent/ZW9883A1/xx unknown
- 1983-05-02 DK DK194783A patent/DK160612C/da not_active IP Right Cessation
- 1983-05-06 IL IL68620A patent/IL68620A/xx not_active IP Right Cessation
- 1983-05-09 IT IT8321000A patent/IT1212738B/it active
- 1983-05-09 HU HU875409A patent/HU199842B/hu not_active IP Right Cessation
- 1983-05-09 CU CU8335899A patent/CU21532A3/xx unknown
- 1983-05-09 NL NL8301640A patent/NL8301640A/nl not_active Application Discontinuation
- 1983-05-09 AU AU14364/83A patent/AU567873B2/en not_active Expired
- 1983-05-09 HU HU831589A patent/HU195965B/hu unknown
- 1983-05-09 HU HU875410A patent/HU198935B/hu unknown
- 1983-05-10 MC MC821633A patent/MC1515A1/xx unknown
- 1983-05-10 DZ DZ836846A patent/DZ540A1/fr active
- 1983-05-10 FR FR8307785A patent/FR2531956B1/fr not_active Expired
- 1983-05-11 ES ES522291A patent/ES522291A0/es active Granted
- 1983-05-11 EP EP83104668A patent/EP0094095B1/de not_active Expired - Lifetime
- 1983-05-11 CS CS833303A patent/CS249128B2/cs unknown
- 1983-05-11 DE DE19833317290 patent/DE3317290A1/de not_active Ceased
- 1983-05-11 DE DE8383104668T patent/DE3381884D1/de not_active Expired - Lifetime
- 1983-05-11 SE SE8302716A patent/SE461792B/sv not_active IP Right Cessation
- 1983-05-11 NO NO831675A patent/NO160368C/no not_active IP Right Cessation
- 1983-05-11 KR KR1019830002033A patent/KR890002106B1/ko not_active IP Right Cessation
- 1983-05-11 IE IE1084/83A patent/IE56480B1/en not_active IP Right Cessation
- 1983-05-11 AR AR292991A patent/AR240940A1/es active
- 1983-05-11 LU LU84803A patent/LU84803A1/de unknown
- 1983-05-12 PT PT76681A patent/PT76681B/pt unknown
- 1983-05-12 GR GR71331A patent/GR77462B/el unknown
- 1983-05-12 US US06/493,876 patent/US4512924A/en not_active Expired - Lifetime
- 1983-05-12 FI FI831661A patent/FI77244C/fi not_active IP Right Cessation
- 1983-05-12 DO DO1983004163A patent/DOP1983004163A/es unknown
-
1984
- 1984-01-02 ES ES528630A patent/ES8607970A1/es not_active Expired
- 1984-01-02 ES ES528628A patent/ES8706672A1/es not_active Expired
- 1984-01-02 ES ES528625A patent/ES528625A0/es active Granted
- 1984-01-02 ES ES528627A patent/ES8601994A1/es not_active Expired
-
1985
- 1985-02-01 US US06/697,559 patent/US4658024A/en not_active Expired - Lifetime
-
1986
- 1986-05-14 ES ES554935A patent/ES8800170A1/es not_active Expired
- 1986-11-28 US US06/936,003 patent/US4772701A/en not_active Expired - Lifetime
-
1987
- 1987-09-08 MY MYPI87001597A patent/MY102889A/en unknown
-
1991
- 1991-12-23 CS CS914021A patent/CS402191A3/cs unknown
-
1992
- 1992-08-12 SG SG811/92A patent/SG81192G/en unknown
- 1992-11-19 HK HK916/92A patent/HK91692A/xx not_active IP Right Cessation
-
1993
- 1993-06-09 LU LU88299C patent/LU88299I2/fr unknown
- 1993-06-11 NL NL930055C patent/NL930055I2/nl unknown
-
1994
- 1994-02-21 BG BG98502A patent/BG61123B2/bg unknown
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