DK160554C - Substituerede phenylalkyl(piperazinyl eller homopiperazinyl)-alkyl-(urinstoffer eller thiourinstoffer), analogifremgangsmaade til fremstilling heraf og farmaceutisk praeparat indeholdende en saadan forbindelse - Google Patents

Substituerede phenylalkyl(piperazinyl eller homopiperazinyl)-alkyl-(urinstoffer eller thiourinstoffer), analogifremgangsmaade til fremstilling heraf og farmaceutisk praeparat indeholdende en saadan forbindelse

Info

Publication number
DK160554C
DK160554C DK294084A DK294084A DK160554C DK 160554 C DK160554 C DK 160554C DK 294084 A DK294084 A DK 294084A DK 294084 A DK294084 A DK 294084A DK 160554 C DK160554 C DK 160554C
Authority
DK
Denmark
Prior art keywords
preparation
thiour
homopiperazinyl
piperazinyl
urine
Prior art date
Application number
DK294084A
Other languages
Danish (da)
English (en)
Other versions
DK294084D0 (da
DK294084A (da
DK160554B (da
Inventor
John P Devlin
Karl D Hargrave
Edward L Barsumian
Genus J Possanza
Original Assignee
Boehringer Ingelheim Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Boehringer Ingelheim Ltd filed Critical Boehringer Ingelheim Ltd
Publication of DK294084D0 publication Critical patent/DK294084D0/da
Publication of DK294084A publication Critical patent/DK294084A/da
Publication of DK160554B publication Critical patent/DK160554B/da
Application granted granted Critical
Publication of DK160554C publication Critical patent/DK160554C/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D295/00—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms
    • C07D295/04—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms
    • C07D295/12—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms
    • C07D295/125—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings
    • C07D295/13—Heterocyclic compounds containing polymethylene-imine rings with at least five ring members, 3-azabicyclo [3.2.2] nonane, piperazine, morpholine or thiomorpholine rings, having only hydrogen atoms directly attached to the ring carbon atoms with substituted hydrocarbon radicals attached to ring nitrogen atoms substituted by singly or doubly bound nitrogen atoms with the ring nitrogen atoms and the substituent nitrogen atoms attached to the same carbon chain, which is not interrupted by carbocyclic rings to an acyclic saturated chain
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P37/00—Drugs for immunological or allergic disorders
    • A61P37/08—Antiallergic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/08—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 not condensed with other rings

Landscapes

  • Organic Chemistry (AREA)
  • Chemical & Material Sciences (AREA)
  • Health & Medical Sciences (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Veterinary Medicine (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Public Health (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Immunology (AREA)
  • Pulmonology (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Hydrogenated Pyridines (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DK294084A 1983-06-16 1984-06-15 Substituerede phenylalkyl(piperazinyl eller homopiperazinyl)-alkyl-(urinstoffer eller thiourinstoffer), analogifremgangsmaade til fremstilling heraf og farmaceutisk praeparat indeholdende en saadan forbindelse DK160554C (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US50483783A 1983-06-16 1983-06-16
US50483783 1983-06-16

Publications (4)

Publication Number Publication Date
DK294084D0 DK294084D0 (da) 1984-06-15
DK294084A DK294084A (da) 1984-12-17
DK160554B DK160554B (da) 1991-03-25
DK160554C true DK160554C (da) 1991-09-09

Family

ID=24007953

Family Applications (1)

Application Number Title Priority Date Filing Date
DK294084A DK160554C (da) 1983-06-16 1984-06-15 Substituerede phenylalkyl(piperazinyl eller homopiperazinyl)-alkyl-(urinstoffer eller thiourinstoffer), analogifremgangsmaade til fremstilling heraf og farmaceutisk praeparat indeholdende en saadan forbindelse

Country Status (25)

Country Link
EP (1) EP0129207B1 (enExample)
JP (1) JPS6075469A (enExample)
KR (1) KR890000175B1 (enExample)
AR (1) AR242377A1 (enExample)
AT (1) ATE33023T1 (enExample)
AU (1) AU565041B2 (enExample)
CA (1) CA1219260A (enExample)
CS (1) CS244821B2 (enExample)
DD (1) DD223710A5 (enExample)
DE (1) DE3469896D1 (enExample)
DK (1) DK160554C (enExample)
ES (3) ES8506651A1 (enExample)
FI (1) FI76327C (enExample)
GR (1) GR82367B (enExample)
HU (1) HU192409B (enExample)
IE (1) IE59034B1 (enExample)
IL (1) IL72123A (enExample)
NO (1) NO161618C (enExample)
NZ (1) NZ208535A (enExample)
PH (1) PH24059A (enExample)
PL (2) PL146314B1 (enExample)
PT (1) PT78729B (enExample)
SU (2) SU1542415A3 (enExample)
YU (2) YU104584A (enExample)
ZA (1) ZA844527B (enExample)

Families Citing this family (11)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4661481A (en) * 1983-06-16 1987-04-28 Boehringer Ingelheim Pharmaceuticals, Inc Substituted phenylalkylhomopiperazinylpropyl(ureas or thioureas) useful for treatment of immulogical, inflammatory and allergic disorders
FR2601366B1 (fr) * 1986-07-10 1988-11-25 Andre Buzas Derives de la benzhydryloxyethyl-piperazine, procedes d'obtention et de compositions pharmaceutiques les contenant.
JP2722250B2 (ja) * 1989-05-30 1998-03-04 興和株式会社 新規なジアミン化合物及びこれを含有する脳機能障害改善剤
JPH0525145A (ja) * 1991-07-15 1993-02-02 Mochida Pharmaceut Co Ltd アレルギー性疾患治療剤
DE4302485A1 (de) * 1993-01-29 1994-08-04 Merck Patent Gmbh Piperazinderivate
JP3719612B2 (ja) * 1993-06-14 2005-11-24 塩野義製薬株式会社 ヘテロ環を含有する尿素誘導体
ITRM20060090A1 (it) * 2006-02-22 2007-08-23 Sigma Tau Ind Farmaceuti Nuovi composti inibitori cpt a livello del snc come farmaci antidiabetici e o antiobesita
BRPI0815591B8 (pt) 2007-08-22 2021-05-25 Astrazeneca Ab composto, composição farmacêutica, e, uso de um composto.
TW201039825A (en) * 2009-02-20 2010-11-16 Astrazeneca Ab Cyclopropyl amide derivatives 983
AU2011218492B2 (en) 2010-02-18 2014-11-13 Astrazeneca Ab New crystalline form of a cyclopropyl benzamide derivative
EP3484880B1 (en) 2016-07-13 2020-09-02 Leo Pharma A/S Heteroaromatic modulators of the retinoid-related orphan receptor gamma

Also Published As

Publication number Publication date
FI842408A7 (fi) 1984-12-17
ES8600255A1 (es) 1985-09-16
NZ208535A (en) 1987-02-20
NO161618B (no) 1989-05-29
ES537662A0 (es) 1985-09-16
FI76327C (fi) 1988-10-10
DE3469896D1 (en) 1988-04-21
FI76327B (fi) 1988-06-30
FI842408A0 (fi) 1984-06-14
IE841499L (en) 1984-12-16
YU150186A (en) 1987-06-30
DK294084D0 (da) 1984-06-15
EP0129207A3 (en) 1985-07-31
IE59034B1 (en) 1993-12-15
HUT34464A (en) 1985-03-28
ES533448A0 (es) 1985-08-01
EP0129207B1 (en) 1988-03-16
DK294084A (da) 1984-12-17
ES8506651A1 (es) 1985-08-01
SU1387877A3 (ru) 1988-04-07
JPS6075469A (ja) 1985-04-27
NO842417L (no) 1984-12-17
AU2940484A (en) 1984-12-20
ES8601928A1 (es) 1985-11-01
PL248207A1 (en) 1985-08-13
PT78729A (en) 1984-07-01
HU192409B (en) 1987-06-29
JPH0469147B2 (enExample) 1992-11-05
SU1542415A3 (ru) 1990-02-07
PT78729B (en) 1986-10-21
ZA844527B (en) 1986-02-26
CS244821B2 (en) 1986-08-14
PL146314B1 (en) 1989-01-31
DK160554B (da) 1991-03-25
ATE33023T1 (de) 1988-04-15
AU565041B2 (en) 1987-09-03
PH24059A (en) 1990-03-05
AR242377A1 (es) 1993-03-31
PL252851A1 (en) 1986-07-01
CA1219260A (en) 1987-03-17
YU104584A (en) 1986-12-31
PL147413B1 (en) 1989-05-31
IL72123A0 (en) 1984-10-31
NO161618C (no) 1989-09-06
EP0129207A2 (en) 1984-12-27
KR890000175B1 (ko) 1989-03-09
GR82367B (enExample) 1984-12-13
DD223710A5 (de) 1985-06-19
ES537661A0 (es) 1985-11-01
IL72123A (en) 1987-09-16
KR850000422A (ko) 1985-02-27

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