DE2954236C2 - - Google Patents

Info

Publication number
DE2954236C2
DE2954236C2 DE2954236A DE2954236A DE2954236C2 DE 2954236 C2 DE2954236 C2 DE 2954236C2 DE 2954236 A DE2954236 A DE 2954236A DE 2954236 A DE2954236 A DE 2954236A DE 2954236 C2 DE2954236 C2 DE 2954236C2
Authority
DE
Germany
Prior art keywords
phenyl
pyrrolidin
cis
amino
trifluoromethylphenyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Expired
Application number
DE2954236A
Other languages
German (de)
English (en)
Inventor
Peter Liestal Ch Hofer
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Mundipharma AG
Original Assignee
Mundipharma AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Mundipharma AG filed Critical Mundipharma AG
Application granted granted Critical
Publication of DE2954236C2 publication Critical patent/DE2954236C2/de
Expired legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
    • C07D207/263—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms
    • C07D207/267—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms
    • C07D207/26—2-Pyrrolidones
    • C07D207/263—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms
    • C07D207/27—2-Pyrrolidones with only hydrogen atoms or radicals containing only hydrogen and carbon atoms directly attached to other ring carbon atoms with substituted hydrocarbon radicals directly attached to the ring nitrogen atom
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/30—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members
    • C07D207/34—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having two double bonds between ring members or between ring members and non-ring members with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/36—Oxygen or sulfur atoms
    • C07D207/38—2-Pyrrolones
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07F—ACYCLIC, CARBOCYCLIC OR HETEROCYCLIC COMPOUNDS CONTAINING ELEMENTS OTHER THAN CARBON, HYDROGEN, HALOGEN, OXYGEN, NITROGEN, SULFUR, SELENIUM OR TELLURIUM
    • C07F9/00—Compounds containing elements of Groups 5 or 15 of the Periodic Table
    • C07F9/02—Phosphorus compounds
    • C07F9/28—Phosphorus compounds with one or more P—C bonds
    • C07F9/54—Quaternary phosphonium compounds
    • C07F9/5407—Acyclic saturated phosphonium compounds

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Biochemistry (AREA)
  • General Health & Medical Sciences (AREA)
  • Molecular Biology (AREA)
  • Pyrrole Compounds (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Saccharide Compounds (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
DE2954236A 1978-06-12 1979-06-09 Expired DE2954236C2 (en, 2012)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US91468278A 1978-06-12 1978-06-12
US1249679A 1979-02-15 1979-02-15

Publications (1)

Publication Number Publication Date
DE2954236C2 true DE2954236C2 (en, 2012) 1988-10-06

Family

ID=26683628

Family Applications (3)

Application Number Title Priority Date Filing Date
DE2954237A Expired DE2954237C2 (en, 2012) 1978-06-12 1979-06-09
DE19792923553 Granted DE2923553A1 (de) 1978-06-12 1979-06-09 Verfahren zur herstellung von delta hoch 3 -pyrrolin-(2)-derivaten sowie verwendung von delta hoch 3 -pyrrolin-(2)- derivaten zur herstellung von pyrrolidon- (2)-derivaten
DE2954236A Expired DE2954236C2 (en, 2012) 1978-06-12 1979-06-09

Family Applications Before (2)

Application Number Title Priority Date Filing Date
DE2954237A Expired DE2954237C2 (en, 2012) 1978-06-12 1979-06-09
DE19792923553 Granted DE2923553A1 (de) 1978-06-12 1979-06-09 Verfahren zur herstellung von delta hoch 3 -pyrrolin-(2)-derivaten sowie verwendung von delta hoch 3 -pyrrolin-(2)- derivaten zur herstellung von pyrrolidon- (2)-derivaten

Country Status (19)

Country Link
AR (1) AR222997A1 (en, 2012)
AT (1) ATA386679A (en, 2012)
AU (1) AU529479B2 (en, 2012)
CA (1) CA1108628A (en, 2012)
CH (1) CH650772A5 (en, 2012)
DE (3) DE2954237C2 (en, 2012)
DK (1) DK157847C (en, 2012)
ES (1) ES481315A1 (en, 2012)
FI (1) FI70209C (en, 2012)
FR (1) FR2434151A1 (en, 2012)
GB (1) GB2028307B (en, 2012)
GR (1) GR68438B (en, 2012)
IL (1) IL57266A (en, 2012)
IT (1) IT1116891B (en, 2012)
NL (1) NL7904584A (en, 2012)
NO (1) NO791943L (en, 2012)
NZ (1) NZ190705A (en, 2012)
PT (1) PT69716A (en, 2012)
SE (1) SE431644B (en, 2012)

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US4943640A (en) * 1983-10-14 1990-07-24 The Dow Chemical Company Preparation of 5-(1-alkyl-carbonyloxy)alkylpyrrolidin-2-one
AU4809390A (en) * 1988-12-27 1990-08-01 Ici Americas Inc. Process for the preparation of 3-carboalkoxypyrrolidones
US5021587A (en) * 1990-01-24 1991-06-04 Petrolite Corporation Synthesis of N,3,4-trisubstituted-3-azoline-2-ones

Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1350582A (en) * 1970-07-24 1974-04-18 Ucb Sa Cerivatives of 2-pyrrolidinone
US4012495A (en) * 1974-03-20 1977-03-15 Schering Aktiengesellschaft 4-(Polyalkoxyphenyl)-2-pyrrolidones

Family Cites Families (1)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3272842A (en) * 1965-06-25 1966-09-13 Lilly Co Eli Novel pyrrolinones

Patent Citations (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
GB1350582A (en) * 1970-07-24 1974-04-18 Ucb Sa Cerivatives of 2-pyrrolidinone
US4012495A (en) * 1974-03-20 1977-03-15 Schering Aktiengesellschaft 4-(Polyalkoxyphenyl)-2-pyrrolidones

Non-Patent Citations (4)

* Cited by examiner, † Cited by third party
Title
Chemical Abstracts, Bd.75, 1971, 98437 u *
J. Am. Chem. Soc. 1959, 81, S.6029-6041 *
J. org. Chem. 1966, 31, S.48-52 *
J. org.Chem. 1967, 32, S.1346-1353 *

Also Published As

Publication number Publication date
FI791866A7 (fi) 1979-12-13
AU529479B2 (en) 1983-06-09
GB2028307A (en) 1980-03-05
FR2434151B3 (en, 2012) 1982-04-30
IL57266A0 (en) 1979-09-30
DE2923553C2 (en, 2012) 1988-06-01
ATA386679A (de) 1983-12-15
FI70209B (fi) 1986-02-28
IT1116891B (it) 1986-02-10
DK241779A (da) 1979-12-13
DK157847C (da) 1990-09-17
PT69716A (en) 1979-07-01
DK157847B (da) 1990-02-26
SE431644B (sv) 1984-02-20
NZ190705A (en) 1981-10-19
FI70209C (fi) 1986-09-15
CH650772A5 (de) 1985-08-15
DE2954237C2 (en, 2012) 1989-09-21
NL7904584A (nl) 1979-12-14
CA1108628A (en) 1981-09-08
SE7905079L (sv) 1979-12-13
GB2028307B (en) 1983-01-19
AU4767079A (en) 1979-12-20
NO791943L (no) 1979-12-13
AR222997A1 (es) 1981-07-15
FR2434151A1 (fr) 1980-03-21
IT7949373A0 (it) 1979-06-11
DE2923553A1 (de) 1979-12-20
GR68438B (en, 2012) 1981-12-30
IL57266A (en) 1982-12-31
ES481315A1 (es) 1980-08-16

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