DE2240442A1 - Verfahren zur herstellung von aminopenicillinen - Google Patents

Verfahren zur herstellung von aminopenicillinen

Info

Publication number
DE2240442A1
DE2240442A1 DE2240442A DE2240442A DE2240442A1 DE 2240442 A1 DE2240442 A1 DE 2240442A1 DE 2240442 A DE2240442 A DE 2240442A DE 2240442 A DE2240442 A DE 2240442A DE 2240442 A1 DE2240442 A1 DE 2240442A1
Authority
DE
Germany
Prior art keywords
condensation
water
aminopenicillins
substituted
crystallization
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE2240442A
Other languages
German (de)
English (en)
Inventor
Artur Pereira Da Luz
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
CIPAN COMP IND PROD
Original Assignee
CIPAN COMP IND PROD
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by CIPAN COMP IND PROD filed Critical CIPAN COMP IND PROD
Publication of DE2240442A1 publication Critical patent/DE2240442A1/de
Pending legal-status Critical Current

Links

Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D499/00—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring
    • C07D499/21—Heterocyclic compounds containing 4-thia-1-azabicyclo [3.2.0] heptane ring systems, i.e. compounds containing a ring system of the formula:, e.g. penicillins, penems; Such ring systems being further condensed, e.g. 2,3-condensed with an oxygen-, nitrogen- or sulfur-containing hetero ring with a nitrogen atom directly attached in position 6 and a carbon atom having three bonds to hetero atoms with at the most one bond to halogen, e.g. an ester or nitrile radical, directly attached in position 2
    • C07D499/44—Compounds with an amino radical acylated by carboxylic acids, attached in position 6
    • C07D499/48—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical
    • C07D499/58—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical
    • C07D499/64—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms
    • C07D499/68—Compounds with an amino radical acylated by carboxylic acids, attached in position 6 with a carbon chain, substituted by hetero atoms or by carbon atoms having three bonds to hetero atoms with at the most one bond to halogen, e.g. ester or nitrile radicals, attached to the carboxamido radical substituted in alpha-position to the carboxamido radical by nitrogen atoms with aromatic rings as additional substituents on the carbon chain

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE2240442A 1971-12-17 1972-08-17 Verfahren zur herstellung von aminopenicillinen Pending DE2240442A1 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
PT5696671 1971-12-17

Publications (1)

Publication Number Publication Date
DE2240442A1 true DE2240442A1 (de) 1973-07-26

Family

ID=20081760

Family Applications (1)

Application Number Title Priority Date Filing Date
DE2240442A Pending DE2240442A1 (de) 1971-12-17 1972-08-17 Verfahren zur herstellung von aminopenicillinen

Country Status (13)

Country Link
JP (1) JPS5318515B2 (xx)
AT (1) AT327377B (xx)
BE (1) BE790466A (xx)
CA (1) CA1003407A (xx)
CH (1) CH561725A5 (xx)
DE (1) DE2240442A1 (xx)
DK (1) DK140669B (xx)
FI (1) FI60209C (xx)
FR (1) FR2165409A5 (xx)
GB (1) GB1400236A (xx)
NL (1) NL7215359A (xx)
SE (1) SE414768B (xx)
ZA (1) ZA725231B (xx)

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2527235A1 (de) * 1974-06-19 1976-01-08 Bristol Myers Co Verfahren zur herstellung von phenylglycinderivaten
DE2718741A1 (de) 1976-04-27 1977-11-17 Bristol Myers Co Cephalosporinverbindungen und verfahren zu deren herstellung
DE2732528A1 (de) * 1976-07-20 1978-01-26 Bristol Myers Co Verfahren zur herstellung von amoxicillintrihydrat

Families Citing this family (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
FR2364217A1 (fr) * 1976-09-08 1978-04-07 Biocraft Laboratories Inc Procede pour la preparation de derives de l'acide 6-aminopenicillanique
NL162387C (nl) * 1977-09-06 1980-05-16 Gist Brocades Nv Werkwijze voor het bereiden van 6-(d-alpha-amino-p- -hydroxyfenylacetamido)penicillanzuur.
DE2817228A1 (de) * 1978-04-20 1979-10-31 Bayer Ag Verfahren zur herstellung halbsynthetischer beta-lactamantibiotika

Cited By (3)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
DE2527235A1 (de) * 1974-06-19 1976-01-08 Bristol Myers Co Verfahren zur herstellung von phenylglycinderivaten
DE2718741A1 (de) 1976-04-27 1977-11-17 Bristol Myers Co Cephalosporinverbindungen und verfahren zu deren herstellung
DE2732528A1 (de) * 1976-07-20 1978-01-26 Bristol Myers Co Verfahren zur herstellung von amoxicillintrihydrat

Also Published As

Publication number Publication date
AU4697172A (en) 1974-03-28
FI60209B (fi) 1981-08-31
FI60209C (fi) 1981-12-10
DK140669C (xx) 1980-03-24
ATA647772A (de) 1975-04-15
DK140669B (da) 1979-10-22
ZA725231B (en) 1973-05-30
SE414768B (sv) 1980-08-18
CH561725A5 (xx) 1975-05-15
FR2165409A5 (xx) 1973-08-03
JPS4867297A (xx) 1973-09-13
AT327377B (de) 1976-01-26
CA1003407A (en) 1977-01-11
JPS5318515B2 (xx) 1978-06-15
GB1400236A (en) 1975-07-16
NL7215359A (xx) 1973-06-19
BE790466A (fr) 1973-02-15

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Legal Events

Date Code Title Description
OHA Expiration of time for request for examination