DE1545965A1 - Verfahren zur Herstellung von Benzodiazepin-Derivaten - Google Patents

Verfahren zur Herstellung von Benzodiazepin-Derivaten

Info

Publication number
DE1545965A1
DE1545965A1 DE19651545965 DE1545965A DE1545965A1 DE 1545965 A1 DE1545965 A1 DE 1545965A1 DE 19651545965 DE19651545965 DE 19651545965 DE 1545965 A DE1545965 A DE 1545965A DE 1545965 A1 DE1545965 A1 DE 1545965A1
Authority
DE
Germany
Prior art keywords
general formula
cor
compound
amino
formula
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19651545965
Other languages
German (de)
English (en)
Inventor
Archer Giles Allan
Sternbach Leo Henryk
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
F Hoffmann La Roche AG
Original Assignee
F Hoffmann La Roche AG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by F Hoffmann La Roche AG filed Critical F Hoffmann La Roche AG
Publication of DE1545965A1 publication Critical patent/DE1545965A1/de
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/33—Heterocyclic compounds
    • A61K31/395—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins
    • A61K31/55—Heterocyclic compounds having nitrogen as a ring hetero atom, e.g. guanethidine or rifamycins having seven-membered rings, e.g. azelastine, pentylenetetrazole
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D243/00—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms
    • C07D243/06—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4
    • C07D243/10—Heterocyclic compounds containing seven-membered rings having two nitrogen atoms as the only ring hetero atoms having the nitrogen atoms in positions 1 and 4 condensed with carbocyclic rings or ring systems
    • C07D243/14—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines
    • C07D243/16—1,4-Benzodiazepines; Hydrogenated 1,4-benzodiazepines substituted in position 5 by aryl radicals

Landscapes

  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
DE19651545965 1964-10-01 1965-09-28 Verfahren zur Herstellung von Benzodiazepin-Derivaten Pending DE1545965A1 (de)

Applications Claiming Priority (4)

Application Number Priority Date Filing Date Title
US400891A US3317518A (en) 1964-10-01 1964-10-01 Novel 5-aryl-1, 2, 4, 5-tetrahydrobenzo-diazepin-3-one compounds
US60414266A 1966-12-23 1966-12-23
US60414166A 1966-12-23 1966-12-23
US60414866A 1966-12-23 1966-12-23

Publications (1)

Publication Number Publication Date
DE1545965A1 true DE1545965A1 (de) 1969-12-11

Family

ID=27503456

Family Applications (4)

Application Number Title Priority Date Filing Date
DE19651543654 Pending DE1543654A1 (de) 1964-10-01 1965-09-28 Verfahren zur Herstellung von Aminen
DE19651545965 Pending DE1545965A1 (de) 1964-10-01 1965-09-28 Verfahren zur Herstellung von Benzodiazepin-Derivaten
DE19651695143 Pending DE1695143A1 (de) 1964-10-01 1965-10-06 Verfahren zur Herstellung von Benzodiazepin-Derivaten
DE19651543655 Pending DE1543655A1 (de) 1964-10-01 1965-10-06 Verfahren zur Herstellung von 2-Acylamino-phenyl-arylketonen

Family Applications Before (1)

Application Number Title Priority Date Filing Date
DE19651543654 Pending DE1543654A1 (de) 1964-10-01 1965-09-28 Verfahren zur Herstellung von Aminen

Family Applications After (2)

Application Number Title Priority Date Filing Date
DE19651695143 Pending DE1695143A1 (de) 1964-10-01 1965-10-06 Verfahren zur Herstellung von Benzodiazepin-Derivaten
DE19651543655 Pending DE1543655A1 (de) 1964-10-01 1965-10-06 Verfahren zur Herstellung von 2-Acylamino-phenyl-arylketonen

Country Status (11)

Country Link
US (4) US3317518A (cg-RX-API-DMAC10.html)
BE (1) BE670394A (cg-RX-API-DMAC10.html)
BR (1) BR6573560D0 (cg-RX-API-DMAC10.html)
CH (1) CH484162A (cg-RX-API-DMAC10.html)
DE (4) DE1543654A1 (cg-RX-API-DMAC10.html)
FR (1) FR5206M (cg-RX-API-DMAC10.html)
GB (4) GB1081635A (cg-RX-API-DMAC10.html)
IL (1) IL24380A (cg-RX-API-DMAC10.html)
NL (1) NL6512775A (cg-RX-API-DMAC10.html)
NO (1) NO121040B (cg-RX-API-DMAC10.html)
SE (1) SE330177B (cg-RX-API-DMAC10.html)

Families Citing this family (2)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3997591A (en) * 1975-03-11 1976-12-14 Hoffmann-La Roche Inc. Tricyclic benzodiazepines
GB9507661D0 (en) * 1995-04-13 1995-05-31 Ass Octel Process

Family Cites Families (7)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3121074A (en) * 1964-02-11 Nitro substituted jh-l
US3182054A (en) * 1965-05-04 Benzodiazepine - compounds
US3121075A (en) * 1961-10-20 1964-02-11 Hoffmann La Roche Aminobenzodiazepines
US3186996A (en) * 1961-10-30 1965-06-01 Nihon Surfactant Ind Co Ltd Pyridoxine 3, 4-diacylates and their preparation
US3182067A (en) * 1964-04-09 1965-05-04 Hoffmann La Roche Benzodiazepine compounds
US3182065A (en) * 1964-04-09 1965-05-04 Hoffmann La Roche 2-acetamidobenzoyl-pyridines
US3182066A (en) * 1964-04-09 1965-05-04 Hoffmann La Roche Aminophenyl-pyridyl ketones

Also Published As

Publication number Publication date
SE330177B (cg-RX-API-DMAC10.html) 1970-11-09
FR5206M (cg-RX-API-DMAC10.html) 1967-07-03
CH484162A (de) 1970-01-15
US3504015A (en) 1970-03-31
GB1081637A (en) 1967-08-31
DE1543655A1 (de) 1969-10-02
DE1543654A1 (de) 1970-03-19
BR6573560D0 (pt) 1973-08-02
US3317518A (en) 1967-05-02
US3504013A (en) 1970-03-31
GB1081635A (en) 1967-08-31
GB1081636A (en) 1967-08-31
US3504014A (en) 1970-03-31
GB1081634A (en) 1967-08-31
BE670394A (cg-RX-API-DMAC10.html) 1966-04-01
DE1695143A1 (de) 1970-02-12
NO121040B (cg-RX-API-DMAC10.html) 1971-01-11
IL24380A (en) 1969-05-28
NL6512775A (cg-RX-API-DMAC10.html) 1966-04-04

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