DE60313872T2 - Pyrazoloä1,5-aüpyrimidine als hemmstoffe cyclin-abhängiger kinasen - Google Patents

Pyrazoloä1,5-aüpyrimidine als hemmstoffe cyclin-abhängiger kinasen Download PDF

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Publication number
DE60313872T2
DE60313872T2 DE60313872T DE60313872T DE60313872T2 DE 60313872 T2 DE60313872 T2 DE 60313872T2 DE 60313872 T DE60313872 T DE 60313872T DE 60313872 T DE60313872 T DE 60313872T DE 60313872 T2 DE60313872 T2 DE 60313872T2
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alkyl
group
cycloalkyl
aryl
compound according
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DE60313872D1 (de
Inventor
Timothy J. Chatham GUZI
Kamil Garwood PARUCH
Michael P. Scotch Plains DWYER
Ronald J. Convent Station DOLL
Viyyoor Moopil Parsippany GIRIJAVALLABHAN
Carmen S. Livingston ALVAREZ
Tin-Yau Edison CHAN
Chad Garwood KNUTSON
Vincent Mountain Lakes MADISON
Thierry O. Scotch Plains FISCHMANN
Lawrence W. Yardley DILLARD
Vinh D. Fountain Valley TRAN
Zhen Min Princeton HE
Ray Anthony Bensalem JAMES
Haengsoon Plainsboro PARK
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Merck Sharp and Dohme LLC
Pharmacopeia LLC
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Pharmacopeia Drug Discovery Inc
Schering Corp
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    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D487/00—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00
    • C07D487/02—Heterocyclic compounds containing nitrogen atoms as the only ring hetero atoms in the condensed system, not provided for by groups C07D451/00 - C07D477/00 in which the condensed system contains two hetero rings
    • C07D487/04—Ortho-condensed systems
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    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/495—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having six-membered rings with two or more nitrogen atoms as the only ring heteroatoms, e.g. piperazine or tetrazines
    • A61K31/505—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim
    • A61K31/519—Pyrimidines; Hydrogenated pyrimidines, e.g. trimethoprim ortho- or peri-condensed with heterocyclic rings
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  • Hematology (AREA)
  • Communicable Diseases (AREA)
  • Heart & Thoracic Surgery (AREA)
  • Orthopedic Medicine & Surgery (AREA)
  • Pain & Pain Management (AREA)
  • Rheumatology (AREA)
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  • Urology & Nephrology (AREA)
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DE60313872T 2002-09-04 2003-09-03 Pyrazoloä1,5-aüpyrimidine als hemmstoffe cyclin-abhängiger kinasen Expired - Lifetime DE60313872T2 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
US40802902P 2002-09-04 2002-09-04
US408029P 2002-09-04
PCT/US2003/027491 WO2004026229A2 (en) 2002-09-04 2003-09-03 Pyrazolo[1,5-a]pyrimidines compounds as cyclin dependent kinase inhibitors

Publications (2)

Publication Number Publication Date
DE60313872D1 DE60313872D1 (de) 2007-06-28
DE60313872T2 true DE60313872T2 (de) 2008-01-17

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DE60313872T Expired - Lifetime DE60313872T2 (de) 2002-09-04 2003-09-03 Pyrazoloä1,5-aüpyrimidine als hemmstoffe cyclin-abhängiger kinasen

Country Status (18)

Country Link
US (2) US7067661B2 (https=)
EP (1) EP1534712B1 (https=)
JP (2) JP4790265B2 (https=)
KR (1) KR20050033659A (https=)
CN (1) CN1701073B (https=)
AR (1) AR041133A1 (https=)
AT (1) ATE362474T1 (https=)
AU (1) AU2003298571B2 (https=)
CA (1) CA2497544C (https=)
DE (1) DE60313872T2 (https=)
ES (1) ES2283868T3 (https=)
MX (1) MXPA05002572A (https=)
MY (2) MY145332A (https=)
NZ (1) NZ539161A (https=)
PE (1) PE20041000A1 (https=)
TW (1) TWI329645B (https=)
WO (1) WO2004026229A2 (https=)
ZA (1) ZA200501846B (https=)

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