CA1184903A - Process for preparing 3'-deamino analogs of glycoside anthracycline antibiotics - Google Patents

Process for preparing 3'-deamino analogs of glycoside anthracycline antibiotics

Info

Publication number
CA1184903A
CA1184903A CA000411403A CA411403A CA1184903A CA 1184903 A CA1184903 A CA 1184903A CA 000411403 A CA000411403 A CA 000411403A CA 411403 A CA411403 A CA 411403A CA 1184903 A CA1184903 A CA 1184903A
Authority
CA
Canada
Prior art keywords
deamino
doxorubicin
daunorubicin
diepi
preparing
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
CA000411403A
Other languages
English (en)
French (fr)
Inventor
Giuseppe Cassinelli
Federico Arcamone
Anna M. Casazza
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Pfizer Italia SRL
Original Assignee
Farmitalia Carlo Erba SRL
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Farmitalia Carlo Erba SRL filed Critical Farmitalia Carlo Erba SRL
Application granted granted Critical
Publication of CA1184903A publication Critical patent/CA1184903A/en
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07H—SUGARS; DERIVATIVES THEREOF; NUCLEOSIDES; NUCLEOTIDES; NUCLEIC ACIDS
    • C07H15/00—Compounds containing hydrocarbon or substituted hydrocarbon radicals directly attached to hetero atoms of saccharide radicals
    • C07H15/20—Carbocyclic rings
    • C07H15/24—Condensed ring systems having three or more rings
    • C07H15/252—Naphthacene radicals, e.g. daunomycins, adriamycins
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P35/00—Antineoplastic agents

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biotechnology (AREA)
  • Engineering & Computer Science (AREA)
  • Molecular Biology (AREA)
  • Genetics & Genomics (AREA)
  • Biochemistry (AREA)
  • Veterinary Medicine (AREA)
  • Public Health (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • General Chemical & Material Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
CA000411403A 1981-09-18 1982-09-14 Process for preparing 3'-deamino analogs of glycoside anthracycline antibiotics Expired CA1184903A (en)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
GB8128252 1981-09-18
GB8128252 1981-09-18

Publications (1)

Publication Number Publication Date
CA1184903A true CA1184903A (en) 1985-04-02

Family

ID=10524593

Family Applications (1)

Application Number Title Priority Date Filing Date
CA000411403A Expired CA1184903A (en) 1981-09-18 1982-09-14 Process for preparing 3'-deamino analogs of glycoside anthracycline antibiotics

Country Status (24)

Country Link
JP (1) JPS5862184A (enExample)
KR (1) KR880001573B1 (enExample)
AU (1) AU549656B2 (enExample)
BE (1) BE894418A (enExample)
CA (1) CA1184903A (enExample)
CH (1) CH654014A5 (enExample)
CS (1) CS236682B2 (enExample)
DE (1) DE3233898A1 (enExample)
DK (1) DK157030C (enExample)
ES (1) ES515690A0 (enExample)
FI (1) FI823169L (enExample)
FR (1) FR2513255A1 (enExample)
GR (1) GR77639B (enExample)
HU (1) HU186971B (enExample)
IE (1) IE53330B1 (enExample)
IL (1) IL66775A (enExample)
IT (1) IT1210481B (enExample)
NL (1) NL8203548A (enExample)
NO (1) NO153335C (enExample)
NZ (1) NZ201899A (enExample)
PT (1) PT75575B (enExample)
SE (1) SE456587B (enExample)
YU (1) YU204982A (enExample)
ZA (1) ZA826806B (enExample)

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1506200A (en) * 1975-04-30 1978-04-05 Farmaceutici Italia Glycosides

Also Published As

Publication number Publication date
PT75575A (en) 1982-10-01
IL66775A (en) 1986-11-30
ZA826806B (en) 1983-07-27
IL66775A0 (en) 1982-12-31
NO153335C (no) 1986-02-26
JPS5862184A (ja) 1983-04-13
FI823169A7 (fi) 1983-03-19
IE822246L (en) 1983-03-18
CH654014A5 (it) 1986-01-31
KR880001573B1 (ko) 1988-08-23
DE3233898C2 (enExample) 1988-01-28
NL8203548A (nl) 1983-04-18
IT8223240A0 (it) 1982-09-14
FI823169L (fi) 1983-03-19
IE53330B1 (en) 1988-10-12
NO823148L (no) 1983-03-21
IT1210481B (it) 1989-09-14
AU549656B2 (en) 1986-02-06
FR2513255A1 (fr) 1983-03-25
DE3233898A1 (de) 1983-04-07
FR2513255B1 (enExample) 1984-11-30
GR77639B (enExample) 1984-09-25
DK157030C (da) 1990-04-02
ES8400120A1 (es) 1983-10-16
HU186971B (en) 1985-10-28
FI823169A0 (fi) 1982-09-14
DK157030B (da) 1989-10-30
DK411382A (da) 1983-03-19
JPS6260396B2 (enExample) 1987-12-16
PT75575B (en) 1984-12-10
YU204982A (en) 1985-03-20
AU8832382A (en) 1983-03-24
KR840001592A (ko) 1984-05-07
SE456587B (sv) 1988-10-17
NZ201899A (en) 1985-09-13
NO153335B (no) 1985-11-18
SE8205288L (sv) 1983-03-19
SE8205288D0 (sv) 1982-09-15
ES515690A0 (es) 1983-10-16
BE894418A (fr) 1983-01-17
CS236682B2 (en) 1985-05-15

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Legal Events

Date Code Title Description
MKEC Expiry (correction)
MKEX Expiry