DK1477472T3 - Substituerede phenylalkansyrederivater og anvendelse deraf - Google Patents

Substituerede phenylalkansyrederivater og anvendelse deraf

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Publication number
DK1477472T3
DK1477472T3 DK03706983T DK03706983T DK1477472T3 DK 1477472 T3 DK1477472 T3 DK 1477472T3 DK 03706983 T DK03706983 T DK 03706983T DK 03706983 T DK03706983 T DK 03706983T DK 1477472 T3 DK1477472 T3 DK 1477472T3
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group
carbon atoms
alkyl group
acid derivatives
integer
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DK03706983T
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Danish (da)
English (en)
Inventor
Motoshi Shoda
Hiroshi Kuriyama
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Asahi Kasei Pharma Corp
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Publication of DK1477472T3 publication Critical patent/DK1477472T3/da

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    • C07C59/68—Unsaturated compounds containing ether groups, groups, groups, or groups containing six-membered aromatic rings the non-carboxylic part of the ether containing six-membered aromatic rings the oxygen atom of the ether group being bound to a non-condensed six-membered aromatic ring
    • C—CHEMISTRY; METALLURGY
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    • C07C59/00—Compounds having carboxyl groups bound to acyclic carbon atoms and containing any of the groups OH, O—metal, —CHO, keto, ether, groups, groups, or groups
    • C07C59/40—Unsaturated compounds
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    • C07C69/00—Esters of carboxylic acids; Esters of carbonic or haloformic acids
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    • C07C69/73—Esters of carboxylic acids having esterified carboxylic groups bound to acyclic carbon atoms and having any of the groups OH, O—metal, —CHO, keto, ether, acyloxy, groups, groups, or in the acid moiety of unsaturated acids
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    • C07D209/04—Indoles; Hydrogenated indoles
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    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/10—Indoles; Hydrogenated indoles with substituted hydrocarbon radicals attached to carbon atoms of the hetero ring
    • C07D209/18—Radicals substituted by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals
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    • C07C2601/08—Systems containing only non-condensed rings with a five-membered ring the ring being saturated

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DK03706983T 2002-02-21 2003-02-20 Substituerede phenylalkansyrederivater og anvendelse deraf DK1477472T3 (da)

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DK1477472T3 (da) * 2002-02-21 2009-04-06 Asahi Kasei Pharma Corp Substituerede phenylalkansyrederivater og anvendelse deraf
AU2003277576A1 (en) 2002-11-08 2004-06-07 Takeda Pharmaceutical Company Limited Receptor function controlling agent
JP4594611B2 (ja) * 2002-11-08 2010-12-08 武田薬品工業株式会社 受容体機能調節剤
PL377712A1 (pl) * 2003-02-13 2006-02-06 Wellstat Therapeutics Corporation Związki do leczenia zaburzeń metabolicznych
CA2535665A1 (en) * 2003-08-14 2005-02-24 Asahi Kasei Pharma Corporation Substituted arylalkanoic acid derivative and use thereof
WO2005051373A1 (ja) * 2003-11-26 2005-06-09 Takeda Pharmaceutical Company Limited 受容体機能調節剤
US20070185152A1 (en) * 2004-03-02 2007-08-09 Smithkline Beecham Corporation Inhibitors of akt activity
GB0409921D0 (en) * 2004-05-04 2004-06-09 Novartis Ag Organic compounds
TW200716588A (en) * 2005-06-02 2007-05-01 Kyowa Hakko Kogyo Kk A process for preparing dibenzoxepin derivative
US7405302B2 (en) * 2005-10-11 2008-07-29 Amira Pharmaceuticals, Inc. 5-lipoxygenase-activating protein (FLAP) inhibitors
KR101440255B1 (ko) 2006-07-20 2014-09-17 아사히 가세이 파마 가부시키가이샤 치환 페닐알칸산의 신규 결정 및 제조 방법
CL2008000973A1 (es) * 2007-04-05 2009-01-02 Astrazeneca Ab Compuestos derivados de 1-oxo-isoquinolina; procedimiento de preparación; composición farmacéutica; y su uso en el tratamiento de enfermedades pulmonares obstructvas crónicas (epoc) y asma.
EP2154131A4 (en) * 2007-04-26 2011-09-21 Pharmafrontier Co Ltd INHIBITOR OF THE G-PROTEIN-COUPLED RECEPTOR AND PHARMACEUTICAL PRODUCT
US7928140B2 (en) * 2007-08-02 2011-04-19 Amgen Inc. Benzothiazole PI3 kinase modulators for cancer treatment
CN101932317B (zh) 2008-01-18 2013-03-27 旭化成制药株式会社 稳定的药物组合物
CN104710365A (zh) 2008-04-28 2015-06-17 旭化成制药株式会社 苯丙酸衍生物及其用途
PT2292592E (pt) 2008-06-05 2012-11-12 Asahi Kasei Pharma Corp Composto de sulfonamida e sua aplicação
CN102391264A (zh) * 2011-09-21 2012-03-28 河北九派制药有限公司 6-溴咪唑并[1,2-a]吡啶的制备方法
JP5802518B2 (ja) 2011-10-31 2015-10-28 公益財団法人微生物化学研究会 新規化合物、その製造方法、及びその用途
US8889730B2 (en) 2012-04-10 2014-11-18 Pfizer Inc. Indole and indazole compounds that activate AMPK
EP2970177A1 (en) 2013-03-15 2016-01-20 Pfizer Inc. Indole compounds that activate ampk
CN105315167A (zh) * 2014-08-01 2016-02-10 华东师范大学 一种2,2,3-三芳基-3-芳基氨基丙酸甲酯衍生物及其合成方法和应用
MX2017007874A (es) 2014-12-24 2018-01-24 Lg Chemical Ltd Derivado de biarilo como agonista de gpr120.
JP6635999B2 (ja) * 2017-10-13 2020-01-29 株式会社ダイセル カリウム塩の製造方法、及びカリウム塩
CN110092774B (zh) * 2018-01-29 2022-04-08 中国科学院上海药物研究所 芳香丙酸类衍生物、及其制备方法和用途
WO2022174253A1 (en) * 2021-02-12 2022-08-18 Nimbus Saturn, Inc. Hpk1 antagonists and uses thereof
JP2024509192A (ja) 2021-03-05 2024-02-29 ニンバス サターン， インコーポレイテッド Ｈｐｋ１アンタゴニスト及びその使用

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JP3802581B2 (ja) * 1995-03-01 2006-07-26 富山化学工業株式会社 新規なビフェニル誘導体またはその塩およびそれらを含有する抗炎症剤
WO1999019291A1 (fr) * 1997-10-14 1999-04-22 Asahi Kasei Kogyo Kabushiki Kaisha Derives de biphenyl-5-acide alcanoique et leurs applications
DK1477472T3 (da) * 2002-02-21 2009-04-06 Asahi Kasei Pharma Corp Substituerede phenylalkansyrederivater og anvendelse deraf

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HK1076445A1 (en) 2006-01-20
AU2003211384A1 (en) 2003-09-09
JP5048017B2 (ja) 2012-10-17
ES2319753T3 (es) 2009-05-12
AU2003211384B2 (en) 2008-12-11
JP4390563B2 (ja) 2009-12-24
CA2477208C (en) 2010-11-30
KR100938950B1 (ko) 2010-01-26
EP1477472A1 (en) 2004-11-17
WO2003070686A1 (fr) 2003-08-28
DE60325830D1 (de) 2009-03-05
JP2009167217A (ja) 2009-07-30
CN1653032A (zh) 2005-08-10
PT1477472E (pt) 2009-03-17
KR20040094712A (ko) 2004-11-10
EP1477472A4 (en) 2005-12-14
CA2477208A1 (en) 2003-08-28
JP2009167216A (ja) 2009-07-30
CN100387576C (zh) 2008-05-14
JPWO2003070686A1 (ja) 2005-06-09
ATE420847T1 (de) 2009-01-15
JP5000683B2 (ja) 2012-08-15
MXPA04008176A (es) 2004-11-26
EP1477472B1 (en) 2009-01-14

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