DE1543372A1 - Verfahren zur Herstellung von o-substituierten 3,4-Dioxyphenylalkanolaminen - Google Patents

Verfahren zur Herstellung von o-substituierten 3,4-Dioxyphenylalkanolaminen

Info

Publication number
DE1543372A1
DE1543372A1 DE19661543372 DE1543372A DE1543372A1 DE 1543372 A1 DE1543372 A1 DE 1543372A1 DE 19661543372 DE19661543372 DE 19661543372 DE 1543372 A DE1543372 A DE 1543372A DE 1543372 A1 DE1543372 A1 DE 1543372A1
Authority
DE
Germany
Prior art keywords
carbon atoms
general formula
group
acid
compounds
Prior art date
Legal status (The legal status is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the status listed.)
Pending
Application number
DE19661543372
Other languages
German (de)
English (en)
Inventor
Anton Dr Mentrup
Kurt Dr Schromm
Otto Dr Thomae
Karl Prof Zeile
Current Assignee (The listed assignees may be inaccurate. Google has not performed a legal analysis and makes no representation or warranty as to the accuracy of the list.)
CH Boehringer Sohn AG and Co KG
Original Assignee
CH Boehringer Sohn AG and Co KG
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by CH Boehringer Sohn AG and Co KG filed Critical CH Boehringer Sohn AG and Co KG
Publication of DE1543372A1 publication Critical patent/DE1543372A1/de
Pending legal-status Critical Current

Links

Classifications

    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61K—PREPARATIONS FOR MEDICAL, DENTAL OR TOILETRY PURPOSES
    • A61K31/00—Medicinal preparations containing organic active ingredients
    • A61K31/13—Amines
    • A61K31/135—Amines having aromatic rings, e.g. ketamine, nortriptyline

Landscapes

  • Health & Medical Sciences (AREA)
  • Animal Behavior & Ethology (AREA)
  • Medicinal Chemistry (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Epidemiology (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • Chemical & Material Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Low-Molecular Organic Synthesis Reactions Using Catalysts (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DE19661543372 1966-10-18 1966-10-18 Verfahren zur Herstellung von o-substituierten 3,4-Dioxyphenylalkanolaminen Pending DE1543372A1 (de)

Applications Claiming Priority (3)

Application Number Priority Date Filing Date Title
DEB0089417 1966-10-18
DEB0089476 1966-10-20
DEB0090062 1966-11-29

Publications (1)

Publication Number Publication Date
DE1543372A1 true DE1543372A1 (de) 1971-04-01

Family

ID=27209389

Family Applications (2)

Application Number Title Priority Date Filing Date
DE19661543372 Pending DE1543372A1 (de) 1966-10-18 1966-10-18 Verfahren zur Herstellung von o-substituierten 3,4-Dioxyphenylalkanolaminen
DE1543374A Expired DE1543374C3 (de) 1966-10-18 1966-10-20 3,4 Dihydroxyphenylalkanolamine und ihre Saureadditionssalze, Verfahren zu ihrer Herstellung und pharmazeutische Zubereitungen

Family Applications After (1)

Application Number Title Priority Date Filing Date
DE1543374A Expired DE1543374C3 (de) 1966-10-18 1966-10-20 3,4 Dihydroxyphenylalkanolamine und ihre Saureadditionssalze, Verfahren zu ihrer Herstellung und pharmazeutische Zubereitungen

Country Status (11)

Country Link
US (1) US3657244A (xx)
AT (3) AT288357B (xx)
BE (1) BE705312A (xx)
CH (4) CH490323A (xx)
DE (2) DE1543372A1 (xx)
DK (1) DK130070B (xx)
ES (6) ES346057A1 (xx)
FR (1) FR7338M (xx)
GB (1) GB1204195A (xx)
NL (1) NL158480B (xx)
SE (2) SE380792B (xx)

Families Citing this family (31)

* Cited by examiner, † Cited by third party
Publication number Priority date Publication date Assignee Title
US3969410A (en) * 1972-01-12 1976-07-13 Boehringer Ingelheim Gmbh 1-(2'-Alkyl-3',4'-dihydroxy-phenyl)-2-(phenylalkyl-amino)-alkanols-(1) and salts thereof
US4042713A (en) * 1966-10-18 1977-08-16 Boehringer Ingelheim Gmbh Pharmaceutical compositions containing a 1-(2-alkyl-3,4-dihydroxy-phenyl)-2-(phenylalkyl-amino)-alkanol-(1) and method of use
US4336400A (en) * 1969-04-01 1982-06-22 Sterling Drug Inc. 3-(Hydroxy or hydroxymethyl)-4-hydroxy-alpha(aminomethyl)benzyl alcohols and methods of use
US4138581A (en) * 1969-04-01 1979-02-06 Sterling Drugs Inc. 3(Hydroxy or hydroxymethyl)-4(hydroxy)-α-(aminomethyl)benzyl alcohols
DE1962497C3 (de) * 1969-12-12 1979-09-20 C.H. Boehringer Sohn, 6507 Ingelheim Naphthylalkyl- a -hydroxyphenäthyl-amine, ihre Herstellung und diese enthaltende Arzneimittel
US4147799A (en) * 1971-06-24 1979-04-03 Kyowa Hakko Kogyo Co., Ltd. Process for reducing blood pressure and blocking β-adrenergic receptor
US3868461A (en) * 1972-11-22 1975-02-25 Interx Research Corp Ester of 3,4-dihydroxy-alpha (isopropylamino) methyl benzyl alcohol, composition and anti-asthma use thereof
US3908017A (en) * 1973-04-26 1975-09-23 Interx Research Corp Sympathomimetic compositions containing an ester of -3-hydroxy-{60 -{8 (methylamino)methyl{8 benzyl alcohol and methods of use
US4046913A (en) * 1973-08-18 1977-09-06 Boehringer Ingelheim Gmbh 1-(M-alkanoyloxy-phenyl)-1-hydroxy-2-(N-lower alkyl-amino)-ethanes and salts thereof
US4192805A (en) * 1975-11-27 1980-03-11 Nicholas International Limited Process of preparing amino ethanols
US4287212A (en) * 1976-04-30 1981-09-01 American Hoechst Corporation 2-Aryl-1,2-dialkylcycloalkylamines
US4115585A (en) * 1976-05-17 1978-09-19 Instituto Luso Farmaco D'italia S.R.L. Esters of 1-(p-hydroxyphenyl)-2-(1'-methyl-2'-phenoxyethylamino)-1-propanol
US4094983A (en) * 1977-01-17 1978-06-13 Interx Research Corporation Method for reducing intraocular pressure in warm-blooded animals
US4590210A (en) * 1979-03-09 1986-05-20 Langham Maurice E Compositions for treatment of ocular hypertension
US4275074A (en) * 1979-03-09 1981-06-23 Graham J. Dobbie Catecholamine treatment of ocular hypertension
JPS55124742A (en) * 1979-03-20 1980-09-26 Kyowa Hakko Kogyo Co Ltd Novel aminoalcohol derivative
JPS6241829Y2 (xx) * 1980-03-28 1987-10-26
CY1273A (en) 1980-07-09 1985-03-08 Draco Ab 1-(dihydroxyphenyl)-2-amino-ethanol derivatives;preparation,compositions and intermediates
DE3128117A1 (de) * 1980-07-29 1982-03-11 Yamanouchi Pharmaceutical Co., Ltd., Tokyo Neue phenyl-aethylaminderivate, verfahren zu ihrer herstellung
US4472427A (en) * 1980-12-23 1984-09-18 Merck & Co., Inc. (Aralkylamino-2-OR-propoxy)heterocyclic compounds
ES502470A0 (es) * 1981-05-13 1982-04-01 Ferrer Int Procedimiento de obtencion de nuevos aminoderivados en posi-cion 1, del 1-(3',4'-metilendioxifenil)propan-2-ol
US4461914A (en) * 1983-02-01 1984-07-24 American Cyanamid Company Method for the preparation of 1-(4'-amino-3',5'-dichlorophenyl)-2-alkyl(or dialkyl)aminoethanols
LU85856A1 (fr) * 1984-04-17 1986-06-11 Glaxo Group Ltd Composes de phenethanolamine
US4699928A (en) * 1984-07-13 1987-10-13 Merrell Dow Pharmaceuticals Inc. Fluoroallylamine derivatives
US4843160A (en) * 1984-10-01 1989-06-27 The Dow Chemical Company Preparation of alpha-aminoalkylphenols
US5068432A (en) * 1988-03-30 1991-11-26 Aldrich Chemical Company, Inc. Process for producing optically pure 2-phenoxyphenylalkylamines
JPH02124884A (ja) * 1988-07-08 1990-05-14 Zhongguo Yixuekexueyuan Yaowo Yanjiusuo Ｎ―置換アミド誘導体
DE10246374A1 (de) * 2002-10-04 2004-04-15 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Betamimetika mit verlängerter Wirkungsdauer, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
US6951888B2 (en) 2002-10-04 2005-10-04 Boehringer Ingelheim Pharma Gmbh & Co. Kg Betamimetics with a prolonged duration of activity, processes for preparing them, and their use as pharmaceutical compositions
DE10253220A1 (de) * 2002-11-15 2004-05-27 Boehringer Ingelheim Pharma Gmbh & Co. Kg Neue Dihydroxy-Methyl-Phenyl-Derivate, Verfahren zu deren Herstellung und deren Verwendung als Arzneimittel
CN110743544B (zh) * 2019-11-07 2023-02-24 西安凯立新材料股份有限公司 一种苯乙酮选择加氢制备α-苯乙醇用钯炭催化剂及其制备方法与应用

Also Published As

Publication number Publication date
SE380792B (sv) 1975-11-17
AT288357B (de) 1971-03-10
GB1204195A (en) 1970-09-03
CH548365A (de) 1974-04-30
ES346057A1 (es) 1969-03-16
NL6714161A (xx) 1968-04-19
AT285582B (de) 1970-11-10
ES360963A1 (es) 1970-11-16
NL158480B (nl) 1978-11-15
ES360965A1 (es) 1970-11-16
ES360964A1 (es) 1970-10-16
CH523219A (de) 1972-05-31
CH507200A (de) 1971-05-15
DE1543374C3 (de) 1973-10-04
ES360962A1 (es) 1970-11-16
US3657244A (en) 1972-04-18
DK130070B (da) 1974-12-16
AT288358B (de) 1971-03-10
ES360961A1 (es) 1970-11-16
BE705312A (xx) 1968-04-18
DE1543374A1 (de) 1972-04-20
DK130070C (xx) 1975-05-26
SE368196B (xx) 1974-06-24
CH490323A (de) 1970-05-15
DE1543374B2 (de) 1973-02-22
FR7338M (xx) 1969-10-13

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