DD140354A5 - Verfahren zur herstellung von 4-hydroxy-2h-1,2-benzothiazin-3-carboxamid-1,1-dioxid - Google Patents

Verfahren zur herstellung von 4-hydroxy-2h-1,2-benzothiazin-3-carboxamid-1,1-dioxid Download PDF

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Publication number
DD140354A5
DD140354A5 DD78209763A DD20976378A DD140354A5 DD 140354 A5 DD140354 A5 DD 140354A5 DD 78209763 A DD78209763 A DD 78209763A DD 20976378 A DD20976378 A DD 20976378A DD 140354 A5 DD140354 A5 DD 140354A5
Authority
DD
German Democratic Republic
Prior art keywords
methyl
group
hydroxy
dioxide
general formula
Prior art date
Application number
DD78209763A
Other languages
German (de)
English (en)
Inventor
Guenter Trummlitz
Wolfhard Engel
Ernst Seeger
Guenter Engelhardt
Original Assignee
Thomae Gmbh Dr K
Priority date (The priority date is an assumption and is not a legal conclusion. Google has not performed a legal analysis and makes no representation as to the accuracy of the date listed.)
Filing date
Publication date
Application filed by Thomae Gmbh Dr K filed Critical Thomae Gmbh Dr K
Publication of DD140354A5 publication Critical patent/DD140354A5/de

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Classifications

    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D275/00—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings
    • C07D275/04—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems
    • C07D275/06—Heterocyclic compounds containing 1,2-thiazole or hydrogenated 1,2-thiazole rings condensed with carbocyclic rings or ring systems with hetero atoms directly attached to the ring sulfur atom
    • A—HUMAN NECESSITIES
    • A61—MEDICAL OR VETERINARY SCIENCE; HYGIENE
    • A61P—SPECIFIC THERAPEUTIC ACTIVITY OF CHEMICAL COMPOUNDS OR MEDICINAL PREPARATIONS
    • A61P29/00—Non-central analgesic, antipyretic or antiinflammatory agents, e.g. antirheumatic agents; Non-steroidal antiinflammatory drugs [NSAID]
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D279/00—Heterocyclic compounds containing six-membered rings having one nitrogen atom and one sulfur atom as the only ring hetero atoms
    • C07D279/02—1,2-Thiazines; Hydrogenated 1,2-thiazines
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D417/00—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00
    • C07D417/02—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings
    • C07D417/12—Heterocyclic compounds containing two or more hetero rings, at least one ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for by group C07D415/00 containing two hetero rings linked by a chain containing hetero atoms as chain links
    • C—CHEMISTRY; METALLURGY
    • C07—ORGANIC CHEMISTRY
    • C07D—HETEROCYCLIC COMPOUNDS
    • C07D513/00—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00
    • C07D513/12—Heterocyclic compounds containing in the condensed system at least one hetero ring having nitrogen and sulfur atoms as the only ring hetero atoms, not provided for in groups C07D463/00, C07D477/00 or C07D499/00 - C07D507/00 in which the condensed system contains three hetero rings
    • C07D513/14—Ortho-condensed systems

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  • Chemical & Material Sciences (AREA)
  • Organic Chemistry (AREA)
  • Health & Medical Sciences (AREA)
  • Life Sciences & Earth Sciences (AREA)
  • General Health & Medical Sciences (AREA)
  • Chemical Kinetics & Catalysis (AREA)
  • General Chemical & Material Sciences (AREA)
  • Medicinal Chemistry (AREA)
  • Nuclear Medicine, Radiotherapy & Molecular Imaging (AREA)
  • Pharmacology & Pharmacy (AREA)
  • Pain & Pain Management (AREA)
  • Animal Behavior & Ethology (AREA)
  • Rheumatology (AREA)
  • Public Health (AREA)
  • Veterinary Medicine (AREA)
  • Pharmaceuticals Containing Other Organic And Inorganic Compounds (AREA)
  • Nitrogen- Or Sulfur-Containing Heterocyclic Ring Compounds With Rings Of Six Or More Members (AREA)
  • Plural Heterocyclic Compounds (AREA)
  • Heterocyclic Carbon Compounds Containing A Hetero Ring Having Nitrogen And Oxygen As The Only Ring Hetero Atoms (AREA)
  • Organic Low-Molecular-Weight Compounds And Preparation Thereof (AREA)
  • Acyclic And Carbocyclic Compounds In Medicinal Compositions (AREA)
DD78209763A 1977-12-16 1978-12-14 Verfahren zur herstellung von 4-hydroxy-2h-1,2-benzothiazin-3-carboxamid-1,1-dioxid DD140354A5 (de)

Applications Claiming Priority (1)

Application Number Priority Date Filing Date Title
DE19772756113 DE2756113A1 (de) 1977-12-16 1977-12-16 Neue 4-hydroxy-2h-1,2-benzothiazin- 3-carboxamid-1,1-dioxide, verfahren zu ihrer herstellung und diese enthaltende arzneimittel

Publications (1)

Publication Number Publication Date
DD140354A5 true DD140354A5 (de) 1980-02-27

Family

ID=6026297

Family Applications (1)

Application Number Title Priority Date Filing Date
DD78209763A DD140354A5 (de) 1977-12-16 1978-12-14 Verfahren zur herstellung von 4-hydroxy-2h-1,2-benzothiazin-3-carboxamid-1,1-dioxid

Country Status (27)

Country Link
US (1) US4233299A (fi)
EP (1) EP0002482B1 (fi)
JP (1) JPS5492976A (fi)
AT (1) AT365589B (fi)
AU (1) AU522538B2 (fi)
BG (2) BG33286A3 (fi)
CA (1) CA1102802A (fi)
CS (2) CS202515B2 (fi)
DD (1) DD140354A5 (fi)
DE (2) DE2756113A1 (fi)
DK (1) DK149344C (fi)
ES (2) ES475677A1 (fi)
FI (1) FI61896C (fi)
GR (1) GR65626B (fi)
HU (1) HU175846B (fi)
IE (1) IE48042B1 (fi)
IL (1) IL56206A (fi)
LU (1) LU88557I2 (fi)
MX (1) MX9202949A (fi)
NL (1) NL940002I2 (fi)
NO (2) NO150203C (fi)
NZ (1) NZ189186A (fi)
PL (1) PL115756B1 (fi)
PT (1) PT68915A (fi)
RO (1) RO75792A (fi)
SU (1) SU841588A3 (fi)
YU (1) YU294978A (fi)

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US4074048A (en) * 1976-05-10 1978-02-14 Warner-Lambert Company Process for the preparation of 4-hydroxy-2H-1,2-benzothiazine-3-carboxamide 1,1-dioxides
US4100347A (en) * 1976-06-10 1978-07-11 Pfizer Inc. 3,4-Dihydro-2-methyl-4-oxo-2H-1,2-benzothiazine-3-carboxylic acid-1,1-dioxide

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ATA863078A (de) 1981-06-15
DK562078A (da) 1979-06-17
NO150203B (no) 1984-05-28
EP0002482B1 (de) 1981-01-07
DE2756113A1 (de) 1979-06-21
CA1102802A (en) 1981-06-09
YU294978A (en) 1982-10-31
NO1997002I1 (no) 1997-01-14
FI61896B (fi) 1982-06-30
HU175846B (hu) 1980-10-28
NL940002I1 (nl) 1994-03-16
DK149344B (da) 1986-05-12
JPS5492976A (en) 1979-07-23
IL56206A0 (en) 1979-03-12
ES8802454A3 (es) 1988-06-16
IE48042B1 (en) 1984-09-05
CS202515B2 (en) 1981-01-30
NL940002I2 (nl) 1997-05-01
BG33286A3 (en) 1983-01-14
ES550377A0 (es) 1988-06-16
NZ189186A (en) 1981-03-16
BG60475B2 (bg) 1995-04-28
LU88557I2 (fr) 1995-03-21
FI783867A (fi) 1979-06-17
DE2860445D1 (en) 1981-02-26
AU4253078A (en) 1979-06-21
FI61896C (fi) 1982-10-11
US4233299A (en) 1980-11-11
IL56206A (en) 1982-04-30
AU522538B2 (en) 1982-06-10
PL211753A1 (pl) 1979-08-13
NO784231L (no) 1979-06-19
GR65626B (en) 1980-10-15
JPS6324997B2 (fi) 1988-05-23
IE782482L (en) 1979-06-16
SU841588A3 (ru) 1981-06-23
PT68915A (de) 1979-01-01
DK149344C (da) 1986-10-13
NO150203C (no) 1984-09-05
PL115756B1 (en) 1981-04-30
EP0002482A1 (de) 1979-06-27
RO75792A (ro) 1981-02-28
MX9202949A (es) 1992-07-01
AT365589B (de) 1982-01-25
CS410091A3 (en) 1992-06-17
ES475677A1 (es) 1979-04-16

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