DE2623077A1 - Verfahren zur herstellung von n-(1- ethyl-2-pyrrolidinylmethyl)-2-methoxy-5- sulfamoylbenzamid - Google Patents
Verfahren zur herstellung von n-(1- ethyl-2-pyrrolidinylmethyl)-2-methoxy-5- sulfamoylbenzamidInfo
- Publication number
- DE2623077A1 DE2623077A1 DE19762623077 DE2623077A DE2623077A1 DE 2623077 A1 DE2623077 A1 DE 2623077A1 DE 19762623077 DE19762623077 DE 19762623077 DE 2623077 A DE2623077 A DE 2623077A DE 2623077 A1 DE2623077 A1 DE 2623077A1
- Authority
- DE
- Germany
- Prior art keywords
- methoxy
- ethyl
- pyrrolidinylmethyl
- sulfamoylbenzamide
- preparation
- Prior art date
- Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
- Withdrawn
Links
- 238000000034 method Methods 0.000 title claims description 6
- 238000002360 preparation method Methods 0.000 title claims description 3
- BGRJTUBHPOOWDU-UHFFFAOYSA-N sulpiride Chemical compound CCN1CCCC1CNC(=O)C1=CC(S(N)(=O)=O)=CC=C1OC BGRJTUBHPOOWDU-UHFFFAOYSA-N 0.000 title 1
- KXDAEFPNCMNJSK-UHFFFAOYSA-N Benzamide Chemical compound NC(=O)C1=CC=CC=C1 KXDAEFPNCMNJSK-UHFFFAOYSA-N 0.000 claims description 6
- 125000002496 methyl group Chemical group [H]C([H])([H])* 0.000 claims description 2
- 150000007522 mineralic acids Chemical class 0.000 claims description 2
- 150000007524 organic acids Chemical class 0.000 claims description 2
- 235000005985 organic acids Nutrition 0.000 claims description 2
- 150000003242 quaternary ammonium salts Chemical class 0.000 claims description 2
- 150000003839 salts Chemical class 0.000 claims description 2
- 125000003142 tertiary amide group Chemical group 0.000 claims description 2
- 150000003863 ammonium salts Chemical class 0.000 claims 1
- XTHFKEDIFFGKHM-UHFFFAOYSA-N Dimethoxyethane Chemical compound COCCOC XTHFKEDIFFGKHM-UHFFFAOYSA-N 0.000 description 5
- VSCWAEJMTAWNJL-UHFFFAOYSA-K aluminium trichloride Chemical compound Cl[Al](Cl)Cl VSCWAEJMTAWNJL-UHFFFAOYSA-K 0.000 description 4
- XEKOWRVHYACXOJ-UHFFFAOYSA-N Ethyl acetate Chemical compound CCOC(C)=O XEKOWRVHYACXOJ-UHFFFAOYSA-N 0.000 description 3
- 239000000203 mixture Substances 0.000 description 3
- 239000002904 solvent Substances 0.000 description 3
- -1 1-ethyl-2-pyrrolidinylmethyl Chemical group 0.000 description 2
- QGZKDVFQNNGYKY-UHFFFAOYSA-N Ammonia Chemical compound N QGZKDVFQNNGYKY-UHFFFAOYSA-N 0.000 description 2
- LFQSCWFLJHTTHZ-UHFFFAOYSA-N Ethanol Chemical compound CCO LFQSCWFLJHTTHZ-UHFFFAOYSA-N 0.000 description 2
- VEXZGXHMUGYJMC-UHFFFAOYSA-N Hydrochloric acid Chemical compound Cl VEXZGXHMUGYJMC-UHFFFAOYSA-N 0.000 description 2
- XLYOFNOQVPJJNP-UHFFFAOYSA-N water Substances O XLYOFNOQVPJJNP-UHFFFAOYSA-N 0.000 description 2
- 125000001931 aliphatic group Chemical group 0.000 description 1
- 229910052783 alkali metal Inorganic materials 0.000 description 1
- 150000001340 alkali metals Chemical class 0.000 description 1
- 150000001408 amides Chemical class 0.000 description 1
- 229910021529 ammonia Inorganic materials 0.000 description 1
- 125000003118 aryl group Chemical group 0.000 description 1
- 238000009835 boiling Methods 0.000 description 1
- 239000003054 catalyst Substances 0.000 description 1
- 239000003610 charcoal Substances 0.000 description 1
- 239000003153 chemical reaction reagent Substances 0.000 description 1
- 238000001816 cooling Methods 0.000 description 1
- 238000001704 evaporation Methods 0.000 description 1
- 230000008020 evaporation Effects 0.000 description 1
- UPWPDUACHOATKO-UHFFFAOYSA-K gallium trichloride Chemical compound Cl[Ga](Cl)Cl UPWPDUACHOATKO-UHFFFAOYSA-K 0.000 description 1
- 150000004820 halides Chemical class 0.000 description 1
- 238000004519 manufacturing process Methods 0.000 description 1
- 229910052751 metal Inorganic materials 0.000 description 1
- 239000002184 metal Substances 0.000 description 1
- 230000000144 pharmacologic effect Effects 0.000 description 1
- 150000003334 secondary amides Chemical group 0.000 description 1
- NVIFVTYDZMXWGX-UHFFFAOYSA-N sodium metaborate Chemical compound [Na+].[O-]B=O NVIFVTYDZMXWGX-UHFFFAOYSA-N 0.000 description 1
- 239000000725 suspension Substances 0.000 description 1
Classifications
-
- C—CHEMISTRY; METALLURGY
- C07—ORGANIC CHEMISTRY
- C07D—HETEROCYCLIC COMPOUNDS
- C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
- C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
- C07D207/04—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members
- C07D207/08—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having no double bonds between ring members or between ring members and non-ring members with hydrocarbon radicals, substituted by hetero atoms, attached to ring carbon atoms
- C07D207/09—Radicals substituted by nitrogen atoms, not forming part of a nitro radical
Landscapes
- Chemical & Material Sciences (AREA)
- Organic Chemistry (AREA)
- Pyrrole Compounds (AREA)
- Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
- Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
Applications Claiming Priority (1)
| Application Number | Priority Date | Filing Date | Title |
|---|---|---|---|
| FR7518180A FR2314178A1 (fr) | 1975-06-11 | 1975-06-11 | Nouveau procede de preparation du n-(1-ethyl-2-pyrrolidylmethyl) 2-methoxy 5-methoxy 5-sulfamoyl benzamide |
Publications (1)
| Publication Number | Publication Date |
|---|---|
| DE2623077A1 true DE2623077A1 (de) | 1976-12-30 |
Family
ID=9156330
Family Applications (1)
| Application Number | Title | Priority Date | Filing Date |
|---|---|---|---|
| DE19762623077 Withdrawn DE2623077A1 (de) | 1975-06-11 | 1976-05-22 | Verfahren zur herstellung von n-(1- ethyl-2-pyrrolidinylmethyl)-2-methoxy-5- sulfamoylbenzamid |
Country Status (10)
| Country | Link |
|---|---|
| JP (1) | JPS5231068A (enExample) |
| AT (1) | AT349458B (enExample) |
| CA (1) | CA1064944A (enExample) |
| DE (1) | DE2623077A1 (enExample) |
| FI (1) | FI761680A7 (enExample) |
| FR (1) | FR2314178A1 (enExample) |
| GB (1) | GB1497005A (enExample) |
| IE (1) | IE43001B1 (enExample) |
| MX (1) | MX3519E (enExample) |
| PT (1) | PT65165B (enExample) |
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0692470A1 (de) * | 1994-07-15 | 1996-01-17 | Degussa Aktiengesellschaft | Verfahren zur Herstellung optisch aktiver 1-substituierter 2-(Aminomethyl)pyrrolidinderivaten |
Families Citing this family (3)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| IT1141095B (it) * | 1980-11-27 | 1986-10-01 | Ravizza Spa | Processo di risoluzione della sulpiride racema |
| EP0091528B1 (fr) * | 1982-04-08 | 1986-07-23 | Societe D'etudes Scientifiques Et Industrielles De L'ile-De-France | Nouvel agent utilisable pour le traitement de certaines formes de la dépression constitué par le N-(1-propyl-2-pyrrolidylméthyl)-2-méthoxy 5-sulfamoyl benzamide |
| JP7406897B2 (ja) * | 2018-12-07 | 2023-12-28 | キヤノン株式会社 | 搬送装置および物品の製造方法 |
-
1975
- 1975-06-11 FR FR7518180A patent/FR2314178A1/fr active Granted
-
1976
- 1976-05-22 DE DE19762623077 patent/DE2623077A1/de not_active Withdrawn
- 1976-06-01 IE IE1167/76A patent/IE43001B1/en unknown
- 1976-06-01 AT AT400076A patent/AT349458B/de not_active IP Right Cessation
- 1976-06-01 PT PT65165A patent/PT65165B/pt unknown
- 1976-06-08 JP JP51067551A patent/JPS5231068A/ja active Pending
- 1976-06-08 GB GB23696/76A patent/GB1497005A/en not_active Expired
- 1976-06-09 CA CA254,479A patent/CA1064944A/en not_active Expired
- 1976-06-09 MX MX76292U patent/MX3519E/es unknown
- 1976-06-11 FI FI761680A patent/FI761680A7/fi not_active Application Discontinuation
Cited By (1)
| Publication number | Priority date | Publication date | Assignee | Title |
|---|---|---|---|---|
| EP0692470A1 (de) * | 1994-07-15 | 1996-01-17 | Degussa Aktiengesellschaft | Verfahren zur Herstellung optisch aktiver 1-substituierter 2-(Aminomethyl)pyrrolidinderivaten |
Also Published As
| Publication number | Publication date |
|---|---|
| IE43001L (en) | 1976-12-11 |
| GB1497005A (en) | 1978-01-05 |
| FR2314178B1 (enExample) | 1979-04-27 |
| JPS5231068A (en) | 1977-03-09 |
| FI761680A7 (enExample) | 1976-12-12 |
| PT65165B (fr) | 1977-11-17 |
| ATA400076A (de) | 1978-09-15 |
| MX3519E (es) | 1981-01-20 |
| FR2314178A1 (fr) | 1977-01-07 |
| CA1064944A (en) | 1979-10-23 |
| AT349458B (de) | 1979-04-10 |
| PT65165A (fr) | 1976-07-01 |
| IE43001B1 (en) | 1980-12-03 |
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Legal Events
| Date | Code | Title | Description |
|---|---|---|---|
| 8139 | Disposal/non-payment of the annual fee |