DE3233898A1 - 3'-deaminoanaloge von glykosidanthracyclin-antibiotika, verfahren zu deren herstellung und zusammensetzungen, welche diese enthalten - Google Patents

3'-deaminoanaloge von glykosidanthracyclin-antibiotika, verfahren zu deren herstellung und zusammensetzungen, welche diese enthalten

Info

Publication number
DE3233898A1
DE3233898A1 DE19823233898 DE3233898A DE3233898A1 DE 3233898 A1 DE3233898 A1 DE 3233898A1 DE 19823233898 DE19823233898 DE 19823233898 DE 3233898 A DE3233898 A DE 3233898A DE 3233898 A1 DE3233898 A1 DE 3233898A1
Authority
DE
Germany
Prior art keywords
deep
deamino
doxorubicin
daunorubicin
iii
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Granted
Application number
DE19823233898
Other languages
German (de)
English (en)
Other versions
DE3233898C2 (enExample
Inventor
Federico 20014 Nerviano Milano Arcamone
Anna Maria 20133 Milano Casazza
Giuseppe 27058 Voghera Milano Cassinelli
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL filed Critical Farmitalia Carlo Erba SRL
Publication of DE3233898A1 publication Critical patent/DE3233898A1/de
Application granted granted Critical
Publication of DE3233898C2 publication Critical patent/DE3233898C2/de
Granted legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
DE19823233898 1981-09-18 1982-09-13 3'-deaminoanaloge von glykosidanthracyclin-antibiotika, verfahren zu deren herstellung und zusammensetzungen, welche diese enthalten Granted DE3233898A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
GB8128252 1981-09-18

Publications (2)

Publication Number Publication Date
DE3233898A1 true DE3233898A1 (de) 1983-04-07
DE3233898C2 DE3233898C2 (enExample) 1988-01-28

Family

ID=10524593

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19823233898 Granted DE3233898A1 (de) 1981-09-18 1982-09-13 3'-deaminoanaloge von glykosidanthracyclin-antibiotika, verfahren zu deren herstellung und zusammensetzungen, welche diese enthalten

Country Status (24)

Country Link
JP (1) JPS5862184A (enExample)
KR (1) KR880001573B1 (enExample)
AU (1) AU549656B2 (enExample)
BE (1) BE894418A (enExample)
CA (1) CA1184903A (enExample)
CH (1) CH654014A5 (enExample)
CS (1) CS236682B2 (enExample)
DE (1) DE3233898A1 (enExample)
DK (1) DK157030C (enExample)
ES (1) ES8400120A1 (enExample)
FI (1) FI823169L (enExample)
FR (1) FR2513255A1 (enExample)
GR (1) GR77639B (enExample)
HU (1) HU186971B (enExample)
IE (1) IE53330B1 (enExample)
IL (1) IL66775A (enExample)
IT (1) IT1210481B (enExample)
NL (1) NL8203548A (enExample)
NO (1) NO153335C (enExample)
NZ (1) NZ201899A (enExample)
PT (1) PT75575B (enExample)
SE (1) SE456587B (enExample)
YU (1) YU204982A (enExample)
ZA (1) ZA826806B (enExample)

Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4112076A (en) * 1975-04-30 1978-09-05 Societa' Farmaceutici Italia S.P.A. Epi-daunomycin and epi-adriamycin compounds and method of use

Patent Citations (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4112076A (en) * 1975-04-30 1978-09-05 Societa' Farmaceutici Italia S.P.A. Epi-daunomycin and epi-adriamycin compounds and method of use

Non-Patent Citations (1)

* Cited by examiner, † Cited by third party
Title
US-Buch: H.S.El Khadem,Academic Press, Anthracycline Antibiotics (Symposium 24. - 25.8.1981) New York, 1982, S. 1 - 57, S. 59 - 73, S.197 - 224 *

Also Published As

Publication number Publication date
DE3233898C2 (enExample) 1988-01-28
DK157030C (da) 1990-04-02
CA1184903A (en) 1985-04-02
SE456587B (sv) 1988-10-17
HU186971B (en) 1985-10-28
IT1210481B (it) 1989-09-14
NZ201899A (en) 1985-09-13
SE8205288L (sv) 1983-03-19
ES515690A0 (es) 1983-10-16
CS236682B2 (en) 1985-05-15
PT75575B (en) 1984-12-10
FI823169A7 (fi) 1983-03-19
IE822246L (en) 1983-03-18
ZA826806B (en) 1983-07-27
JPS6260396B2 (enExample) 1987-12-16
AU8832382A (en) 1983-03-24
KR840001592A (ko) 1984-05-07
GR77639B (enExample) 1984-09-25
FR2513255A1 (fr) 1983-03-25
NL8203548A (nl) 1983-04-18
AU549656B2 (en) 1986-02-06
NO153335C (no) 1986-02-26
ES8400120A1 (es) 1983-10-16
SE8205288D0 (sv) 1982-09-15
KR880001573B1 (ko) 1988-08-23
NO823148L (no) 1983-03-21
YU204982A (en) 1985-03-20
FR2513255B1 (enExample) 1984-11-30
PT75575A (en) 1982-10-01
FI823169L (fi) 1983-03-19
NO153335B (no) 1985-11-18
IT8223240A0 (it) 1982-09-14
IL66775A (en) 1986-11-30
DK411382A (da) 1983-03-19
FI823169A0 (fi) 1982-09-14
BE894418A (fr) 1983-01-17
JPS5862184A (ja) 1983-04-13
IL66775A0 (en) 1982-12-31
DK157030B (da) 1989-10-30
IE53330B1 (en) 1988-10-12
CH654014A5 (it) 1986-01-31

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Legal Events

Date Code Title Description
8101 Request for examination as to novelty
8105 Search report available
8110 Request for examination paragraph 44
D2 Grant after examination
8364 No opposition during term of opposition
8327 Change in the person/name/address of the patent owner

Owner name: FARMITALIA CARLO ERBA S.R.L., MAILAND/MILANO, IT

8328 Change in the person/name/address of the agent

Free format text: EITLE, W., DIPL.-ING. HOFFMANN, K., DIPL.-ING. DR.RER.NAT. LEHN, W., DIPL.-ING. FUECHSLE, K., DIPL.-ING. HANSEN, B., DIPL.-CHEM. DR.RER.NAT. BRAUNS, H., DIPL.-CHEM. DR.RER.NAT. GOERG, K., DIPL.-ING. KOHLMANN, K., DIPL.-ING. KOLB, H., DIPL.-CHEM. DR.RER.NAT. RITTER UND EDLER VON FISCHERN, B., DIPL.-ING., PAT.-ANWAELTE, 8000 MUENCHEN

8339 Ceased/non-payment of the annual fee