DK0982032T3 - Anvendelse af en sulfamatesterholdig sterolforbindelse til fremstilling af et lægemiddel til kontrol af østrogenproduktion - Google Patents

Anvendelse af en sulfamatesterholdig sterolforbindelse til fremstilling af et lægemiddel til kontrol af østrogenproduktion

Info

Publication number
DK0982032T3
DK0982032T3 DK99203449T DK99203449T DK0982032T3 DK 0982032 T3 DK0982032 T3 DK 0982032T3 DK 99203449 T DK99203449 T DK 99203449T DK 99203449 T DK99203449 T DK 99203449T DK 0982032 T3 DK0982032 T3 DK 0982032T3
Authority
DK
Denmark
Prior art keywords
sub
compound
drug
manufacture
ester containing
Prior art date
Application number
DK99203449T
Other languages
Danish (da)
English (en)
Inventor
Michael John Reed
Barry Victor Lloyd Potter
Original Assignee
Sterix Ltd
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Sterix Ltd filed Critical Sterix Ltd
Application granted granted Critical
Publication of DK0982032T3 publication Critical patent/DK0982032T3/da

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/56—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids
    • A61K31/565—Compounds containing cyclopenta[a]hydrophenanthrene ring systems; Derivatives thereof, e.g. steroids not substituted in position 17 beta by a carbon atom, e.g. estrane, estradiol
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P43/00—Drugs for specific purposes, not provided for in groups A61P1/00-A61P41/00
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/30—Oestrogens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/32—Antioestrogens
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P5/00—Drugs for disorders of the endocrine system
    • A61P5/24—Drugs for disorders of the endocrine system of the sex hormones
    • A61P5/36—Antigestagens
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07J—STEROIDS
    • C07J41/00—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring
    • C07J41/0033—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005
    • C07J41/0072—Normal steroids containing one or more nitrogen atoms not belonging to a hetero ring not covered by C07J41/0005 the A ring of the steroid being aromatic

Landscapes

  • Health & Medical Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Medicinal Chemistry (AREA)
  • Animal Behavior & Ethology (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Engineering & Computer Science (AREA)
  • Bioinformatics & Cheminformatics (AREA)
  • Diabetes (AREA)
  • Endocrinology (AREA)
  • Epidemiology (AREA)
  • Steroid Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
  • Enzymes And Modification Thereof (AREA)
  • Nitrogen Condensed Heterocyclic Rings (AREA)
  • Medicinal Preparation (AREA)
  • Surgical Instruments (AREA)
  • Mechanical Treatment Of Semiconductor (AREA)
  • Medicines That Contain Protein Lipid Enzymes And Other Medicines (AREA)
  • Nitrogen And Oxygen Or Sulfur-Condensed Heterocyclic Ring Systems (AREA)
  • Preparation Of Compounds By Using Micro-Organisms (AREA)
DK99203449T 1991-08-29 1992-08-28 Anvendelse af en sulfamatesterholdig sterolforbindelse til fremstilling af et lægemiddel til kontrol af østrogenproduktion DK0982032T3 (da)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB919118478A GB9118478D0 (en) 1991-08-29 1991-08-29 Steroid sulphatase inhibitors
PCT/GB1992/001587 WO1993005064A1 (en) 1991-08-29 1992-08-28 Steroid sulphatase inhibitors

Publications (1)

Publication Number Publication Date
DK0982032T3 true DK0982032T3 (da) 2003-11-03

Family

ID=10700604

Family Applications (4)

Application Number Title Priority Date Filing Date
DK92918285T DK0641355T3 (da) 1991-08-29 1992-08-28 Anvendelse af sulfamatderivater som steroid-sulfatase-inhibitorer
DK99203449T DK0982032T3 (da) 1991-08-29 1992-08-28 Anvendelse af en sulfamatesterholdig sterolforbindelse til fremstilling af et lægemiddel til kontrol af østrogenproduktion
DK98204340T DK0921130T3 (da) 1991-08-29 1992-08-28 Steroid-sulfatase-inhibitorer
DK98204337T DK0928609T3 (da) 1991-08-29 1992-08-28 Farmaceutiske præparater indeholdende sulfamatderivater som steroidsulfatase-inhibitorer

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DK92918285T DK0641355T3 (da) 1991-08-29 1992-08-28 Anvendelse af sulfamatderivater som steroid-sulfatase-inhibitorer

Family Applications After (2)

Application Number Title Priority Date Filing Date
DK98204340T DK0921130T3 (da) 1991-08-29 1992-08-28 Steroid-sulfatase-inhibitorer
DK98204337T DK0928609T3 (da) 1991-08-29 1992-08-28 Farmaceutiske præparater indeholdende sulfamatderivater som steroidsulfatase-inhibitorer

Country Status (25)

Country Link
US (3) US5616574A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
EP (6) EP0921130B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
JP (6) JP3219408B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
KR (4) KR100258396B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AT (5) ATE246706T1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
AU (2) AU689043B2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
BR (1) BR9206434A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CA (4) CA2305758A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CY (4) CY2253B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
CZ (1) CZ295939B6 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DE (5) DE69233149T2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
DK (4) DK0641355T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
ES (4) ES2148178T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
FI (5) FI940903A7 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GB (1) GB9118478D0 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GE (6) GEP20063773B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
GR (1) GR3034579T3 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
HU (1) HUT66097A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
LV (1) LV12618B (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
NO (6) NO307301B1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
RU (4) RU2001125673A (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SG (7) SG88783A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
SK (4) SK282187B6 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
UA (4) UA41875C2 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)
WO (1) WO1993005064A1 (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html)

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Also Published As

Publication number Publication date
AU689043B2 (en) 1998-03-19
RU94019334A (ru) 1996-10-20
UA70958C2 (uk) 2004-11-15
HU9400583D0 (en) 1994-05-30
DE69233053D1 (de) 2003-06-12
AU668882B2 (en) 1996-05-23
UA70956C2 (uk) 2004-11-15
SK24694A3 (en) 1994-11-09
JP2000355598A (ja) 2000-12-26
DE69231280D1 (de) 2000-08-24
ATE239753T1 (de) 2003-05-15
ES2204059T3 (es) 2004-04-16
FI940903A7 (fi) 1994-04-20
HK1020672A1 (en) 2000-05-19
JPH07501515A (ja) 1995-02-16
AU2490592A (en) 1993-04-05
GEP20022803B (en) 2002-09-25
CA2114630A1 (en) 1993-03-18
NO308903B1 (no) 2000-11-13
NO995075D0 (no) 1999-10-18
AU5837396A (en) 1996-09-05
JP2000038341A (ja) 2000-02-08
EP0982032A3 (en) 2002-03-20
FI20002259A7 (fi) 2000-10-13
FI20002261A7 (fi) 2000-10-13
DE69233431D1 (de) 2004-11-11
DK0641355T3 (da) 2000-10-09
ATE194843T1 (de) 2000-08-15
CA2114630C (en) 2003-09-30
GEP20022637B (en) 2002-02-25
EP1099706B1 (en) 2004-10-06
KR100321019B1 (ko) 2002-03-20
HK1019753A1 (en) 2000-02-25
DE69233020D1 (de) 2003-05-22
DE69233431T2 (de) 2006-02-23
DE69233149D1 (de) 2003-09-11
EP0928609B1 (en) 2003-04-16
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SG88782A1 (en) 2002-05-21
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US5830886A (en) 1998-11-03
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JP2000355542A (ja) 2000-12-26
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JP3581802B2 (ja) 2004-10-27
NO940635L (GUID-C5D7CC26-194C-43D0-91A1-9AE8C70A9BFF.html) 1994-04-29
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ATE246706T1 (de) 2003-08-15
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AU1007799A (en) 1999-03-04
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CA2305767A1 (en) 1993-03-18
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JP2003176297A (ja) 2003-06-24
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