DE2559211A1 - Substituierte indole - Google Patents

Substituierte indole

Info

Publication number
DE2559211A1
DE2559211A1 DE19752559211 DE2559211A DE2559211A1 DE 2559211 A1 DE2559211 A1 DE 2559211A1 DE 19752559211 DE19752559211 DE 19752559211 DE 2559211 A DE2559211 A DE 2559211A DE 2559211 A1 DE2559211 A1 DE 2559211A1
Authority
DE
Germany
Prior art keywords
general formula
salts
acids
indole
methyl
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Ceased
Application number
DE19752559211
Other languages
German (de)
English (en)
Inventor
David Mccomsey
Michael Zelesko
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
Janssen Pharmaceuticals Inc
Original Assignee
McNeilab Inc
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by McNeilab Inc filed Critical McNeilab Inc
Publication of DE2559211A1 publication Critical patent/DE2559211A1/de
Ceased legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D209/00—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D209/02—Heterocyclic compounds containing five-membered rings, condensed with other rings, with one nitrogen atom as the only ring hetero atom condensed with one carbocyclic ring
    • C07D209/04—Indoles; Hydrogenated indoles
    • C07D209/30—Indoles; Hydrogenated indoles with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, directly attached to carbon atoms of the hetero ring
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D207/00—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom
    • C07D207/02—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom
    • C07D207/18—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member
    • C07D207/22—Heterocyclic compounds containing five-membered rings not condensed with other rings, with one nitrogen atom as the only ring hetero atom with only hydrogen or carbon atoms directly attached to the ring nitrogen atom having one double bond between ring members or between a ring member and a non-ring member with hetero atoms or with carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, directly attached to ring carbon atoms
    • C07D207/24—Oxygen or sulfur atoms

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Indole Compounds (AREA)
  • Plural Heterocyclic Compounds (AREA)
DE19752559211 1974-12-30 1975-12-30 Substituierte indole Ceased DE2559211A1 (de)

Applications Claiming Priority (2)

Application Number Priority Date Filing Date Title
US53761274A 1974-12-30 1974-12-30
US63179875A 1975-11-13 1975-11-13

Publications (1)

Publication Number Publication Date
DE2559211A1 true DE2559211A1 (de) 1976-07-08

Family

ID=27065555

Family Applications (1)

Application Number Title Priority Date Filing Date
DE19752559211 Ceased DE2559211A1 (de) 1974-12-30 1975-12-30 Substituierte indole

Country Status (27)

Country Link
JP (1) JPS51131872A (xx)
AR (1) AR219052A1 (xx)
AT (1) AT356648B (xx)
AU (1) AU505215B2 (xx)
CA (1) CA1065874A (xx)
CH (1) CH622516A5 (xx)
DD (1) DD125781A5 (xx)
DE (1) DE2559211A1 (xx)
DK (1) DK580175A (xx)
ES (1) ES443935A1 (xx)
FI (1) FI64590C (xx)
FR (2) FR2296413A1 (xx)
GB (1) GB1527510A (xx)
HU (2) HU174948B (xx)
IE (1) IE42390B1 (xx)
IL (1) IL48756A (xx)
IN (1) IN142735B (xx)
IT (1) IT1052654B (xx)
NL (1) NL7515100A (xx)
NO (1) NO145383C (xx)
NZ (1) NZ179580A (xx)
PH (1) PH12328A (xx)
PL (1) PL99353B1 (xx)
RO (1) RO69196A (xx)
SE (1) SE422210B (xx)
SU (1) SU667132A3 (xx)
YU (1) YU332275A (xx)

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5356325A (en) * 1976-10-12 1978-05-22 Wellcome Found Composition having antiicoagulation effect
WO2004041782A1 (en) * 2002-11-07 2004-05-21 Akzo Nobel N.V. Indoles useful in the treatment of androgen-receptor related diseases
US7795280B2 (en) 2002-11-07 2010-09-14 N.V. Organon Indoles useful in the treatment of androgen-receptor related diseases
US7812036B2 (en) 2004-04-23 2010-10-12 N.V. Organon Androgens

Families Citing this family (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2540109B1 (fr) * 1983-01-28 1985-08-30 Logeais Labor Jacques Imino-2 pyrrolidines, leur procede de preparation et leurs applications en therapeutique
US4558048A (en) * 1984-04-06 1985-12-10 Pfizer Inc. Method of treating diarrhoea using indole compounds
EP1216988A4 (en) * 1999-09-28 2005-04-20 Nihon Nohyaku Co Ltd THIOALKYLAMINE DERIVATIVES AND METHOD FOR THE PRODUCTION THEREOF
WO2007020653A1 (en) * 2005-08-12 2007-02-22 Suven Life Sciences Limited Thioether derivatives as functional 5-ht6 ligands

Cited By (4)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
JPS5356325A (en) * 1976-10-12 1978-05-22 Wellcome Found Composition having antiicoagulation effect
WO2004041782A1 (en) * 2002-11-07 2004-05-21 Akzo Nobel N.V. Indoles useful in the treatment of androgen-receptor related diseases
US7795280B2 (en) 2002-11-07 2010-09-14 N.V. Organon Indoles useful in the treatment of androgen-receptor related diseases
US7812036B2 (en) 2004-04-23 2010-10-12 N.V. Organon Androgens

Also Published As

Publication number Publication date
IT1052654B (it) 1981-07-20
HU174948B (hu) 1980-04-28
DK580175A (da) 1976-07-01
IE42390B1 (en) 1980-07-30
FR2315921B1 (xx) 1979-09-28
FR2315921A1 (fr) 1977-01-28
YU332275A (en) 1983-02-28
IL48756A (en) 1979-03-12
JPS51131872A (en) 1976-11-16
IL48756A0 (en) 1976-02-29
FI753669A (xx) 1976-07-01
DD125781A5 (xx) 1977-05-18
AU8791675A (en) 1977-07-07
CA1065874A (en) 1979-11-06
AR219052A1 (es) 1980-07-31
GB1527510A (en) 1978-10-04
AU505215B2 (en) 1979-11-15
NZ179580A (en) 1978-04-03
SE7514458L (sv) 1976-07-01
IE42390L (en) 1976-06-30
ATA986075A (de) 1979-10-15
FR2296413A1 (fr) 1976-07-30
NO145383B (no) 1981-11-30
FI64590B (fi) 1983-08-31
HU174949B (hu) 1980-04-28
PL99353B1 (pl) 1978-07-31
NL7515100A (nl) 1976-07-02
SU667132A3 (ru) 1979-06-05
PH12328A (en) 1979-01-16
FI64590C (fi) 1983-12-12
NO754313L (xx) 1976-07-01
CH622516A5 (en) 1981-04-15
AT356648B (de) 1980-05-12
FR2296413B1 (xx) 1980-06-27
NO145383C (no) 1982-03-10
ES443935A1 (es) 1977-08-16
SE422210B (sv) 1982-02-22
RO69196A (ro) 1980-08-15
IN142735B (xx) 1977-08-20

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Legal Events

Date Code Title Description
8110 Request for examination paragraph 44
8131 Rejection